Compile Data Set for Download or QSAR
Report error Found 54 Enz. Inhib. hit(s) with all data for entry = 50015704
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to MAP4K5 (unknown origin) assessed as dissociation constant by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataKd:  0.260nMAssay Description:Binding affinity to AXL (unknown origin) assessed as dissociation constant by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataKd:  29nMAssay Description:Binding affinity to CSF1R (unknown origin) assessed as dissociation constant by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to DDR1 (unknown origin) assessed as dissociation constant by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetEphrin type-B receptor 6(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to EPHB6 (unknown origin) assessed as dissociation constant by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataKd:  14nMAssay Description:Binding affinity to FLT1 (unknown origin) assessed as dissociation constant by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataKd:  2.5nMAssay Description:Binding affinity to FLT3 (unknown origin) assessed as dissociation constant by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetVascular endothelial growth factor receptor 3(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataKd:  19nMAssay Description:Binding affinity to FLT4 (unknown origin) assessed as dissociation constant by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataKd:  2.60nMAssay Description:Binding affinity to KIT (unknown origin) assessed as dissociation constant by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase 10(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataKd:  880nMAssay Description:Binding affinity to LOK (unknown origin) assessed as dissociation constant by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase Mer(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataKd:  560nMAssay Description:Binding affinity to MERTK (unknown origin) assessed as dissociation constant by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetHepatocyte growth factor receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to MET (unknown origin) assessed as dissociation constant by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetMacrophage-stimulating protein receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to MSTIR (unknown origin) assessed as dissociation constant by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor beta(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataKd:  2.30nMAssay Description:Binding affinity to PDGFRB (unknown origin) assessed as dissociation constant by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataKd:  600nMAssay Description:Binding affinity to RET (unknown origin) assessed as dissociation constant by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase receptor Tie-1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataKd:  0.740nMAssay Description:Binding affinity to TIE1 (unknown origin) assessed as dissociation constant by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetAngiopoietin-1 receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataKd:  950nMAssay Description:Binding affinity to TIE2 (unknown origin) assessed as dissociation constant by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50021574(CHEBI:72317 | CABOZANTINIB | BMS-907351 | Cometriq...)
Affinity DataIC50: 0.0350nMAssay Description:Inhibition of recombinant human full length KDR using poly(Glu, Tyr) as substrate by alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetHepatocyte growth factor receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50021574(CHEBI:72317 | CABOZANTINIB | BMS-907351 | Cometriq...)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of recombinant human full length MET using poly(Glu, Tyr) as substrate by alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of recombinant AXL (unknown origin) using poly (Glu,Tyr) 4:1 as substrate incubated for 60 mins in presence of ATP by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588795(CHEMBL5184891)
Affinity DataIC50: 2.90nMAssay Description:Inhibition of recombinant AXL (unknown origin) using poly (Glu,Tyr) 4:1 as substrate incubated for 60 mins in presence of ATP by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588793(CHEMBL5193925)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of recombinant AXL (unknown origin) using poly (Glu,Tyr) 4:1 as substrate incubated for 60 mins in presence of ATP by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588794(CHEMBL5208952)
Affinity DataIC50: 5.60nMAssay Description:Inhibition of recombinant AXL (unknown origin) using poly (Glu,Tyr) 4:1 as substrate incubated for 60 mins in presence of ATP by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50021574(CHEBI:72317 | CABOZANTINIB | BMS-907351 | Cometriq...)
Affinity DataIC50: 7nMAssay Description:Inhibition of AXL (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588791(CHEMBL5206835)
Affinity DataIC50: 7.80nMAssay Description:Inhibition of recombinant AXL (unknown origin) using poly (Glu,Tyr) 4:1 as substrate incubated for 60 mins in presence of ATP by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588792(CHEMBL5198669)
Affinity DataIC50: 8.60nMAssay Description:Inhibition of recombinant AXL (unknown origin) using poly (Glu,Tyr) 4:1 as substrate incubated for 60 mins in presence of ATP by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50571423(CHEMBL4857746)
Affinity DataIC50: 9.90nMAssay Description:Inhibition of AXL in human HeLa cells incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588780(CHEMBL5174389)
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant AXL (unknown origin) using poly (Glu,Tyr) 4:1 as substrate incubated for 60 mins in presence of ATP by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588782(CHEMBL5184070)
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant AXL (unknown origin) using poly (Glu,Tyr) 4:1 as substrate incubated for 60 mins in presence of ATP by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588781(CHEMBL5188331)
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant AXL (unknown origin) using poly (Glu,Tyr) 4:1 as substrate incubated for 60 mins in presence of ATP by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50571423(CHEMBL4857746)
Affinity DataIC50: 14nMAssay Description:Inhibition of AXL (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588775(CHEMBL5189364)
Affinity DataIC50: 23nMAssay Description:Inhibition of recombinant AXL (unknown origin) using poly (Glu,Tyr) 4:1 as substrate incubated for 60 mins in presence of ATP by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588773(CHEMBL5206823)
Affinity DataIC50: 25nMAssay Description:Inhibition of recombinant AXL (unknown origin) using poly (Glu,Tyr) 4:1 as substrate incubated for 60 mins in presence of ATP by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataIC50: 27nMAssay Description:Inhibition of CSF1R (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588783(CHEMBL5182518)
Affinity DataIC50: 27nMAssay Description:Inhibition of recombinant AXL (unknown origin) using poly (Glu,Tyr) 4:1 as substrate incubated for 60 mins in presence of ATP by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588788(CHEMBL5175952)
Affinity DataIC50: 35nMAssay Description:Inhibition of recombinant AXL (unknown origin) using poly (Glu,Tyr) 4:1 as substrate incubated for 60 mins in presence of ATP by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588790(CHEMBL5188384)
Affinity DataIC50: 40nMAssay Description:Inhibition of recombinant AXL (unknown origin) using poly (Glu,Tyr) 4:1 as substrate incubated for 60 mins in presence of ATP by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588789(CHEMBL5194396)
Affinity DataIC50: 40nMAssay Description:Inhibition of recombinant AXL (unknown origin) using poly (Glu,Tyr) 4:1 as substrate incubated for 60 mins in presence of ATP by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588769(CHEMBL5209372)
Affinity DataIC50: 40nMAssay Description:Inhibition of recombinant AXL (unknown origin) using poly (Glu,Tyr) 4:1 as substrate incubated for 60 mins in presence of ATP by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588777(CHEMBL5183197)
Affinity DataIC50: 64nMAssay Description:Inhibition of recombinant AXL (unknown origin) using poly (Glu,Tyr) 4:1 as substrate incubated for 60 mins in presence of ATP by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588786(CHEMBL5182869)
Affinity DataIC50: 65nMAssay Description:Inhibition of recombinant AXL (unknown origin) using poly (Glu,Tyr) 4:1 as substrate incubated for 60 mins in presence of ATP by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588776(CHEMBL5169745)
Affinity DataIC50: 87nMAssay Description:Inhibition of recombinant AXL (unknown origin) using poly (Glu,Tyr) 4:1 as substrate incubated for 60 mins in presence of ATP by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588785(CHEMBL5197327)
Affinity DataIC50: 120nMAssay Description:Inhibition of recombinant AXL (unknown origin) using poly (Glu,Tyr) 4:1 as substrate incubated for 60 mins in presence of ATP by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588772(CHEMBL5197167)
Affinity DataIC50: 142nMAssay Description:Inhibition of recombinant AXL (unknown origin) using poly (Glu,Tyr) 4:1 as substrate incubated for 60 mins in presence of ATP by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataIC50: 151nMAssay Description:Inhibition of KIT (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataIC50: 156nMAssay Description:Inhibition of FLT3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588771(CHEMBL5191629)
Affinity DataIC50: 238nMAssay Description:Inhibition of recombinant AXL (unknown origin) using poly (Glu,Tyr) 4:1 as substrate incubated for 60 mins in presence of ATP by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588774(CHEMBL5196451)
Affinity DataIC50: 266nMAssay Description:Inhibition of recombinant AXL (unknown origin) using poly (Glu,Tyr) 4:1 as substrate incubated for 60 mins in presence of ATP by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588784(CHEMBL5188942)
Affinity DataIC50: 586nMAssay Description:Inhibition of recombinant AXL (unknown origin) using poly (Glu,Tyr) 4:1 as substrate incubated for 60 mins in presence of ATP by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588770(CHEMBL5179429)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of recombinant AXL (unknown origin) using poly (Glu,Tyr) 4:1 as substrate incubated for 60 mins in presence of ATP by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
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