Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50019813
TargetCatenin beta-1(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50623192(CHEMBL5428813)
Affinity DataKd:  1.23E+3nMAssay Description:Binding affinity to full length His-tagged beta-catenin (1 to 781 residues) (unknown origin) expressed in Escherichia coli DE3 by surface plasmon res...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetB-cell CLL/lymphoma 9 protein(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50623192(CHEMBL5428813)
Affinity DataIC50: 2.75E+3nMAssay Description:Inhibition of full length beta-catenin (unknown origin) to BCL9-FAM (350 to 375 residues) (unknown origin) protein-protein interaction incubated for ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetB-cell CLL/lymphoma 9 protein(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50623192(CHEMBL5428813)
Affinity DataIC50: 2.78E+3nMAssay Description:Inhibition of beta-catenin (unknown origin) to BCL9-FAM (unknown origin) protein-protein interaction preincubated for 2 hrs followed by BCL9 addition...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetB-cell CLL/lymphoma 9 protein(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50623193(CHEMBL5412280)
Affinity DataIC50: 3.13E+3nMAssay Description:Inhibition of beta-catenin (unknown origin) to BCL9-FAM (unknown origin) protein-protein interaction preincubated for 2 hrs followed by BCL9 addition...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetB-cell CLL/lymphoma 9 protein(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50623195(CHEMBL5416319)
Affinity DataIC50: 4.46E+3nMAssay Description:Inhibition of beta-catenin (unknown origin) to BCL9-FAM (unknown origin) protein-protein interaction preincubated for 2 hrs followed by BCL9 addition...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCatenin beta-1(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-chromone;...)
Affinity DataKd:  5.58E+3nMAssay Description:Binding affinity to full length His-tagged beta-catenin (1 to 781 residues) (unknown origin) expressed in Escherichia coli DE3 by surface plasmon res...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetB-cell CLL/lymphoma 9 protein(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50623189(CHEMBL5435849)
Affinity DataIC50: 6.09E+3nMAssay Description:Inhibition of beta-catenin (unknown origin) to BCL9-FAM (unknown origin) protein-protein interaction preincubated for 2 hrs followed by BCL9 addition...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetB-cell CLL/lymphoma 9 protein(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50623190(CHEMBL5424377)
Affinity DataIC50: 9.13E+3nMAssay Description:Inhibition of beta-catenin (unknown origin) to BCL9-FAM (unknown origin) protein-protein interaction preincubated for 2 hrs followed by BCL9 addition...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetB-cell CLL/lymphoma 9 protein(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50623188(CHEMBL5403811)
Affinity DataIC50: 9.69E+3nMAssay Description:Inhibition of beta-catenin (unknown origin) to BCL9-FAM (unknown origin) protein-protein interaction preincubated for 2 hrs followed by BCL9 addition...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetB-cell CLL/lymphoma 9 protein(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-chromone;...)
Affinity DataIC50: 1.01E+4nMAssay Description:Inhibition of full length beta-catenin (unknown origin) to BCL9-FAM (350 to 375 residues) (unknown origin) protein-protein interaction incubated for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetB-cell CLL/lymphoma 9 protein(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-chromone;...)
Affinity DataIC50: 1.01E+4nMAssay Description:Inhibition of beta-catenin (unknown origin) to BCL9-FAM (unknown origin) protein-protein interaction preincubated for 2 hrs followed by BCL9 addition...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetB-cell CLL/lymphoma 9 protein(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50623205(CHEMBL5425670)
Affinity DataIC50: 1.17E+4nMAssay Description:Inhibition of beta-catenin (unknown origin) to BCL9-FAM (unknown origin) protein-protein interaction preincubated for 2 hrs followed by BCL9 addition...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetB-cell CLL/lymphoma 9 protein(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50623191(CHEMBL5429055)
Affinity DataIC50: 1.23E+4nMAssay Description:Inhibition of beta-catenin (unknown origin) to BCL9-FAM (unknown origin) protein-protein interaction preincubated for 2 hrs followed by BCL9 addition...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetB-cell CLL/lymphoma 9 protein(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50623203(CHEMBL5398792)
Affinity DataIC50: 1.86E+4nMAssay Description:Inhibition of beta-catenin (unknown origin) to BCL9-FAM (unknown origin) protein-protein interaction preincubated for 2 hrs followed by BCL9 addition...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetB-cell CLL/lymphoma 9 protein(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50623194(CHEMBL5398914)
Affinity DataIC50: 1.88E+4nMAssay Description:Inhibition of beta-catenin (unknown origin) to BCL9-FAM (unknown origin) protein-protein interaction preincubated for 2 hrs followed by BCL9 addition...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetB-cell CLL/lymphoma 9 protein(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50623204(CHEMBL5396319)
Affinity DataIC50: 2.01E+4nMAssay Description:Inhibition of beta-catenin (unknown origin) to BCL9-FAM (unknown origin) protein-protein interaction preincubated for 2 hrs followed by BCL9 addition...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetB-cell CLL/lymphoma 9 protein(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50623202(CHEMBL5420574)
Affinity DataIC50: 2.57E+4nMAssay Description:Inhibition of beta-catenin (unknown origin) to BCL9-FAM (unknown origin) protein-protein interaction preincubated for 2 hrs followed by BCL9 addition...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetB-cell CLL/lymphoma 9 protein(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50623201(CHEMBL5436043)
Affinity DataIC50: 2.79E+4nMAssay Description:Inhibition of beta-catenin (unknown origin) to BCL9-FAM (unknown origin) protein-protein interaction preincubated for 2 hrs followed by BCL9 addition...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetB-cell CLL/lymphoma 9 protein(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50623200(CHEMBL5423865)
Affinity DataIC50: 3.02E+4nMAssay Description:Inhibition of beta-catenin (unknown origin) to BCL9-FAM (unknown origin) protein-protein interaction preincubated for 2 hrs followed by BCL9 addition...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetB-cell CLL/lymphoma 9 protein(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50623197(CHEMBL5414209)
Affinity DataIC50: 3.11E+4nMAssay Description:Inhibition of beta-catenin (unknown origin) to BCL9-FAM (unknown origin) protein-protein interaction preincubated for 2 hrs followed by BCL9 addition...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetB-cell CLL/lymphoma 9 protein(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50623198(CHEMBL5431923)
Affinity DataIC50: 3.74E+4nMAssay Description:Inhibition of beta-catenin (unknown origin) to BCL9-FAM (unknown origin) protein-protein interaction preincubated for 2 hrs followed by BCL9 addition...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetB-cell CLL/lymphoma 9 protein(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50623196(CHEMBL5397763)
Affinity DataIC50: 5.68E+4nMAssay Description:Inhibition of beta-catenin (unknown origin) to BCL9-FAM (unknown origin) protein-protein interaction preincubated for 2 hrs followed by BCL9 addition...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetB-cell CLL/lymphoma 9 protein(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50623199(CHEMBL5436470)
Affinity DataIC50: 7.89E+4nMAssay Description:Inhibition of beta-catenin (unknown origin) to BCL9-FAM (unknown origin) protein-protein interaction preincubated for 2 hrs followed by BCL9 addition...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed