Compile Data Set for Download or QSAR
Report error Found 35 Enz. Inhib. hit(s) with all data for entry = 50020251
TargetAryl hydrocarbon receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50628134(CHEMBL5410096)
Affinity DataEC50:  15nMAssay Description:Agonist activity at AHR in human HepG2-Lucia AhR cells stably transfected with DRE by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50603566(TAPINAROF | Tapinarof | Benvitimod | Vtama | Wbi-1...)
Affinity DataEC50:  27nMAssay Description:Agonist activity at AHR in human HepG2-Lucia AhR cells stably transfected with DRE by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50628135(CHEMBL5418753)
Affinity DataEC50:  35nMAssay Description:Agonist activity at AHR in human HepG2-Lucia AhR cells stably transfected with DRE by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50628125(CHEMBL5419477)
Affinity DataEC50:  49nMAssay Description:Agonist activity at AHR in human HepG2-Lucia AhR cells stably transfected with DRE by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50628133(CHEMBL5406192)
Affinity DataEC50:  52nMAssay Description:Agonist activity at AHR in human HepG2-Lucia AhR cells stably transfected with DRE by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50628117(CHEMBL5439352)
Affinity DataEC50:  143nMAssay Description:Agonist activity at AHR in human HepG2-Lucia AhR cells stably transfected with DRE by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50628130(CHEMBL5434388)
Affinity DataEC50:  163nMAssay Description:Agonist activity at AHR in human HepG2-Lucia AhR cells stably transfected with DRE by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50628132(CHEMBL5416301)
Affinity DataEC50:  219nMAssay Description:Agonist activity at AHR in human HepG2-Lucia AhR cells stably transfected with DRE by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50628136(CHEMBL5399322)
Affinity DataEC50:  528nMAssay Description:Agonist activity at AHR in human HepG2-Lucia AhR cells stably transfected with DRE by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50628121(CHEMBL5419189)
Affinity DataEC50:  613nMAssay Description:Agonist activity at AHR in human HepG2-Lucia AhR cells stably transfected with DRE by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50628122(CHEMBL5426272)
Affinity DataEC50:  858nMAssay Description:Agonist activity at AHR in human HepG2-Lucia AhR cells stably transfected with DRE by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50628119(CHEMBL5429807)
Affinity DataEC50:  1.80E+3nMAssay Description:Agonist activity at AHR in human HepG2-Lucia AhR cells stably transfected with DRE by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50628126(CHEMBL5435523)
Affinity DataEC50:  1.80E+3nMAssay Description:Agonist activity at AHR in human HepG2-Lucia AhR cells stably transfected with DRE by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50628131(CHEMBL5413861)
Affinity DataEC50:  2.50E+3nMAssay Description:Agonist activity at AHR in human HepG2-Lucia AhR cells stably transfected with DRE by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50628124(CHEMBL5434232)
Affinity DataEC50:  2.77E+3nMAssay Description:Agonist activity at AHR in human HepG2-Lucia AhR cells stably transfected with DRE by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50628118(CHEMBL5411787)
Affinity DataEC50:  2.80E+3nMAssay Description:Agonist activity at AHR in human HepG2-Lucia AhR cells stably transfected with DRE by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50628120(CHEMBL5410987)
Affinity DataEC50:  3.20E+3nMAssay Description:Agonist activity at AHR in human HepG2-Lucia AhR cells stably transfected with DRE by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50628111(CHEMBL5398518)
Affinity DataEC50:  3.40E+3nMAssay Description:Agonist activity at AHR in human HepG2-Lucia AhR cells stably transfected with DRE by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM51057(4-[4-(4-methyl-2-quinolinyl)phenyl]morpholine;hydr...)
Affinity DataEC50:  4.70E+3nMAssay Description:Agonist activity at AHR in human HepG2-Lucia AhR cells stably transfected with DRE by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50628112(CHEMBL5419047)
Affinity DataEC50:  5.90E+3nMAssay Description:Agonist activity at AHR in human HepG2-Lucia AhR cells stably transfected with DRE by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50628116(CHEMBL5400187)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at AHR in human HepG2-Lucia AhR cells stably transfected with DRE by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50347917(CHEMBL38739)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at AHR in human HepG2-Lucia AhR cells stably transfected with DRE by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50628115(CHEMBL5431457)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at AHR in human HepG2-Lucia AhR cells stably transfected with DRE by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50388005(CHEMBL541474)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at AHR in human HepG2-Lucia AhR cells stably transfected with DRE by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50628123(CHEMBL5430036)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at AHR in human HepG2-Lucia AhR cells stably transfected with DRE by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50628127(CHEMBL5418142)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at AHR in human HepG2-Lucia AhR cells stably transfected with DRE by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50628128(CHEMBL5403712)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at AHR in human HepG2-Lucia AhR cells stably transfected with DRE by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50628129(CHEMBL5418120)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at AHR in human HepG2-Lucia AhR cells stably transfected with DRE by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50628138(CHEMBL5398462)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at AHR in human HepG2-Lucia AhR cells stably transfected with DRE by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50628139(CHEMBL5396882)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at AHR in human HepG2-Lucia AhR cells stably transfected with DRE by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50628137(CHEMBL5420784)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at AHR in human HepG2-Lucia AhR cells stably transfected with DRE by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50628113(CHEMBL5420973)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at AHR in human HepG2-Lucia AhR cells stably transfected with DRE by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50628114(CHEMBL5393776)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at AHR in human HepG2-Lucia AhR cells stably transfected with DRE by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50628140(CHEMBL5429469)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at AHR in human HepG2-Lucia AhR cells stably transfected with DRE by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetAryl hydrocarbon receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM36371(CID2828334 | 5-(1H-indol-3-ylmethyl)-3-methyl-2-th...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at AHR in human HepG2-Lucia AhR cells stably transfected with DRE by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed