Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50020171
Affinity DataKd: 110nMAssay Description:Binding affinity to CM5 chip immobilized GST-tagged mouse KEAP1 Kelch domain (322 to 624 residues) expressed in Escherichia coli BL21 (DE3) cells ass...More data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Inhibition of Keap1 Kelch domain (unknown origin)/FITC-labelled-9mer Nrf2 (unknown origin) protein-protein interaction incubated for 30 mins by fluor...More data for this Ligand-Target Pair
Affinity DataIC50: 750nMAssay Description:Inhibition of human Keap1 KELCH domain (321 to 609 residues) expressed in Escherichia coli BL21 DE3 pLysS cells/Nrf2 (unknown origin) protein-protein...More data for this Ligand-Target Pair
Affinity DataIC50: 890nMAssay Description:Inhibition of Keap1 Kelch domain (unknown origin)/FITC-labelled-9mer Nrf2 (unknown origin) protein-protein interaction incubated for 30 mins by fluor...More data for this Ligand-Target Pair
Affinity DataIC50: 3.16E+4nMAssay Description:Inhibition of Keap1 Kelch domain (unknown origin)/FITC-labelled-9mer Nrf2 (unknown origin) protein-protein interaction incubated for 30 mins by fluor...More data for this Ligand-Target Pair
Affinity DataKi: 95nMAssay Description:Inhibition of Keap1 (unknown origin)/Nrf2 (unknown origin) protein-protein interaction assessed as inhibition constant by fluorescence anisotropy ass...More data for this Ligand-Target Pair
3D Structure (crystal)