Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50015708
TargetPotassium channel subfamily K member 3(Human)
Centro De Estudios En Alimentos Procesados-Ceap

Curated by ChEMBL
LigandPNGBDBM50312105(2-methoxy-N-(3-(3-methylbenzamido)phenyl)benzamide...)
Affinity DataIC50: 16nMAssay Description:Inhibition of human TASK-1 expressed in CHO cells assessed as inhibition of channel current at -30mV holding potential incubated for 5 mins by two-el...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetPotassium channel subfamily K member 3(Human)
Centro De Estudios En Alimentos Procesados-Ceap

Curated by ChEMBL
LigandPNGBDBM50123519(2'-{[2-(4-Methoxy-phenyl)-acetylamino]-methyl}-bip...)
Affinity DataIC50: 35nMAssay Description:Inhibition of human TASK-1 expressed in Xenopus laevis oocytes assessed as inhibition of channel current at +40mV holding potential by two-electrode ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetPotassium channel subfamily K member 3(Human)
Centro De Estudios En Alimentos Procesados-Ceap

Curated by ChEMBL
LigandPNGBDBM50588810(CHEMBL5201126)
Affinity DataIC50: 148nMAssay Description:Inhibition of human TASK-1 expressed in Xenopus laevis oocytes assessed as inhibition of channel current at +40mV holding potential by two-electrode ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetPotassium channel subfamily K member 3(Human)
Centro De Estudios En Alimentos Procesados-Ceap

Curated by ChEMBL
LigandPNGBDBM50123508([2'-(2-Pyridin-2-yl-ethylcarbamoyl)-biphenyl-2-ylm...)
Affinity DataIC50: 200nMAssay Description:Inhibition of human TASK-1 expressed in Xenopus laevis oocytes assessed as inhibition of channel current at +40mV holding potential by two-electrode ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetPotassium channel subfamily K member 3(Human)
Centro De Estudios En Alimentos Procesados-Ceap

Curated by ChEMBL
LigandPNGBDBM50588811(CHEMBL5195455)
Affinity DataIC50: 200nMAssay Description:Inhibition of human TASK-1 expressed in Xenopus laevis oocytes assessed as inhibition of channel current at +40mV holding potential by two-electrode ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetPotassium channel subfamily K member 3(Human)
Centro De Estudios En Alimentos Procesados-Ceap

Curated by ChEMBL
LigandPNGBDBM50588809(CHEMBL5181189)
Affinity DataIC50: 388nMAssay Description:Inhibition of human TASK-1 expressed in Xenopus laevis oocytes assessed as inhibition of channel current at +40mV holding potential by two-electrode ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetPotassium channel subfamily K member 3(Human)
Centro De Estudios En Alimentos Procesados-Ceap

Curated by ChEMBL
LigandPNGBDBM50417943(CHEMBL1671897)
Affinity DataIC50: 600nMAssay Description:Inhibition of human TASK-1 expressed in Xenopus laevis oocytes assessed as inhibition of channel current at +40mV holding potential by two-electrode ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetPotassium channel subfamily K member 9(Human)
Centro De Estudios En Alimentos Procesados-Ceap

Curated by ChEMBL
LigandPNGBDBM50588810(CHEMBL5201126)
Affinity DataIC50: 1.75E+3nMAssay Description:Inhibition of human TASK-3 expressed in Xenopus laevis oocytes assessed as inhibition of channel current at +40mV holding potential by two-electrode ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetPotassium channel subfamily K member 9(Human)
Centro De Estudios En Alimentos Procesados-Ceap

Curated by ChEMBL
LigandPNGBDBM50588809(CHEMBL5181189)
Affinity DataIC50: 7.17E+3nMAssay Description:Inhibition of human TASK-3 expressed in Xenopus laevis oocytes assessed as inhibition of channel current at +40mV holding potential by two-electrode ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetPotassium channel subfamily K member 3(Human)
Centro De Estudios En Alimentos Procesados-Ceap

Curated by ChEMBL
LigandPNGBDBM459029((4-{[2-(4-Chlorophenyl)imidazo [1,2-a]pyridin-3-yl...)
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of human TASK-1 expressed in Xenopus laevis oocytes assessed as inhibition of channel current at +40mV holding potential by two-electrode ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetPotassium channel subfamily K member 3(Human)
Centro De Estudios En Alimentos Procesados-Ceap

Curated by ChEMBL
LigandPNGBDBM458966((4-{[2-(4-Bromophenyl)imidazo [1,2-a]pyridin-3-yl]...)
Affinity DataIC50: 9.50E+3nMAssay Description:Inhibition of human TASK-1 expressed in Xenopus laevis oocytes assessed as inhibition of channel current at +40mV holding potential by two-electrode ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed