Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50020740
TargetSerine/threonine-protein kinase pim-1(Human)
Philipps-Universit£T Marburg

Curated by ChEMBL
LigandPNGBDBM50633211(CHEMBL5407681)
Affinity DataIC50: 600nMAssay Description:Inhibition of Pim-1 activity (unknown origin) by Eurofins radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Philipps-Universit£T Marburg

Curated by ChEMBL
LigandPNGBDBM50633212(CHEMBL5421756)
Affinity DataIC50: 2.74E+3nMAssay Description:Inhibition of Pim-1 activity (unknown origin) by Eurofins radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase pim-1(Human)
Philipps-Universit£T Marburg

Curated by ChEMBL
LigandPNGBDBM50633210(CHEMBL5416674)
Affinity DataIC50: 3.08E+3nMAssay Description:Inhibition of Pim-1 activity (unknown origin) by Eurofins radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase pim-1(Human)
Philipps-Universit£T Marburg

Curated by ChEMBL
LigandPNGBDBM50633209(CHEMBL5398429)
Affinity DataIC50: 2.64E+4nMAssay Description:Inhibition of Pim-1 activity (unknown origin) by Eurofins radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMedPDB3D3D Structure (crystal)