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Report error Found 42 Enz. Inhib. hit(s) with all data for entry = 50018603
TargetCholinesterase(Horse)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50022775(m-Trimethylammoniumphenyldimethylcarbamate | Prost...)
Affinity DataIC50: 160nMAssay Description:Inhibition of equine BChE using acetylthiocholine chloride as substrate preincubated for 15 mins followed by substrate addition and measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50252541(CHEMBL4069293)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of electrical eel AChE using acetylthiocholine chloride as substrate preincubated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM8960(2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimethoxy-2...)
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of electrical eel AChE using acetylthiocholine chloride as substrate preincubated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetCholinesterase(Horse)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50252541(CHEMBL4069293)
Affinity DataIC50: 1.67E+4nMAssay Description:Inhibition of equine BChE using acetylthiocholine chloride as substrate preincubated for 15 mins followed by substrate addition and measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetCholinesterase(Horse)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50610173(CHEMBL5280702)
Affinity DataIC50: 2.63E+4nMAssay Description:Inhibition of equine BChE using acetylthiocholine chloride as substrate preincubated for 15 mins followed by substrate addition and measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetCholinesterase(Horse)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50610168(CHEMBL5289654)
Affinity DataIC50: 4.07E+4nMAssay Description:Inhibition of equine BChE using acetylthiocholine chloride as substrate preincubated for 15 mins followed by substrate addition and measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetCholinesterase(Horse)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50610169(CHEMBL5270151)
Affinity DataIC50: 4.37E+4nMAssay Description:Inhibition of equine BChE using acetylthiocholine chloride as substrate preincubated for 15 mins followed by substrate addition and measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50610168(CHEMBL5289654)
Affinity DataIC50: 5.37E+4nMAssay Description:Inhibition of electrical eel AChE using acetylthiocholine chloride as substrate preincubated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetCholinesterase(Horse)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50610174(CHEMBL4293814)
Affinity DataIC50: 5.37E+4nMAssay Description:Inhibition of equine BChE using acetylthiocholine chloride as substrate preincubated for 15 mins followed by substrate addition and measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50610170(CHEMBL5278711)
Affinity DataIC50: 5.72E+4nMAssay Description:Inhibition of electrical eel AChE using acetylthiocholine chloride as substrate preincubated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetCholinesterase(Horse)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50610175(CHEMBL5283987)
Affinity DataIC50: 5.75E+4nMAssay Description:Inhibition of equine BChE using acetylthiocholine chloride as substrate preincubated for 15 mins followed by substrate addition and measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetCholinesterase(Horse)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50610171(CHEMBL5276899)
Affinity DataIC50: 5.89E+4nMAssay Description:Inhibition of equine BChE using acetylthiocholine chloride as substrate preincubated for 15 mins followed by substrate addition and measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetCholinesterase(Horse)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50610172(CHEMBL5267271)
Affinity DataIC50: 7.85E+4nMAssay Description:Inhibition of equine BChE using acetylthiocholine chloride as substrate preincubated for 15 mins followed by substrate addition and measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetCholinesterase(Horse)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50610176(CHEMBL5265920)
Affinity DataIC50: 8.51E+4nMAssay Description:Inhibition of equine BChE using acetylthiocholine chloride as substrate preincubated for 15 mins followed by substrate addition and measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetCholinesterase(Horse)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50610170(CHEMBL5278711)
Affinity DataIC50: 9.77E+4nMAssay Description:Inhibition of equine BChE using acetylthiocholine chloride as substrate preincubated for 15 mins followed by substrate addition and measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50610169(CHEMBL5270151)
Affinity DataIC50: 9.78E+4nMAssay Description:Inhibition of electrical eel AChE using acetylthiocholine chloride as substrate preincubated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetD(3) dopamine receptor(Human)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50610174(CHEMBL4293814)
Affinity DataKi:  0.340nMAssay Description:Binding affinity to human D3 receptor expressed in CHO cells assessed as inhibition constant by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetD(3) dopamine receptor(Human)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50610173(CHEMBL5280702)
Affinity DataKi:  0.700nMAssay Description:Binding affinity to human D3 receptor expressed in CHO cells assessed as inhibition constant by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetD(3) dopamine receptor(Human)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50610180(CHEMBL5276588)
