Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50018566
TargetSerine/threonine-protein kinase PAK 1(Human)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50609598(CHEMBL5274607)
Affinity DataIC50: 30nMAssay Description:Inhibition of human recombinant PAK1 assessed as phosphorylation FRET peptide substrate measured after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PAK 1(Human)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50609599(CHEMBL5281068)
Affinity DataIC50: 233nMAssay Description:Inhibition of human recombinant PAK1 assessed as phosphorylation FRET peptide substrate measured after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PAK 2(Human)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50609598(CHEMBL5274607)
Affinity DataIC50: 824nMAssay Description:Inhibition of human recombinant full length PAK2 assessed as phosphorylation FRET peptide substrate measured after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PAK 2(Human)
Fox Chase Cancer Center

Curated by ChEMBL
LigandPNGBDBM50609599(CHEMBL5281068)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant full length PAK2 assessed as phosphorylation FRET peptide substrate measured after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed