Compile Data Set for Download or QSAR
Report error Found 60 Enz. Inhib. hit(s) with all data for entry = 50019509
TargetFatty-acid amide hydrolase 1(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50395423(CHEMBL2165084)
Affinity DataIC50: 3.70nMAssay Description:Inhibition of human recombinant FAAH using AMC-AA as substrate preincubated for 30 mins followed by substrate addition and measured after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619997(CHEMBL5401122)
Affinity DataIC50: 7.5nMAssay Description:Inhibition of human recombinant FAAH using AMC-AA as substrate preincubated for 30 mins followed by substrate addition and measured after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619983(CHEMBL5430250)
Affinity DataIC50: 8.30nMAssay Description:Inhibition of human recombinant FAAH using AMC-AA as substrate preincubated for 30 mins followed by substrate addition and measured after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619992(CHEMBL5417524)
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant FAAH using AMC-AA as substrate preincubated for 30 mins followed by substrate addition and measured after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619995(CHEMBL5410254)
Affinity DataIC50: 11nMAssay Description:Inhibition of human recombinant FAAH using AMC-AA as substrate preincubated for 30 mins followed by substrate addition and measured after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619984(CHEMBL5432036)
Affinity DataIC50: 12nMAssay Description:Inhibition of human recombinant FAAH using AMC-AA as substrate preincubated for 30 mins followed by substrate addition and measured after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619989(CHEMBL5405509)
Affinity DataIC50: 16nMAssay Description:Inhibition of human recombinant FAAH using AMC-AA as substrate preincubated for 30 mins followed by substrate addition and measured after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619993(CHEMBL5420923)
Affinity DataIC50: 16nMAssay Description:Inhibition of human recombinant FAAH using AMC-AA as substrate preincubated for 30 mins followed by substrate addition and measured after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619985(CHEMBL5436635)
Affinity DataIC50: 26nMAssay Description:Inhibition of human recombinant FAAH using AMC-AA as substrate preincubated for 30 mins followed by substrate addition and measured after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM26739(URB 597 | URB597 | CHEMBL184238 | 3-(3-carbamoylph...)
Affinity DataIC50: 31nMAssay Description:Inhibition of human recombinant FAAH using AMC-AA as substrate preincubated for 30 mins followed by substrate addition and measured after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619994(CHEMBL5429985)
Affinity DataIC50: 47nMAssay Description:Inhibition of human recombinant FAAH using AMC-AA as substrate preincubated for 30 mins followed by substrate addition and measured after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50395421(CHEMBL2165094)
Affinity DataIC50: 102nMAssay Description:Inhibition of human recombinant FAAH using AMC-AA as substrate preincubated for 30 mins followed by substrate addition and measured after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619996(CHEMBL5440014)
Affinity DataIC50: 128nMAssay Description:Inhibition of human recombinant FAAH using AMC-AA as substrate preincubated for 30 mins followed by substrate addition and measured after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619986(CHEMBL5419246)
Affinity DataIC50: 165nMAssay Description:Inhibition of human recombinant FAAH using AMC-AA as substrate preincubated for 30 mins followed by substrate addition and measured after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619980(CHEMBL5403566)
Affinity DataIC50: 188nMAssay Description:Inhibition of human recombinant FAAH using AMC-AA as substrate preincubated for 30 mins followed by substrate addition and measured after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619987(CHEMBL5403865)
Affinity DataIC50: 194nMAssay Description:Inhibition of human recombinant FAAH using AMC-AA as substrate preincubated for 30 mins followed by substrate addition and measured after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619998(CHEMBL5419615)
Affinity DataIC50: 253nMAssay Description:Inhibition of human recombinant FAAH using AMC-AA as substrate preincubated for 30 mins followed by substrate addition and measured after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619990(CHEMBL5427155)
Affinity DataIC50: 315nMAssay Description:Inhibition of human recombinant FAAH using AMC-AA as substrate preincubated for 30 mins followed by substrate addition and measured after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619981(CHEMBL5396366)
Affinity DataIC50: 407nMAssay Description:Inhibition of human recombinant FAAH using AMC-AA as substrate preincubated for 30 mins followed by substrate addition and measured after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetMonoglyceride lipase(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619993(CHEMBL5420923)
Affinity DataIC50: 479nMAssay Description:Inhibition of human recombinant MAGL using 7-hydroxycoumarinyl arachidonate as substrate preincubated for 30 mins followed by substrate addition and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619979(CHEMBL5416058)
Affinity DataIC50: 1.04E+3nMAssay Description:Inhibition of human recombinant FAAH using AMC-AA as substrate preincubated for 30 mins followed by substrate addition and measured after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetMonoglyceride lipase(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619995(CHEMBL5410254)
Affinity DataIC50: 2.44E+3nMAssay Description:Inhibition of human recombinant MAGL using 7-hydroxycoumarinyl arachidonate as substrate preincubated for 30 mins followed by substrate addition and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetMonoglyceride lipase(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619994(CHEMBL5429985)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of human recombinant MAGL using 7-hydroxycoumarinyl arachidonate as substrate preincubated for 30 mins followed by substrate addition and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetMonoglyceride lipase(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619984(CHEMBL5432036)
Affinity DataIC50: 4.12E+3nMAssay Description:Inhibition of human recombinant MAGL using 7-hydroxycoumarinyl arachidonate as substrate preincubated for 30 mins followed by substrate addition and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetMonoglyceride lipase(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619983(CHEMBL5430250)
Affinity DataIC50: 5.06E+3nMAssay Description:Inhibition of human recombinant MAGL using 7-hydroxycoumarinyl arachidonate as substrate preincubated for 30 mins followed by substrate addition and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619982(CHEMBL5419776)
Affinity DataIC50: 6.56E+3nMAssay Description:Inhibition of human recombinant FAAH using AMC-AA as substrate preincubated for 30 mins followed by substrate addition and measured after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetMonoglyceride lipase(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619997(CHEMBL5401122)
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibition of human recombinant MAGL using 7-hydroxycoumarinyl arachidonate as substrate preincubated for 30 mins followed by substrate addition and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619988(CHEMBL5430706)
Affinity DataIC50: 8.45E+3nMAssay Description:Inhibition of human recombinant FAAH using AMC-AA as substrate preincubated for 30 mins followed by substrate addition and measured after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetMonoglyceride lipase(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM26739(URB 597 | URB597 | CHEMBL184238 | 3-(3-carbamoylph...)