Affinity DataKi:  0.860nMAssay Description:Binding affinity to human D3 receptor expressed in CHO cells assessed as inhibition constant by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetD(3) dopamine receptor(Human)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50610177(CHEMBL5268329)
Affinity DataKi:  0.920nMAssay Description:Inhibition of human D3 receptor expressed in CHO cells assessed as inhibition constant by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetD(3) dopamine receptor(Human)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50610178(CHEMBL5289468)
Affinity DataKi:  0.920nMAssay Description:Binding affinity to human D3 receptor expressed in CHO cells assessed as inhibition constant by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetD(3) dopamine receptor(Human)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50610182(CHEMBL5287235)
Affinity DataKi:  1.40nMAssay Description:Binding affinity to human D3 receptor expressed in CHO cells assessed as inhibition constant by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetD(3) dopamine receptor(Human)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50610169(CHEMBL5270151)
Affinity DataKi:  3.10nMAssay Description:Binding affinity to human D3 receptor expressed in CHO cells assessed as inhibition constant by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetD(3) dopamine receptor(Human)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50610176(CHEMBL5265920)
Affinity DataKi: >10nMAssay Description:Binding affinity to human D3 receptor expressed in CHO cells assessed as inhibition constant by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetD(3) dopamine receptor(Human)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50610170(CHEMBL5278711)
Affinity DataKi: >10nMAssay Description:Binding affinity to human D3 receptor expressed in CHO cells assessed as inhibition constant by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetD(3) dopamine receptor(Human)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50610181(CHEMBL5270288)
Affinity DataKi: >10nMAssay Description:Binding affinity to human D3 receptor expressed in CHO cells assessed as inhibition constant by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetD(3) dopamine receptor(Human)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50610179(CHEMBL5282002)
Affinity DataKi: >10nMAssay Description:Binding affinity to human D3 receptor expressed in CHO cells assessed as inhibition constant by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetD(3) dopamine receptor(Human)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50610175(CHEMBL5283987)
Affinity DataKi: >10nMAssay Description:Binding affinity to human D3 receptor expressed in CHO cells assessed as inhibition constant by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50405713(CHEMBL4173854)
Affinity DataKi:  16nMAssay Description:Inhibition of human H3 receptor assessed as inhibition constant incubated for 90 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetD(3) dopamine receptor(Human)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  54nMAssay Description:Binding affinity to human D3 receptor expressed in CHO cells assessed as inhibition constant by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50610170(CHEMBL5278711)
Affinity DataKi:  270nMAssay Description:Binding affinity to human H3 receptor assessed as inhibition constant incubated for 90 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50610176(CHEMBL5265920)
Affinity DataKi:  910nMAssay Description:Binding affinity to human H3 receptor assessed as inhibition constant incubated for 90 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50610169(CHEMBL5270151)
Affinity DataKi:  1.10E+3nMAssay Description:Binding affinity to human H3 receptor assessed as inhibition constant incubated for 90 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50610182(CHEMBL5287235)
Affinity DataKi:  1.70E+3nMAssay Description:Binding affinity to human H3 receptor assessed as inhibition constant incubated for 90 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50610180(CHEMBL5276588)
Affinity DataKi:  1.90E+3nMAssay Description:Binding affinity to human H3 receptor assessed as inhibition constant incubated for 90 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50610175(CHEMBL5283987)
Affinity DataKi:  2.20E+3nMAssay Description:Binding affinity to human H3 receptor assessed as inhibition constant incubated for 90 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50610173(CHEMBL5280702)
Affinity DataKi:  2.80E+3nMAssay Description:Binding affinity to human H3 receptor assessed as inhibition constant incubated for 90 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50610181(CHEMBL5270288)
Affinity DataKi:  3.30E+3nMAssay Description:Binding affinity to human H3 receptor assessed as inhibition constant incubated for 90 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50610179(CHEMBL5282002)
Affinity DataKi:  3.70E+3nMAssay Description:Binding affinity to human H3 receptor assessed as inhibition constant incubated for 90 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50610178(CHEMBL5289468)
Affinity DataKi:  4.00E+3nMAssay Description:Binding affinity to human H3 receptor assessed as inhibition constant incubated for 90 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50610174(CHEMBL4293814)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human H3 receptor assessed as inhibition constant incubated for 90 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Universidade Federal De Sao Paulo

Curated by ChEMBL
LigandPNGBDBM50247053(Tiprolisant | 1-(3-(3-(4-chlorophenyl)propoxy)prop...)
Affinity DataKi:  1.34E+4nMAssay Description:Binding affinity to human H3 receptor assessed as inhibition constant incubated for 90 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed