Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50019013
Affinity DataEC50: 140nMAssay Description:Partial agonist activity at FXR-LBD-GST (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 490nMAssay Description:Partial agonist activity at FXR-LBD-GST (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 250nMAssay Description:Partial agonist activity at FXR-LBD-GST (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 410nMAssay Description:Partial agonist activity at FXR-LBD-GST (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 630nMAssay Description:Partial agonist activity at FXR-LBD-GST (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 640nMAssay Description:Partial agonist activity at FXR-LBD-GST (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 760nMAssay Description:Partial agonist activity at FXR-LBD-GST (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 510nMAssay Description:Partial agonist activity at FXR-LBD-GST (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 140nMAssay Description:Partial agonist activity at FXR-LBD-GST (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.20E+3nMAssay Description:Partial agonist activity at human FXR expressed in Huh-7 cells in presence of CDCA by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.90E+3nMAssay Description:Partial agonist activity at human FXR expressed in Huh-7 cells in presence of CDCA by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Human)
Hiroshima International University
Curated by ChEMBL
Hiroshima International University
Curated by ChEMBL
Affinity DataEC50: 2.10E+3nMAssay Description:Partial agonist activity at PPARgamma (unknown origin) by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Human)
Hiroshima International University
Curated by ChEMBL
Hiroshima International University
Curated by ChEMBL
Affinity DataIC50: 5.30E+3nMAssay Description:Partial agonist activity at PPARgamma (unknown origin) in presence of GW1929More data for this Ligand-Target Pair
Affinity DataIC50: 9.90E+3nMAssay Description:Antagonist activity at FXR-LBD-GST (unknown origin) in presence of GW4064More data for this Ligand-Target Pair
Affinity DataIC50: 2.07E+4nMAssay Description:Antagonist activity at FXR-LBD-GST (unknown origin) in presence of GW4064More data for this Ligand-Target Pair
