Compile Data Set for Download or QSAR
Report error Found 64 Enz. Inhib. hit(s) with all data for entry = 50016007
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591380(CHEMBL5180611 | US20240190828, Compound 34)
Affinity DataIC50: 160nMAssay Description:Inhibition of biotinylated histone H3K14 (1 to 20 residues) peptide binding to His6-tagged recombinant human PBRM1 BD2 transfected in Escherichia col...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50184981(CHEMBL3823055 | US20240190828, Compound 7)
Affinity DataIC50: 200nMAssay Description:Inhibition of biotinylated histone H3K14 (1 to 20 residues) peptide binding to His6-tagged recombinant human PBRM1 BD2 transfected in Escherichia col...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591362(CHEMBL5195502 | US20240190828, Compound 15)
Affinity DataIC50: 200nMAssay Description:Inhibition of biotinylated histone H3K14 (1 to 20 residues) peptide binding to His6-tagged recombinant human PBRM1 BD2 transfected in Escherichia col...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591371(CHEMBL5187356 | US20240190828, Compound 25)
Affinity DataIC50: 220nMAssay Description:Inhibition of biotinylated histone H3K14 (1 to 20 residues) peptide binding to His6-tagged recombinant human PBRM1 BD2 transfected in Escherichia col...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591363(CHEMBL5170275 | US20240190828, Compound 16)
Affinity DataIC50: 260nMAssay Description:Inhibition of biotinylated histone H3K14 (1 to 20 residues) peptide binding to His6-tagged recombinant human PBRM1 BD2 transfected in Escherichia col...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591372(CHEMBL5207236 | US20240190828, Compound 26)
Affinity DataIC50: 290nMAssay Description:Inhibition of biotinylated histone H3K14 (1 to 20 residues) peptide binding to His6-tagged recombinant human PBRM1 BD2 transfected in Escherichia col...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591381(CHEMBL5184118)
Affinity DataIC50: 290nMAssay Description:Inhibition of biotinylated histone H3K14 (1 to 20 residues) peptide binding to His6-tagged recombinant human PBRM1 BD2 transfected in Escherichia col...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50184981(CHEMBL3823055 | US20240190828, Compound 7)
Affinity DataKd:  350nMAssay Description:Binding affinity to His-TEV-tagged human PBRM1 BD5 transfected in Escherichia coli BL21 (DE3) assessed as dissociation constant at 30 uM by ITC analy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591370(CHEMBL5185774 | US20240190828, Compound 24)
Affinity DataIC50: 430nMAssay Description:Inhibition of biotinylated histone H3K14 (1 to 20 residues) peptide binding to His6-tagged recombinant human PBRM1 BD2 transfected in Escherichia col...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50184981(CHEMBL3823055 | US20240190828, Compound 7)
Affinity DataKd:  700nMAssay Description:Binding affinity to His-TEV-tagged recombinant human PBRM1 BD2 transfected in Escherichia coli BL21 (DE3) assessed as dissociation constant at 30 uM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591367(CHEMBL5195542 | US20240190828, Compound 21)
Affinity DataIC50: 860nMAssay Description:Inhibition of biotinylated histone H3K14 (1 to 20 residues) peptide binding to His6-tagged recombinant human PBRM1 BD2 transfected in Escherichia col...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591364(CHEMBL5194300 | US20240190828, Compound 17)
Affinity DataIC50: 870nMAssay Description:Inhibition of biotinylated histone H3K14 (1 to 20 residues) peptide binding to His6-tagged recombinant human PBRM1 BD2 transfected in Escherichia col...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591358(CHEMBL5204703 | US20240190828, Compound 11)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of biotinylated histone H3K14 (1 to 20 residues) peptide binding to His6-tagged recombinant human PBRM1 BD2 transfected in Escherichia col...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591359(CHEMBL5170175 | US20240190828, Compound 12)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of biotinylated histone H3K14 (1 to 20 residues) peptide binding to His6-tagged recombinant human PBRM1 BD2 transfected in Escherichia col...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591368(CHEMBL5181215 | US20240190828, Compound 22)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of biotinylated histone H3K14 (1 to 20 residues) peptide binding to His6-tagged recombinant human PBRM1 BD2 transfected in Escherichia col...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591379(CHEMBL5176658 | US20240190828, Compound 33)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of biotinylated histone H3K14 (1 to 20 residues) peptide binding to His6-tagged recombinant human PBRM1 BD2 transfected in Escherichia col...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591363(CHEMBL5170275 | US20240190828, Compound 16)
Affinity DataKd:  1.50E+3nMAssay Description:Binding affinity to His-TEV-tagged recombinant human PBRM1 BD2 transfected in Escherichia coli BL21 (DE3) assessed as dissociation constant at 30 uM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591360(CHEMBL5205087 | US20240190828, Compound 13)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of biotinylated histone H3K14 (1 to 20 residues) peptide binding to His6-tagged recombinant human PBRM1 BD2 transfected in Escherichia col...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591361(CHEMBL5197320 | US20240190828, Compound 14)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of biotinylated histone H3K14 (1 to 20 residues) peptide binding to His6-tagged recombinant human PBRM1 BD2 transfected in Escherichia col...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591365(CHEMBL5171156 | US20240190828, Compound 18)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of biotinylated histone H3K14 (1 to 20 residues) peptide binding to His6-tagged recombinant human PBRM1 BD2 transfected in Escherichia col...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591357(CHEMBL5205514 | US20240190828, Compound 8)
Affinity DataKd:  3.30E+3nMAssay Description:Binding affinity to His-TEV-tagged human PBRM1 BD5 transfected in Escherichia coli BL21 (DE3) assessed as dissociation constant at 30 uM by ITC analy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591363(CHEMBL5170275 | US20240190828, Compound 16)
Affinity DataKd:  3.90E+3nMAssay Description:Binding affinity to His-TEV-tagged human PBRM1 BD5 transfected in Escherichia coli BL21 (DE3) assessed as dissociation constant at 30 uM by ITC analy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591380(CHEMBL5180611 | US20240190828, Compound 34)
Affinity DataKd:  4.40E+3nMAssay Description:Binding affinity to His-TEV-tagged recombinant human PBRM1 BD2 transfected in Escherichia coli BL21 (DE3) assessed as dissociation constant at 30 uM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetTranscription activator BRG1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50184981(CHEMBL3823055 | US20240190828, Compound 7)
Affinity DataKd:  5.00E+3nMAssay Description:Binding affinity to N-terminal His-TEV-tagged human SMARCA4 transfected in Escherichia coli BL21 (DE3) assessed as dissociation constant at 30 uM by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591362(CHEMBL5195502 | US20240190828, Compound 15)
Affinity DataKd:  5.50E+3nMAssay Description:Binding affinity to His-TEV-tagged recombinant human PBRM1 BD2 transfected in Escherichia coli BL21 (DE3) assessed as dissociation constant at 30 uM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591378(CHEMBL5178860 | US20240190828, Compound 32)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of biotinylated histone H3K14 (1 to 20 residues) peptide binding to His6-tagged recombinant human PBRM1 BD2 transfected in Escherichia col...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591366(CHEMBL5203878 | US20240190828, Compound 20)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of biotinylated histone H3K14 (1 to 20 residues) peptide binding to His6-tagged recombinant human PBRM1 BD2 transfected in Escherichia col...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591357(CHEMBL5205514 | US20240190828, Compound 8)
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of biotinylated histone H3K14 (1 to 20 residues) peptide binding to His6-tagged recombinant human PBRM1 BD2 transfected in Escherichia col...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591357(CHEMBL5205514 | US20240190828, Compound 8)
Affinity DataKd:  6.90E+3nMAssay Description:Binding affinity to His-TEV-tagged recombinant human PBRM1 BD2 transfected in Escherichia coli BL21 (DE3) assessed as dissociation constant at 30 uM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591383(CHEMBL5184333 | US20240190828, Compound 36)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of biotinylated histone H3K14 (1 to 20 residues) peptide binding to His6-tagged recombinant human PBRM1 BD2 transfected in Escherichia col...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50184981(CHEMBL3823055 | US20240190828, Compound 7)
Affinity DataKd:  8.10E+3nMAssay Description:Binding affinity to N-terminal His6-TEV-tagged human SMARCA2B transfected in Escherichia coli BL21 (DE3) assessed as dissociation constant at 30 uM b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591358(CHEMBL5204703 | US20240190828, Compound 11)
Affinity DataKd:  9.30E+3nMAssay Description:Binding affinity to His-TEV-tagged recombinant human PBRM1 BD2 transfected in Escherichia coli BL21 (DE3) assessed as dissociation constant at 30 uM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591358(CHEMBL5204703 | US20240190828, Compound 11)
Affinity DataKd:  1.01E+4nMAssay Description:Binding affinity to His-TEV-tagged human PBRM1 BD5 transfected in Escherichia coli BL21 (DE3) assessed as dissociation constant at 30 uM by ITC analy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591362(CHEMBL5195502 | US20240190828, Compound 15)
Affinity DataKd:  1.11E+4nMAssay Description:Binding affinity to His-TEV-tagged human PBRM1 BD5 transfected in Escherichia coli BL21 (DE3) assessed as dissociation constant at 30 uM by ITC analy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591346(CHEMBL5188924 | US20240190828, Compound 5)
Affinity DataKd:  1.59E+4nMAssay Description:Binding affinity to N-terminal His6-TEV-tagged human SMARCA2B transfected in Escherichia coli BL21 (DE3) assessed as dissociation constant at 30 uM b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591374(CHEMBL5172472 | US20240190828, Compound 28)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of biotinylated histone H3K14 (1 to 20 residues) peptide binding to His6-tagged recombinant human PBRM1 BD2 transfected in Escherichia col...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591346(CHEMBL5188924 | US20240190828, Compound 5)
Affinity DataKd:  1.84E+4nMAssay Description:Binding affinity to His-TEV-tagged recombinant human PBRM1 BD2 transfected in Escherichia coli BL21 (DE3) assessed as dissociation constant at 30 uM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591358(CHEMBL5204703 | US20240190828, Compound 11)
Affinity DataKd:  1.84E+4nMAssay Description:Binding affinity to N-terminal His6-TEV-tagged human SMARCA2B transfected in Escherichia coli BL21 (DE3) assessed as dissociation constant at 30 uM b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591380(CHEMBL5180611 | US20240190828, Compound 34)
Affinity DataKd:  2.50E+4nMAssay Description:Binding affinity to His-TEV-tagged human PBRM1 BD5 transfected in Escherichia coli BL21 (DE3) assessed as dissociation constant at 30 uM by ITC analy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591382(CHEMBL5171944 | US20240190828, Compound 35)
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of biotinylated histone H3K14 (1 to 20 residues) peptide binding to His6-tagged recombinant human PBRM1 BD2 transfected in Escherichia col...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591346(CHEMBL5188924 | US20240190828, Compound 5)
Affinity DataKd:  4.53E+4nMAssay Description:Binding affinity to 15N-labeled recombinant human PBRM1 BD2 transfected in Escherichia coli BL21 (DE3) assessed as 1H/13N chemical shift perturbation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50104297(CHEMBL3594130 | US20240190828, Compound 19)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of biotinylated histone H3K14 (1 to 20 residues) peptide binding to His6-tagged recombinant human PBRM1 BD2 transfected in Escherichia col...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetTranscription activator BRG1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591358(CHEMBL5204703 | US20240190828, Compound 11)
Affinity DataKd:  6.90E+4nMAssay Description:Binding affinity to N-terminal His-TEV-tagged human SMARCA4 transfected in Escherichia coli BL21 (DE3) assessed as dissociation constant at 30 uM by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591369(CHEMBL5186537 | US20240190828, Compound 23)
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibition of biotinylated histone H3K14 (1 to 20 residues) peptide binding to His6-tagged recombinant human PBRM1 BD2 transfected in Escherichia col...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591377(CHEMBL5200761 | US20240190828, Compound 31)
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibition of biotinylated histone H3K14 (1 to 20 residues) peptide binding to His6-tagged recombinant human PBRM1 BD2 transfected in Escherichia col...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591347(CHEMBL541514 | US20240190828, Compound 6)
Affinity DataKd:  7.90E+4nMAssay Description:Binding affinity to 15N-labeled recombinant human PBRM1 BD2 transfected in Escherichia coli BL21 (DE3) assessed as 1H/13N chemical shift perturbation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591376(CHEMBL5196748 | US20240190828, Compound 30)
Affinity DataIC50: 8.99E+4nMAssay Description:Inhibition of biotinylated histone H3K14 (1 to 20 residues) peptide binding to His6-tagged recombinant human PBRM1 BD2 transfected in Escherichia col...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591373(CHEMBL5171878 | US20240190828, Compound 27)
Affinity DataIC50: 1.19E+5nMAssay Description:Inhibition of biotinylated histone H3K14 (1 to 20 residues) peptide binding to His6-tagged recombinant human PBRM1 BD2 transfected in Escherichia col...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetProtein polybromo-1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591347(CHEMBL541514 | US20240190828, Compound 6)
Affinity DataIC50: 1.27E+5nMAssay Description:Inhibition of biotinylated histone H3K14 (1 to 20 residues) peptide binding to His6-tagged recombinant human PBRM1 BD2 transfected in Escherichia col...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetTranscription activator BRG1(Human)
Medical College of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50591346(CHEMBL5188924 | US20240190828, Compound 5)
Affinity DataKd:  1.42E+5nMAssay Description:Binding affinity to N-terminal His-TEV-tagged human SMARCA4 transfected in Escherichia coli BL21 (DE3) assessed as dissociation constant at 30 uM by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
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