Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50020722
TargetCollagen alpha-1(I) chain(Homo sapiens)
Chinese Academy of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Chinese Academy of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: 7.80nMAssay Description:Inhibition of COL1A1 (unknown origin) expressed in human LX2 cells incubated for 48 hrs by Bright-Glo luciferase assayMore data for this Ligand-Target Pair
TargetCollagen alpha-1(I) chain(Homo sapiens)
Chinese Academy of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Chinese Academy of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: 8.20nMAssay Description:Inhibition of COL1A1 (unknown origin) expressed in human LX2 cells incubated for 48 hrs by Bright-Glo luciferase assayMore data for this Ligand-Target Pair
TargetCollagen alpha-1(I) chain(Homo sapiens)
Chinese Academy of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Chinese Academy of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of COL1A1 (unknown origin) expressed in human LX2 cells incubated for 48 hrs by Bright-Glo luciferase assayMore data for this Ligand-Target Pair
TargetCollagen alpha-1(I) chain(Homo sapiens)
Chinese Academy of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Chinese Academy of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of COL1A1 (unknown origin) expressed in human LX2 cells incubated for 48 hrs by Bright-Glo luciferase assayMore data for this Ligand-Target Pair
TargetCollagen alpha-1(I) chain(Homo sapiens)
Chinese Academy of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Chinese Academy of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of COL1A1 (unknown origin) expressed in human LX2 cells incubated for 48 hrs by Bright-Glo luciferase assayMore data for this Ligand-Target Pair
TargetCollagen alpha-1(I) chain(Homo sapiens)
Chinese Academy of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Chinese Academy of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of COL1A1 (unknown origin) expressed in human LX2 cells incubated for 48 hrs by Bright-Glo luciferase assayMore data for this Ligand-Target Pair
TargetCollagen alpha-1(I) chain(Homo sapiens)
Chinese Academy of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Chinese Academy of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of COL1A1 (unknown origin) expressed in human LX2 cells incubated for 48 hrs by Bright-Glo luciferase assayMore data for this Ligand-Target Pair
TargetBile acid receptor(Human)
Chinese Academy of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Chinese Academy of Medical Sciences & Peking Union Medical College
Curated by ChEMBL
Affinity DataKd: 84nMAssay Description:Binding affinity to FXR (unknown origin) assessed as dissociation constant by surface plasmon resonance assayMore data for this Ligand-Target Pair






