Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50018797
TargetHistone deacetylase 6(Human)
First Affiliated Hospital of Gannan Medical University
Curated by ChEMBL
First Affiliated Hospital of Gannan Medical University
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Inhibition of human HDAC6More data for this Ligand-Target Pair
TargetHistone deacetylase 3(Human)
First Affiliated Hospital of Gannan Medical University
Curated by ChEMBL
First Affiliated Hospital of Gannan Medical University
Curated by ChEMBL
Affinity DataIC50: 159nMAssay Description:Inhibition of human HDAC3More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Human)
First Affiliated Hospital of Gannan Medical University
Curated by ChEMBL
First Affiliated Hospital of Gannan Medical University
Curated by ChEMBL
Affinity DataIC50: 174nMAssay Description:Inhibition of human HDAC1More data for this Ligand-Target Pair
TargetHistone deacetylase 2(Human)
First Affiliated Hospital of Gannan Medical University
Curated by ChEMBL
First Affiliated Hospital of Gannan Medical University
Curated by ChEMBL
Affinity DataIC50: 248nMAssay Description:Inhibition of human HDAC2More data for this Ligand-Target Pair
TargetProtein fem-1 homolog B(Human)
First Affiliated Hospital of Gannan Medical University
Curated by ChEMBL
First Affiliated Hospital of Gannan Medical University
Curated by ChEMBL
Affinity DataEC50: 250nMAssay Description:Protac activity at FEM1B/BRD4 in human HEK293T cells assessed as degradation of BRD4 incubated for 8 hrs by Western blot analysisMore data for this Ligand-Target Pair
TargetHistone deacetylase 3(Human)
First Affiliated Hospital of Gannan Medical University
Curated by ChEMBL
First Affiliated Hospital of Gannan Medical University
Curated by ChEMBL
Affinity DataIC50: 560nMAssay Description:Inhibition of recombinant human HDAC3 expressed in BTI-TN-5B1-4 insect cells using Ac-Lys-Tyr-Lys(epsilon-acetyl)-AMC as substrate incubated for 24 h...More data for this Ligand-Target Pair


