Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50018211
TargetPlasma kallikrein(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50406180(CHEMBL5276780 | US20240190892, Example 23)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of human plasma kallikrein using Acetyl-K- P-R-AFC as substrate by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetPlasma kallikrein(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50406177(CHEMBL5285047 | US20240190892, Example 15)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of human plasma kallikrein using Acetyl-K- P-R-AFC as substrate by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetPlasma kallikrein(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50406172(CHEMBL5290426 | US20240190892, Example 4)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of human plasma kallikrein using Acetyl-K- P-R-AFC as substrate by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetPlasma kallikrein(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50406178(CHEMBL5267934 | US20240190892, Example 20)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human plasma kallikrein using Acetyl-K- P-R-AFC as substrate by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetPlasma kallikrein(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50406174(CHEMBL5274983 | US20240190892, Example 14)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human plasma kallikrein using Acetyl-K- P-R-AFC as substrate by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetPlasma kallikrein(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50406322(CHEMBL5267385 | US20240190892, Example 43)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of human plasma kallikrein using Acetyl-K- P-R-AFC as substrate by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetPlasma kallikrein(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50406173(CHEMBL5270511 | US20240190892, Example 10)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of human plasma kallikrein using Acetyl-K- P-R-AFC as substrate by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetPlasma kallikrein(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50406171(CHEMBL5283110 | US20240190892, Example 1)
Affinity DataIC50: 19nMAssay Description:Inhibition of human plasma kallikrein using Acetyl-K- P-R-AFC as substrate by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetPlasma kallikrein(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50406323(CHEMBL5273808 | US20240190892, Example 50)
Affinity DataIC50: 27nMAssay Description:Inhibition of human plasma kallikrein using Acetyl-K- P-R-AFC as substrate by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetPlasma kallikrein(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50406182(CHEMBL5268598 | US20240190892, Example 37)
Affinity DataIC50: 44nMAssay Description:Inhibition of human plasma kallikrein using Acetyl-K- P-R-AFC as substrate by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetPlasma kallikrein(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50406172(CHEMBL5290426 | US20240190892, Example 4)
Affinity DataIC50: 7.44E+3nMAssay Description:Inhibition of human factor 11a using GPR-AFC as substrate preincubated for 30 mins followed by substrate addition and measured after 60 mins by fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetPlasma kallikrein(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50406174(CHEMBL5274983 | US20240190892, Example 14)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human factor 11a using GPR-AFC as substrate preincubated for 30 mins followed by substrate addition and measured after 60 mins by fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetPlasma kallikrein(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50406322(CHEMBL5267385 | US20240190892, Example 43)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human factor 11a using GPR-AFC as substrate preincubated for 30 mins followed by substrate addition and measured after 60 mins by fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetPlasma kallikrein(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50406177(CHEMBL5285047 | US20240190892, Example 15)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human factor 11a using GPR-AFC as substrate preincubated for 30 mins followed by substrate addition and measured after 60 mins by fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetPlasma kallikrein(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50406323(CHEMBL5273808 | US20240190892, Example 50)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human factor 11a using GPR-AFC as substrate preincubated for 30 mins followed by substrate addition and measured after 60 mins by fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetPlasma kallikrein(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50406171(CHEMBL5283110 | US20240190892, Example 1)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human factor 11a using GPR-AFC as substrate preincubated for 30 mins followed by substrate addition and measured after 60 mins by fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetPlasma kallikrein(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50406178(CHEMBL5267934 | US20240190892, Example 20)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human factor 11a using GPR-AFC as substrate preincubated for 30 mins followed by substrate addition and measured after 60 mins by fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetPlasma kallikrein(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50406180(CHEMBL5276780 | US20240190892, Example 23)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human factor 11a using GPR-AFC as substrate preincubated for 30 mins followed by substrate addition and measured after 60 mins by fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetPlasma kallikrein(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50406173(CHEMBL5270511 | US20240190892, Example 10)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human factor 11a using GPR-AFC as substrate preincubated for 30 mins followed by substrate addition and measured after 60 mins by fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetPlasma kallikrein(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50406182(CHEMBL5268598 | US20240190892, Example 37)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human factor 11a using GPR-AFC as substrate preincubated for 30 mins followed by substrate addition and measured after 60 mins by fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed