Compile Data Set for Download or QSAR
Report error Found 133 Enz. Inhib. hit(s) with all data for entry = 50018620
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610391(CHEMBL5290966)
Affinity DataIC50: 0.0600nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610384(CHEMBL5268011)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610396(CHEMBL5278104)
Affinity DataIC50: 0.150nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610428(CHEMBL5284020)
Affinity DataIC50: 0.160nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610389(CHEMBL5282887)
Affinity DataIC50: 0.190nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610383(CHEMBL5283410)
Affinity DataIC50: 0.25nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610427(CHEMBL5291181)
Affinity DataIC50: 0.370nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetMicrotubule-associated protein tau(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610396(CHEMBL5278104)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of tau phosphorylation (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610435(CHEMBL5286043)
Affinity DataIC50: 0.460nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610390(CHEMBL5282113)
Affinity DataIC50: 0.490nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610431(CHEMBL5276076)
Affinity DataIC50: 0.620nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610417(CHEMBL5271077)
Affinity DataIC50: 0.720nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610395(CHEMBL5272041)
Affinity DataIC50: 0.790nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610382(CHEMBL5290181)
Affinity DataIC50: 0.850nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610385(CHEMBL5273034)
Affinity DataIC50: 0.950nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610388(CHEMBL5288950)
Affinity DataIC50: 0.990nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610393(CHEMBL5281590)
Affinity DataIC50: 0.990nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610387(CHEMBL5289779)
Affinity DataIC50: 1nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610398(CHEMBL5273531)
Affinity DataIC50: 1nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610433(CHEMBL5286581)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610410(CHEMBL5289493)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610416(CHEMBL5272115)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610436(CHEMBL5271607)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610424(CHEMBL5272651)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610429(CHEMBL5290846)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetMicrotubule-associated protein tau(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610427(CHEMBL5291181)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of tau phosphorylation (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610418(CHEMBL5266570)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610425(CHEMBL5282635)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetMicrotubule-associated protein tau(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610428(CHEMBL5284020)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of tau phosphorylation (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetMicrotubule-associated protein tau(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610391(CHEMBL5290966)
Affinity DataIC50: 2nMAssay Description:Inhibition of tau phosphorylation (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610432(CHEMBL5280118)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610422(CHEMBL5276749)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610414(CHEMBL5287772)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610409(CHEMBL5276314)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610434(CHEMBL5270059)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610437(CHEMBL5269369)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610406(CHEMBL5285048)
Affinity DataIC50: 2.60nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610415(CHEMBL5268820)
Affinity DataIC50: 2.80nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetMicrotubule-associated protein tau(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610384(CHEMBL5268011)
Affinity DataIC50: 2.80nMAssay Description:Inhibition of tau phosphorylation (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610404(CHEMBL5266186)
Affinity DataIC50: 3nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610386(CHEMBL5277764)
Affinity DataIC50: 3.60nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610405(CHEMBL5291257)
Affinity DataIC50: 3.70nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610408(CHEMBL5276201)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610426(CHEMBL5271312)
Affinity DataIC50: 4.10nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610438(CHEMBL5272462)
Affinity DataIC50: 4.10nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610421(CHEMBL5276840)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610377(CHEMBL5265899)
Affinity DataIC50: 4.40nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610439(CHEMBL5283804)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610413(CHEMBL5273399)
Affinity DataIC50: 4.60nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50610407(CHEMBL5285396)
Affinity DataIC50: 4.80nMAssay Description:Inhibition of GSK-3beta (unknown origin) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
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