Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50020399
TargetEstrogen receptor(Human)
Central University of Punjab

Curated by ChEMBL
LigandPNGBDBM349630(US10208011, Compound RAD- | US10981887, Compound R...)
Affinity DataIC50: 48nMAssay Description:Inhibition of ERalpha (unknown origin) incubated for 4 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetEstrogen receptor beta(Human)
Central University of Punjab

Curated by ChEMBL
LigandPNGBDBM349630(US10208011, Compound RAD- | US10981887, Compound R...)
Affinity DataIC50: 870nMAssay Description:Inhibition of ERbeta (unknown origin) incubated for 4 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetEstrogen receptor(Human)
Central University of Punjab

Curated by ChEMBL
LigandPNGBDBM50084948(GW7604 | CHEMBL195515)
Affinity DataKi:  27nMAssay Description:Displacement of Fluormone ES2 from full-length recombinant ER alpha (unknown origin) assessed as inhibition constant incubated for 2 hrs by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetEstrogen receptor(Human)
Central University of Punjab

Curated by ChEMBL
LigandPNGBDBM50629586(CHEMBL5400663)
Affinity DataKi:  210nMAssay Description:Displacement of Fluormone ES2 from full-length recombinant ER alpha (unknown origin) assessed as inhibition constant incubated for 2 hrs by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetEstrogen receptor(Human)
Central University of Punjab

Curated by ChEMBL
LigandPNGBDBM50629585(CHEMBL5408419)
Affinity DataKi:  240nMAssay Description:Displacement of Fluormone ES2 from full-length recombinant ER alpha (unknown origin) assessed as inhibition constant incubated for 2 hrs by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed