Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50020661
TargetAlpha-2B adrenergic receptor(Rat)
Bayer

Curated by ChEMBL
LigandPNGBDBM50632390(CHEMBL5410211)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at rat adrenergic alpha2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(Dog)
Bayer

Curated by ChEMBL
LigandPNGBDBM50632390(CHEMBL5410211)
Affinity DataIC50: 25nMAssay Description:Antagonist activity at dog adrenergic alpha2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50632390(CHEMBL5410211)
Affinity DataKi:  21nMAssay Description:Binding affinity to human recombinant adrenergic alpha2B receptor expressed in CHO cell assessed as inhibition constant by radioactive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed