Report error Found 75 Enz. Inhib. hit(s) with all data for entry = 50018029
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Anhui University of Chinese Medicine
Curated by ChEMBL
Anhui University of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Inhibition of PI3Kdelta (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Anhui University of Chinese Medicine
Curated by ChEMBL
Anhui University of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 2.30nMAssay Description:Inhibition of PI3Kdelta (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Anhui University of Chinese Medicine
Curated by ChEMBL
Anhui University of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 6.10nMAssay Description:Inhibition of PI3Kdelta (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Anhui University of Chinese Medicine
Curated by ChEMBL
Anhui University of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 6.80nMAssay Description:Inhibition of PI3Kdelta (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Anhui University of Chinese Medicine
Curated by ChEMBL
Anhui University of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 6.90nMAssay Description:Inhibition of PI3Kdelta (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Anhui University of Chinese Medicine
Curated by ChEMBL
Anhui University of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of PI3Kdelta (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.40nMAssay Description:Inhibition of HDAC6 (unknown origin) measured by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of HDAC6 (unknown origin) measured by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of HDAC1 (unknown origin) measured by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of HDAC6 (unknown origin) measured by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of HDAC6 (unknown origin) measured by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of HDAC6 (unknown origin) measured by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of HDAC1 (unknown origin) measured by fluorescence based assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Anhui University of Chinese Medicine
Curated by ChEMBL
Anhui University of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of PI3Kdelta (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of HDAC6 (unknown origin) measured by fluorescence based assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Anhui University of Chinese Medicine
Curated by ChEMBL
Anhui University of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of PI3Kdelta (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Anhui University of Chinese Medicine
Curated by ChEMBL
Anhui University of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of PI3Kdelta (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Anhui University of Chinese Medicine
Curated by ChEMBL
Anhui University of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of PI3Kdelta (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Anhui University of Chinese Medicine
Curated by ChEMBL
Anhui University of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of PI3Kdelta (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of HDAC6 (unknown origin) measured by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of HDAC6 (unknown origin) measured by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Inhibition of HDAC6 (unknown origin) measured by fluorescence based assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Human)
Anhui University of Chinese Medicine
Curated by ChEMBL
Anhui University of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Inhibition of PI3Kgamma (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibition of HDAC6 (unknown origin) measured by fluorescence based assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Anhui University of Chinese Medicine
Curated by ChEMBL
Anhui University of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of PI3Kdelta (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Anhui University of Chinese Medicine
Curated by ChEMBL
Anhui University of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Inhibition of PI3Kdelta (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:Inhibition of HDAC6 (unknown origin) measured by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Inhibition of HDAC6 (unknown origin) measured by fluorescence based assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Anhui University of Chinese Medicine
Curated by ChEMBL
Anhui University of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Inhibition of PI3Kdelta (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Anhui University of Chinese Medicine
Curated by ChEMBL
Anhui University of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Inhibition of PI3Kdelta (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
Affinity DataIC50: 43nMAssay Description:Inhibition of HDAC6 (unknown origin) measured by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:Inhibition of HDAC6 (unknown origin) measured by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:Inhibition of HDAC6 (unknown origin) measured by fluorescence based assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Human)
Anhui University of Chinese Medicine
Curated by ChEMBL
Anhui University of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 51nMAssay Description:Inhibition of PI3Kgamma (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
Affinity DataIC50: 66nMAssay Description:Inhibition of HDAC6 (unknown origin) measured by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 67nMAssay Description:Inhibition of HDAC6 (unknown origin) measured by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 72nMAssay Description:Inhibition of HDAC1 (unknown origin) measured by fluorescence based assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Anhui University of Chinese Medicine
Curated by ChEMBL
Anhui University of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 75nMAssay Description:Inhibition of PI3Kdelta (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
Affinity DataIC50: 82nMAssay Description:Inhibition of HDAC1 (unknown origin) measured by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 85nMAssay Description:Inhibition of HDAC1 (unknown origin) measured by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 87nMAssay Description:Inhibition of HDAC6 (unknown origin) measured by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 88nMAssay Description:Inhibition of HDAC1 (unknown origin) measured by fluorescence based assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Anhui University of Chinese Medicine
Curated by ChEMBL
Anhui University of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 99nMAssay Description:Inhibition of PI3Kdelta (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
Affinity DataIC50: 102nMAssay Description:Inhibition of HDAC1 (unknown origin) measured by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 111nMAssay Description:Inhibition of HDAC1 (unknown origin) measured by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 121nMAssay Description:Inhibition of HDAC6 (unknown origin) measured by fluorescence based assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Anhui University of Chinese Medicine
Curated by ChEMBL
Anhui University of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 136nMAssay Description:Inhibition of PI3Kdelta (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
Affinity DataIC50: 161nMAssay Description:Inhibition of HDAC8 (unknown origin) measured by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 168nMAssay Description:Inhibition of HDAC6 (unknown origin) measured by fluorescence based assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Anhui University of Chinese Medicine
Curated by ChEMBL
Anhui University of Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 169nMAssay Description:Inhibition of PI3Kalpha (unknown origin) measured by ADP-Glo assayMore data for this Ligand-Target Pair