Affinity DataIC50: 9.38E+3nMAssay Description:Inhibition of human recombinant MAGL using 7-hydroxycoumarinyl arachidonate as substrate preincubated for 30 mins followed by substrate addition and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetMonoglyceride lipase(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619986(CHEMBL5419246)
Affinity DataIC50: 9.88E+3nMAssay Description:Inhibition of human recombinant MAGL using 7-hydroxycoumarinyl arachidonate as substrate preincubated for 30 mins followed by substrate addition and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetMonoglyceride lipase(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619979(CHEMBL5416058)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant MAGL using 7-hydroxycoumarinyl arachidonate as substrate preincubated for 30 mins followed by substrate addition and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetMonoglyceride lipase(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619980(CHEMBL5403566)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant MAGL using 7-hydroxycoumarinyl arachidonate as substrate preincubated for 30 mins followed by substrate addition and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetMonoglyceride lipase(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619981(CHEMBL5396366)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant MAGL using 7-hydroxycoumarinyl arachidonate as substrate preincubated for 30 mins followed by substrate addition and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetMonoglyceride lipase(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619982(CHEMBL5419776)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant MAGL using 7-hydroxycoumarinyl arachidonate as substrate preincubated for 30 mins followed by substrate addition and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetMonoglyceride lipase(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619987(CHEMBL5403865)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant MAGL using 7-hydroxycoumarinyl arachidonate as substrate preincubated for 30 mins followed by substrate addition and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetMonoglyceride lipase(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619988(CHEMBL5430706)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant MAGL using 7-hydroxycoumarinyl arachidonate as substrate preincubated for 30 mins followed by substrate addition and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetMonoglyceride lipase(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619985(CHEMBL5436635)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant MAGL using 7-hydroxycoumarinyl arachidonate as substrate preincubated for 30 mins followed by substrate addition and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619991(CHEMBL5412058)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant FAAH using AMC-AA as substrate preincubated for 30 mins followed by substrate addition and measured after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetCannabinoid receptor 1(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619998(CHEMBL5419615)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cells assessed as inhibition constant incubated for 90 mins by liquid scintilla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetCannabinoid receptor 2(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619981(CHEMBL5396366)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells assessed as inhibition constant incubated for 60 mins by liquid scintilla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetCannabinoid receptor 1(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619994(CHEMBL5429985)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cells assessed as inhibition constant incubated for 90 mins by liquid scintilla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetCannabinoid receptor 1(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619997(CHEMBL5401122)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cells assessed as inhibition constant incubated for 90 mins by liquid scintilla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetCannabinoid receptor 2(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619989(CHEMBL5405509)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells assessed as inhibition constant incubated for 60 mins by liquid scintilla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetCannabinoid receptor 2(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619992(CHEMBL5417524)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells assessed as inhibition constant incubated for 60 mins by liquid scintilla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetCannabinoid receptor 2(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619983(CHEMBL5430250)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells assessed as inhibition constant incubated for 60 mins by liquid scintilla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetCannabinoid receptor 2(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619985(CHEMBL5436635)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells assessed as inhibition constant incubated for 60 mins by liquid scintilla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetCannabinoid receptor 2(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619998(CHEMBL5419615)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells assessed as inhibition constant incubated for 60 mins by liquid scintilla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetCannabinoid receptor 2(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619994(CHEMBL5429985)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells assessed as inhibition constant incubated for 60 mins by liquid scintilla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetCannabinoid receptor 2(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619997(CHEMBL5401122)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells assessed as inhibition constant incubated for 60 mins by liquid scintilla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetMonoglyceride lipase(Human)
Universit£

Curated by ChEMBL
LigandPNGBDBM50619991(CHEMBL5412058)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant MAGL using 7-hydroxycoumarinyl arachidonate as substrate preincubated for 30 mins followed by substrate addition and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
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