Compile Data Set for Download or QSAR
Report error Found 82 Enz. Inhib. hit(s) with all data for entry = 50019694
TargetTyrosine-protein kinase Yes(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621890(CHEMBL5415503)
Affinity DataKd:  42nMAssay Description:Binding affinity to YES (unknown origin) assessed as dissociation constant by KINOME scan assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM13216(N-(2-Chloro-6-methylphenyl)-2-[[6-[4-(2-hydroxyeth...)
Affinity DataKd:  6nMAssay Description:Binding affinity to ACK1 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetEphrin type-A receptor 3(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621890(CHEMBL5415503)
Affinity DataKd:  23nMAssay Description:Binding affinity to EPHA3 (unknown origin) assessed as dissociation constant by KINOME scan assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetEphrin type-A receptor 8(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621890(CHEMBL5415503)
Affinity DataKd:  15nMAssay Description:Binding affinity to EPHA8 (unknown origin) assessed as dissociation constant by KINOME scan assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetEphrin type-B receptor 6(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621890(CHEMBL5415503)
Affinity DataKd:  10nMAssay Description:Binding affinity to EPHB6 (unknown origin) assessed as dissociation constant by KINOME scan assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-4(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621890(CHEMBL5415503)
Affinity DataKd:  16nMAssay Description:Binding affinity to ERBB4 (unknown origin) assessed as dissociation constant by KINOME scan assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetFocal adhesion kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621890(CHEMBL5415503)
Affinity DataKd:  34nMAssay Description:Binding affinity to FAK (unknown origin) assessed as dissociation constant by KINOME scan assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetFibroblast growth factor receptor 4(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621890(CHEMBL5415503)
Affinity DataKd:  43nMAssay Description:Binding affinity to FGFR4 (unknown origin) assessed as dissociation constant by KINOME scan assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetTyrosine-protein kinase FRK(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621890(CHEMBL5415503)
Affinity DataKd:  6.90nMAssay Description:Binding affinity to FRK (unknown origin) assessed as dissociation constant by KINOME scan assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetCyclin-G-associated kinase(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621890(CHEMBL5415503)
Affinity DataKd:  1nMAssay Description:Binding affinity to GAK (unknown origin) assessed as dissociation constant by KINOME scan assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetTyrosine-protein kinase HCK(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621890(CHEMBL5415503)
Affinity DataKd:  11nMAssay Description:Binding affinity to HCK (unknown origin) assessed as dissociation constant by KINOME scan assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase 8(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621890(CHEMBL5415503)
Affinity DataKd:  20nMAssay Description:Binding affinity to JNK1 (unknown origin) assessed as dissociation constant by KINOME scan assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase 9(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621890(CHEMBL5415503)
Affinity DataKd:  5.80nMAssay Description:Binding affinity to JNK2 (unknown origin) assessed as dissociation constant by KINOME scan assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase 10(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621890(CHEMBL5415503)
Affinity DataKd:  23nMAssay Description:Binding affinity to JNK3 (unknown origin) assessed as dissociation constant by KINOME scan assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetTyrosine-protein kinase Lck(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621890(CHEMBL5415503)
Affinity DataKd:  18nMAssay Description:Binding affinity to LCK (unknown origin) assessed as dissociation constant by KINOME scan assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase 14(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621890(CHEMBL5415503)
Affinity DataKd:  4.40nMAssay Description:Binding affinity to p38-alpha (unknown origin) assessed as dissociation constant by KINOME scan assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetTyrosine-protein kinase receptor Tie-1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621890(CHEMBL5415503)
Affinity DataKd:  67nMAssay Description:Binding affinity to TIE1 (unknown origin) assessed as dissociation constant by KINOME scan assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50621890(CHEMBL5415503)
Affinity DataKd:  1.30nMAssay Description:Binding affinity to MEK5 (unknown origin) assessed as dissociation constant by KINOME scan assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TNK1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621890(CHEMBL5415503)
Affinity DataKd:  15nMAssay Description:Binding affinity to TNK1 (unknown origin) assessed as dissociation constant by KINOME scan assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetTyrosine-protein kinase Srms(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621890(CHEMBL5415503)
Affinity DataKd:  28nMAssay Description:Binding affinity to SRMS (unknown origin) assessed as dissociation constant by KINOME scan assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase SIK1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621890(CHEMBL5415503)
Affinity DataKd:  11nMAssay Description:Binding affinity to SIK (unknown origin) assessed as dissociation constant by KINOME scan assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetProtein-tyrosine kinase 2-beta(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621890(CHEMBL5415503)
Affinity DataKd:  49nMAssay Description:Binding affinity to PYK2 (unknown origin) assessed as dissociation constant by KINOME scan assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PAK 3(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621890(CHEMBL5415503)
Affinity DataKd:  44nMAssay Description:Binding affinity to PAK3 (unknown origin) assessed as dissociation constant by KINOME scan assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase 11(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621890(CHEMBL5415503)
Affinity DataKd:  9.40nMAssay Description:Binding affinity to p38-beta (unknown origin) assessed as dissociation constant by KINOME scan assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase TNNI3K(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621890(CHEMBL5415503)
Affinity DataKd:  39nMAssay Description:Binding affinity to TNNI3K (unknown origin) assessed as dissociation constant by KINOME scan assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621875(CHEMBL5400397)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621877(CHEMBL5408748)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621883(CHEMBL5431206)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621855(CHEMBL5409024)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621888(CHEMBL5419830)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621858(CHEMBL5398945)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621880(CHEMBL5428907)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621878(CHEMBL5405674)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621884(CHEMBL5399309)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621876(CHEMBL5437496)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621882(CHEMBL5439245)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621881(CHEMBL5436567)
Affinity DataIC50: 1nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621879(CHEMBL5434969)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621862(CHEMBL5431312)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621871(CHEMBL5404048)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621890(CHEMBL5415503)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621882(CHEMBL5439245)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of SRC (unknown origin) using ATP as substrate incubated for 1 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621861(CHEMBL5404162)
Affinity DataIC50: 2.60nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621865(CHEMBL5413451)
Affinity DataIC50: 2.80nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621889(CHEMBL5407266)
Affinity DataIC50: 3nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621863(CHEMBL5432622)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621870(CHEMBL5409596)
Affinity DataIC50: 5.10nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621886(CHEMBL5402678)
Affinity DataIC50: 5.70nMAssay Description:Inhibition of SRC (unknown origin) using ATP as substrate incubated for 1 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621864(CHEMBL5437772)
Affinity DataIC50: 5.70nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetActivated CDC42 kinase 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50621869(CHEMBL5432393)
Affinity DataIC50: 5.80nMAssay Description:Inhibition of N-terminal His6-tagged ACK1 (117 to 389 residues) (unknown origin) expressed in Sf9 cells using ATP as substrate incubated for 1 hrs by...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
Displayed 1 to 50 (of 82 total ) | Next | Last >>
Jump to: