Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 50019173
TargetTranscriptional enhancer factor TEF-1(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50616138(CHEMBL5432067)
Affinity DataIC50: 200nMAssay Description:Displacement of FAM- labeled YAP1 peptide (60 to 99 residues) from human TEAD1 (209 to 426 residues) expressed in Escherichia coli BL21 (DE3) cells i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTranscriptional enhancer factor TEF-1(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50616136(CHEMBL5434817)
Affinity DataIC50: 200nMAssay Description:Displacement of FAM- labeled YAP1 peptide (60 to 99 residues) from human TEAD1 (209 to 426 residues) expressed in Escherichia coli BL21 (DE3) cells i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTranscriptional enhancer factor TEF-3(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50616135(CHEMBL5405832)
Affinity DataIC50: 200nMAssay Description:Displacement of FAM- labeled YAP1 peptide (60 to 99 residues) from human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21 (DE3) cells i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTranscriptional enhancer factor TEF-1(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50616135(CHEMBL5405832)
Affinity DataIC50: 300nMAssay Description:Displacement of FAM- labeled YAP1 peptide (60 to 99 residues) from human TEAD1 (209 to 426 residues) expressed in Escherichia coli BL21 (DE3) cells i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTranscriptional enhancer factor TEF-3(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50616135(CHEMBL5405832)
Affinity DataIC50: 300nMAssay Description:Inhibition of TEAD4 (unknown origin) transfected in human HEK293 cells co-transfected with renilla plasmid assessed as inhibition of transcriptional ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTranscriptional enhancer factor TEF-3(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50616139(CHEMBL5424157)
Affinity DataIC50: 400nMAssay Description:Inhibition of TEAD4 (unknown origin) transfected in human HEK293 cells co-transfected with renilla plasmid assessed as inhibition of transcriptional ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTranscriptional enhancer factor TEF-3(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50616138(CHEMBL5432067)
Affinity DataIC50: 600nMAssay Description:Displacement of FAM- labeled YAP1 peptide (60 to 99 residues) from human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21 (DE3) cells i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTranscriptional enhancer factor TEF-3(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50616138(CHEMBL5432067)
Affinity DataIC50: 700nMAssay Description:Inhibition of TEAD4 (unknown origin) transfected in human HEK293 cells co-transfected with renilla plasmid assessed as inhibition of transcriptional ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTranscriptional enhancer factor TEF-4(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50616136(CHEMBL5434817)
Affinity DataIC50: 800nMAssay Description:Displacement of FAM- labeled YAP1 peptide (60 to 99 residues) from human TEAD2 (217 to 447 residues) expressed in Escherichia coli BL21 (DE3) cells i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTranscriptional enhancer factor TEF-1(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50616134(CHEMBL5394226)
Affinity DataIC50: 900nMAssay Description:Displacement of FAM- labeled YAP1 peptide (60 to 99 residues) from human TEAD1 (209 to 426 residues) expressed in Escherichia coli BL21 (DE3) cells i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTranscriptional enhancer factor TEF-3(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50616134(CHEMBL5394226)
Affinity DataIC50: 1.10E+3nMAssay Description:Displacement of FAM- labeled YAP1 peptide (60 to 99 residues) from human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21 (DE3) cells i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTranscriptional enhancer factor TEF-4(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50616134(CHEMBL5394226)
Affinity DataIC50: 1.20E+3nMAssay Description:Displacement of FAM- labeled YAP1 peptide (60 to 99 residues) from human TEAD2 (217 to 447 residues) expressed in Escherichia coli BL21 (DE3) cells i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetTranscriptional enhancer factor TEF-5(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50616139(CHEMBL5424157)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of TEAD3 (unknown origin) transfected in human HEK293 cells co-transfected with renilla plasmid assessed as inhibition of transcriptional ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTranscriptional enhancer factor TEF-1(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50616137(CHEMBL5434933)
Affinity DataIC50: 1.30E+3nMAssay Description:Displacement of FAM- labeled YAP1 peptide (60 to 99 residues) from human TEAD1 (209 to 426 residues) expressed in Escherichia coli BL21 (DE3) cells i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTranscriptional enhancer factor TEF-1(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50616140(CHEMBL5432514)
Affinity DataIC50: 1.50E+3nMAssay Description:Displacement of FAM- labeled YAP1 peptide (60 to 99 residues) from human TEAD1 (209 to 426 residues) expressed in Escherichia coli BL21 (DE3) cells i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTranscriptional enhancer factor TEF-1(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50616139(CHEMBL5424157)
Affinity DataIC50: 1.60E+3nMAssay Description:Displacement of FAM- labeled YAP1 peptide (60 to 99 residues) from human TEAD1 (209 to 426 residues) expressed in Escherichia coli BL21 (DE3) cells i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTranscriptional enhancer factor TEF-1(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50616139(CHEMBL5424157)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of TEAD1 (unknown origin) transfected in human HEK293 cells co-transfected with renilla plasmid assessed as inhibition of transcriptional ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTranscriptional enhancer factor TEF-4(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50616135(CHEMBL5405832)
Affinity DataIC50: 1.70E+3nMAssay Description:Displacement of FAM- labeled YAP1 peptide (60 to 99 residues) from human TEAD2 (217 to 447 residues) expressed in Escherichia coli BL21 (DE3) cells i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTranscriptional enhancer factor TEF-3(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50616136(CHEMBL5434817)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of TEAD4 (unknown origin) transfected in human HEK293 cells co-transfected with renilla plasmid assessed as inhibition of transcriptional ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTranscriptional enhancer factor TEF-4(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50616137(CHEMBL5434933)
Affinity DataIC50: 2.10E+3nMAssay Description:Displacement of FAM- labeled YAP1 peptide (60 to 99 residues) from human TEAD2 (217 to 447 residues) expressed in Escherichia coli BL21 (DE3) cells i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetTranscriptional enhancer factor TEF-5(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50616134(CHEMBL5394226)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of TEAD3 (unknown origin) transfected in human HEK293 cells co-transfected with renilla plasmid assessed as inhibition of transcriptional ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTranscriptional enhancer factor TEF-4(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50616139(CHEMBL5424157)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of TEAD2 (unknown origin) transfected in human HEK293 cells co-transfected with renilla plasmid assessed as inhibition of transcriptional ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTranscriptional enhancer factor TEF-4(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50616138(CHEMBL5432067)
Affinity DataIC50: 2.40E+3nMAssay Description:Displacement of FAM- labeled YAP1 peptide (60 to 99 residues) from human TEAD2 (217 to 447 residues) expressed in Escherichia coli BL21 (DE3) cells i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTranscriptional enhancer factor TEF-4(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50616134(CHEMBL5394226)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of TEAD2 (unknown origin) transfected in human HEK293 cells co-transfected with renilla plasmid assessed as inhibition of transcriptional ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetTranscriptional enhancer factor TEF-3(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50616134(CHEMBL5394226)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of TEAD4 (unknown origin) transfected in human HEK293 cells co-transfected with renilla plasmid assessed as inhibition of transcriptional ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTranscriptional enhancer factor TEF-1(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50616134(CHEMBL5394226)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of TEAD1 (unknown origin) transfected in human HEK293 cells co-transfected with renilla plasmid assessed as inhibition of transcriptional ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTranscriptional enhancer factor TEF-3(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50616137(CHEMBL5434933)
Affinity DataIC50: 5.40E+3nMAssay Description:Displacement of FAM- labeled YAP1 peptide (60 to 99 residues) from human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21 (DE3) cells i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTranscriptional enhancer factor TEF-4(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50616141(CHEMBL5431797)
Affinity DataIC50: 7.50E+3nMAssay Description:Displacement of FAM- labeled YAP1 peptide (60 to 99 residues) from human TEAD2 (217 to 447 residues) expressed in Escherichia coli BL21 (DE3) cells i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTranscriptional enhancer factor TEF-3(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50616137(CHEMBL5434933)
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibition of TEAD4 (unknown origin) transfected in human HEK293 cells co-transfected with renilla plasmid assessed as inhibition of transcriptional ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTranscriptional enhancer factor TEF-4(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50616140(CHEMBL5432514)
Affinity DataIC50: 1.61E+4nMAssay Description:Displacement of FAM- labeled YAP1 peptide (60 to 99 residues) from human TEAD2 (217 to 447 residues) expressed in Escherichia coli BL21 (DE3) cells i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTranscriptional enhancer factor TEF-3(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50616140(CHEMBL5432514)
Affinity DataIC50: 2.01E+4nMAssay Description:Displacement of FAM- labeled YAP1 peptide (60 to 99 residues) from human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21 (DE3) cells i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTranscriptional enhancer factor TEF-4(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50616139(CHEMBL5424157)
Affinity DataIC50: 2.76E+4nMAssay Description:Displacement of FAM- labeled YAP1 peptide (60 to 99 residues) from human TEAD2 (217 to 447 residues) expressed in Escherichia coli BL21 (DE3) cells i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTranscriptional enhancer factor TEF-3(Human)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50616139(CHEMBL5424157)
Affinity DataIC50: 5.17E+4nMAssay Description:Displacement of FAM- labeled YAP1 peptide (60 to 99 residues) from human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21 (DE3) cells i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed