Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50019877
TargetAlpha-ketoglutarate-dependent dioxygenase FTO(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50624049(CHEMBL5410889)
Affinity DataIC50: 120nMAssay Description:Inhibition of FTO (unknown origin) using (5'-AUUGUCA(M6A)CAGCAGC-3') as substrate incubated for 2 hrs by dot-blot assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetAlpha-ketoglutarate-dependent dioxygenase FTO(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM589235(US11555009, Compound 15 | US11555009, Compound 29)
Affinity DataIC50: 400nMAssay Description:Inhibition of FTO (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetAlpha-ketoglutarate-dependent dioxygenase FTO(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50594337(CHEMBL5176730)
Affinity DataIC50: 700nMAssay Description:Inhibition of FTO (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetAlpha-ketoglutarate-dependent dioxygenase FTO(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50624048(CHEMBL5397077)
Affinity DataIC50: 800nMAssay Description:Inhibition of FTO (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetAlpha-ketoglutarate-dependent dioxygenase FTO(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50624049(CHEMBL5410889)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of FTO (unknown origin) by PAGE based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetAlpha-ketoglutarate-dependent dioxygenase FTO(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50624049(CHEMBL5410889)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of FTO (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetAlpha-ketoglutarate-dependent dioxygenase FTO(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50624047(CHEMBL5429303)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of FTO (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetAlpha-ketoglutarate-dependent dioxygenase FTO(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50624044(CHEMBL5396359)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of FTO (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetAlpha-ketoglutarate-dependent dioxygenase FTO(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50624054(CHEMBL5421288)
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of FTO (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetAlpha-ketoglutarate-dependent dioxygenase FTO(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50624052(CHEMBL5414569)
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of FTO (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetAlpha-ketoglutarate-dependent dioxygenase FTO(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50624045(CHEMBL5416975)
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of FTO (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetAlpha-ketoglutarate-dependent dioxygenase FTO(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50624046(CHEMBL5396816)
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of FTO (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetAlpha-ketoglutarate-dependent dioxygenase FTO(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50624051(CHEMBL5423698)
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of FTO (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetAlpha-ketoglutarate-dependent dioxygenase FTO(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50624053(CHEMBL5396378)
Affinity DataIC50: 1.01E+4nMAssay Description:Inhibition of FTO (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetAlpha-ketoglutarate-dependent dioxygenase FTO(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50624050(CHEMBL5421628)
Affinity DataIC50: 1.68E+4nMAssay Description:Inhibition of FTO (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed