Compile Data Set for Download or QSAR
Report error Found 37 Enz. Inhib. hit(s) with all data for entry = 50017477
TargetP2Y purinoceptor 14(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456168(CHEMBL1800685)
Affinity DataIC50: 0.400nMAssay Description:Antagonist activity at P2Y14R (unknown origin) expressed in rat C6 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50602122(CHEMBL5208130)
Affinity DataIC50: 1.90nMAssay Description:Antagonist activity at P2Y14R (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456168(CHEMBL1800685)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at P2Y14R (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50602131(CHEMBL5203559)
Affinity DataIC50: 3.80nMAssay Description:Antagonist activity at P2Y14R (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50602119(CHEMBL5194881)
Affinity DataIC50: 3.80nMAssay Description:Antagonist activity at P2Y14R (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50602108(CHEMBL5182459)
Affinity DataIC50: 4nMAssay Description:Antagonist activity at P2Y14R (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50602109(CHEMBL5175291)
Affinity DataIC50: 4.20nMAssay Description:Antagonist activity at P2Y14R (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50602130(CHEMBL5189241)
Affinity DataIC50: 4.70nMAssay Description:Antagonist activity at P2Y14R (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50602115(CHEMBL5192153)
Affinity DataIC50: 4.70nMAssay Description:Antagonist activity at P2Y14R (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50602117(CHEMBL5185002)
Affinity DataIC50: 4.80nMAssay Description:Antagonist activity at P2Y14R (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50602116(CHEMBL5195243)
Affinity DataIC50: 5nMAssay Description:Antagonist activity at P2Y14R (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50602121(CHEMBL5203936)
Affinity DataIC50: 5.40nMAssay Description:Antagonist activity at P2Y14R (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50602111(CHEMBL5182261)
Affinity DataIC50: 5.80nMAssay Description:Antagonist activity at P2Y14R (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50602125(CHEMBL5208342)
Affinity DataIC50: 7.10nMAssay Description:Antagonist activity at P2Y14R (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50602132(CHEMBL5169372)
Affinity DataIC50: 14nMAssay Description:Antagonist activity at P2Y14R (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50602118(CHEMBL5183974)
Affinity DataIC50: 16nMAssay Description:Antagonist activity at P2Y14R (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50602110(CHEMBL5205552)
Affinity DataIC50: 41nMAssay Description:Antagonist activity at P2Y14R (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50602113(CHEMBL5203764)
Affinity DataIC50: 61nMAssay Description:Antagonist activity at P2Y14R (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50602114(CHEMBL5188038)
Affinity DataIC50: 67nMAssay Description:Antagonist activity at P2Y14R (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50602128(CHEMBL5209515)
Affinity DataIC50: 100nMAssay Description:Antagonist activity at P2Y14R (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50602120(CHEMBL5181115)
Affinity DataIC50: 111nMAssay Description:Antagonist activity at P2Y14R (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50602127(CHEMBL5189945)
Affinity DataIC50: 136nMAssay Description:Antagonist activity at P2Y14R (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50602126(CHEMBL5170216)
Affinity DataIC50: 171nMAssay Description:Antagonist activity at P2Y14R (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50602124(CHEMBL5189099)
Affinity DataIC50: 227nMAssay Description:Antagonist activity at P2Y14R (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50602123(CHEMBL5194765)
Affinity DataIC50: 245nMAssay Description:Antagonist activity at P2Y14R (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetP2Y purinoceptor 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50429537(CHEMBL2333770)
Affinity DataIC50: 350nMAssay Description:Antagonist activity at human P2Y1R expressed in HEK293 cells assessed as inhibition of ADP-induced IP3 production preincubated for 0.5 hrs followed b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetP2Y purinoceptor 14(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50602129(CHEMBL5206480)
Affinity DataIC50: 369nMAssay Description:Antagonist activity at P2Y14R (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetP2Y purinoceptor 14(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50602112(CHEMBL5205688)
Affinity DataIC50: 532nMAssay Description:Antagonist activity at P2Y14R (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetP2Y purinoceptor 13(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50397205(AR-C126532XX | AZD-6140 | AZD6140 | BRILINTA | TIC...)
Affinity DataIC50: 1.40E+3nMAssay Description:Antagonist activity at human P2Y13R expressed in HEK293 cells assessed as inhibition of 2MeSADP-induced cAMP production preincubated for 0.5 hrs foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetP2Y purinoceptor 11(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456168(CHEMBL1800685)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at P2Y11R (unknown origin) expressed in human 1321N1 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetP2Y purinoceptor 6(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456168(CHEMBL1800685)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at P2Y6R (unknown origin) expressed in human 1321N1 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetP2Y purinoceptor 12(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456168(CHEMBL1800685)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at P2Y12R (unknown origin) expressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetP2Y purinoceptor 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456168(CHEMBL1800685)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at P2Y1R (unknown origin) expressed in human 1321N1 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetP2Y purinoceptor 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456168(CHEMBL1800685)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at P2Y4R (unknown origin) expressed in human 1321N1 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetP2Y purinoceptor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456168(CHEMBL1800685)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at P2Y2R (unknown origin) expressed in human 1321N1 cells assessed as inhibition of forskolin-stimulated cAMP accumulation incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetP2Y purinoceptor 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50602133(CHEMBL5191550)
Affinity DataIC50: 1.36E+4nMAssay Description:Antagonist activity at human P2Y4R expressed in HEK293 cells assessed as inhibition of UTP-induced IP3 production preincubated for 0.5 hrs followed b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetP2Y purinoceptor 6(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50454137(CHEMBL1321988)
Affinity DataIC50: 3.95E+4nMAssay Description:Antagonist activity at human P2Y6R expressed in HEK293 cells assessed as inhibition of UDP-induced IP3 production preincubated for 0.5 hrs followed b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed