Compile Data Set for Download or QSAR
Report error Found 47 Enz. Inhib. hit(s) with all data for entry = 50019398
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618851(CHEMBL5408440)
Affinity DataKd:  620nMAssay Description:Inhibition of full length human Pin1 expressed in Escherichia coli assessed as dissociation constant by fluorescence anisotropy binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618850(CHEMBL5423483)
Affinity DataKd:  72nMAssay Description:Inhibition of full length human Pin1 expressed in Escherichia coli assessed as dissociation constant by fluorescence anisotropy binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618845(CHEMBL5408559)
Affinity DataIC50: 31nMAssay Description:Inhibition of Pin1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618848(CHEMBL5427982)
Affinity DataIC50: 72nMAssay Description:Inhibition of Pin1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618839(CHEMBL5430620)
Affinity DataIC50: 210nMAssay Description:Inhibition of Gst-tagged human Pin1 by Western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618846(CHEMBL5406982)
Affinity DataIC50: 220nMAssay Description:Inhibition of Pin1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618849(CHEMBL5437431)
Affinity DataIC50: 245nMAssay Description:Inhibition of Pin1 (unknown origin) by fluorescence anisotropy binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618833(CHEMBL5411977)
Affinity DataIC50: 440nMAssay Description:Inhibition of Pin1 (unknown origin) using Suc-Ala-Glu-Pro-Phe-pNA as substrate by spectrofluorometry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataIC50: 580nMAssay Description:Inhibition of Gst-tagged human Pin1by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618832(CHEMBL5406477)
Affinity DataIC50: 780nMAssay Description:Inhibition of Pin1 (unknown origin) using Suc-Ala-Glu-Pro-Phe-pNA as substrate by spectrofluorometry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618847(CHEMBL5436856)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of Pin1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618852(CHEMBL5405224)
Affinity DataIC50: 1.07E+3nMAssay Description:Inhibition of human Pin1 measured after 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50437711(CHEMBL2409076)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human Pin1 using Suc-Ala-Glu-Pro-Phe-MCA as substrate by fluorescence based microtitre plate analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM24777(5-hydroxy-1,4-dihydronaphthalene-1,4-dione | CHEMB...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human Pin1 using Suc-AEPF-NH-Np as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618863(CHEMBL5433320)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of human Pin1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618838(CHEMBL5427301)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of Gst-tagged human Pin1 by Western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618836(CHEMBL5413642)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of Gst-tagged human Pin1 by Western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618835(CHEMBL5433155)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of Gst-tagged human Pin1 by Western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618837(CHEMBL5424284)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of Gst-tagged human Pin1 by Western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618842(CHEMBL5395865)
Affinity DataKi:  1.20nMAssay Description:Inhibition of Gst-tagged human Pin1 assessed as inhibition constant by Western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50552328(CHEMBL4750217)
Affinity DataKi:  15nMAssay Description:Inhibition of Gst-tagged human Pin1 assessed as inhibition constant measured after 12 hrs by FP binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618843(CHEMBL5400597)
Affinity DataKi:  18nMAssay Description:Inhibition of Gst-tagged human Pin1 assessed as inhibition constant by Western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618840(CHEMBL5430490)
Affinity DataKi:  20nMAssay Description:Inhibition of Gst-tagged human Pin1 assessed as inhibition constant by Western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618867(CHEMBL5405065)
Affinity DataKi:  30nMAssay Description:Inhibition of Gst-tagged human Pin1 assessed as inhibition constant measured after 12 hrs by FP binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618866(CHEMBL5426583)
Affinity DataKi:  70nMAssay Description:Inhibition of Gst-tagged human Pin1 assessed as inhibition constant measured after 12 hrs by FP binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618865(CHEMBL5405609)
Affinity DataKi:  170nMAssay Description:Inhibition of Gst-tagged human Pin1 assessed as inhibition constant measured after 12 hrs by FP binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618841(CHEMBL5396492)
Affinity DataKi:  183nMAssay Description:Inhibition of Gst-tagged human Pin1 assessed as inhibition constant by Western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50381013(CHEMBL2017129)
Affinity DataKi:  200nMAssay Description:Inhibition of human Pin1 assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM92913(Aryl 1-indanylketone, 2)
Affinity DataKi:  400nMAssay Description:Inhibition of human Pin1 assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618862(CHEMBL5424015)
Affinity DataKi:  500nMAssay Description:Inhibition of human Pin1 assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618844(CHEMBL5416154)
Affinity DataKi:  507nMAssay Description:Inhibition of Gst-tagged human Pin1 assessed as inhibition constant by Western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50518736(CHEMBL4526940)
Affinity DataKi:  625nMAssay Description:Inhibition of recombinant human Pin1 assessed as inhibition constant measured upto 180 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618868(CHEMBL5397880)
Affinity DataKi:  700nMAssay Description:Inhibition of Gst-tagged human Pin1 assessed as inhibition constant measured after 14 hrs by FP binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618859(CHEMBL5408460)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of human Pin1 assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618860(CHEMBL5433705)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of human Pin1 assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618858(CHEMBL5410985)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of human Pin1 assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618834(CHEMBL5428388)
Affinity DataKi:  1.74E+3nMAssay Description:Inhibition of Pin1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618864(CHEMBL5413471)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of Gst-tagged human Pin1 assessed as inhibition constant measured after 12 hrs by FP binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618861(CHEMBL5409603)
Affinity DataKi:  3.10E+3nMAssay Description:Inhibition of human Pin1 assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM92914(Aryl 1-indanylketone, 3)
Affinity DataKi:  4.90E+3nMAssay Description:Inhibition of human Pin1 assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618855(CHEMBL5414741)
Affinity DataKi:  5.10E+3nMAssay Description:Inhibition of human Pin1 assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50437706(CHEMBL2409071)
Affinity DataKi:  5.60E+3nMAssay Description:Inhibition of human Pin1 assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618853(CHEMBL5417034)
Affinity DataKi:  6.20E+3nMAssay Description:Inhibition of human Pin1 assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618854(CHEMBL5393924)
Affinity DataKi:  8.70E+3nMAssay Description:Inhibition of human Pin1 assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618856(CHEMBL5394909)
Affinity DataKi:  1.50E+4nMAssay Description:Inhibition of human Pin1 assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM92917(Aryl 1-indanylketone, 6)
Affinity DataKi:  1.90E+4nMAssay Description:Inhibition of human Pin1 assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50618857(CHEMBL2409068)
Affinity DataKi:  5.10E+4nMAssay Description:Inhibition of human Pin1 assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed