Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50022327
TargetEstrogen receptor(Human)
Zhengzhou Normal University

Curated by ChEMBL
LigandPNGBDBM50099585(1-[4-(2-Azepan-1-yl-ethoxy)-benzyl]-2-(4-hydroxy-p...)
Affinity DataIC50: 23nMAssay Description:Displacement of [3H]17 beta estradiol from human ERalpha by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetEstrogen receptor beta(Human)
Zhengzhou Normal University

Curated by ChEMBL
LigandPNGBDBM50099585(1-[4-(2-Azepan-1-yl-ethoxy)-benzyl]-2-(4-hydroxy-p...)
Affinity DataIC50: 99nMAssay Description:Displacement of [3H]17 beta estradiol from human ERbeta by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
Zhengzhou Normal University

Curated by ChEMBL
LigandPNGBDBM50094569(Cyproterone 17-O-acetate | cyproterone acetate | C...)
Affinity DataEC50:  4.00E+3nMAssay Description:Antagonist activity at AR (unknown origin) expressed in chemically activated Luciferase expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed