Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50020014
Affinity DataKd: 4.90nMAssay Description:Binding affinity to CDK13 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of GST-tagged recombinant human CDK12 (696 to 1082 residues) expressed in Insect cell in presence of ATP by Km ATP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of GST-tagged recombinant human CDK12 (696 to 1082 residues) expressed in Insect cell in presence of ATP by Km ATP assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 31nMAssay Description:Inhibition of GST-tagged recombinant human CDK12 (696 to 1082 residues) expressed in Insect cell in presence of ATP by Km ATP assayMore data for this Ligand-Target Pair
Affinity DataEC50: 32nMAssay Description:Inhibition of CDK12 in mouse OV2944-HM-1 cells by Westernblot analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataEC50: 35nMAssay Description:Inhibition of CDK12 in mouse OV2944-HM-1 cells by Westernblot analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 40nMAssay Description:Inhibition of full length recombinant human CDK2 expressed in Insect cell in presence of ATPMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 47nMAssay Description:Inhibition of GST-tagged recombinant human CDK12 (696 to 1082 residues) expressed in Insect cell in presence of ATP by high ATP assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 69nMAssay Description:Inhibition of recombinant human CDK13 expressed in baculovirus infected Insect cell measured after 30 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Affinity DataKd: 98nMAssay Description:Binding affinity to CDK12 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataIC50: 103nMAssay Description:Inhibition of GST-tagged recombinant human CDK12 (696 to 1082 residues) expressed in Insect cell in presence of ATP by high ATP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Inhibition of recombinant human CDK12 expressed in baculovirus infected Insect cell measured after 30 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 238nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 240nMAssay Description:Inhibition of full length recombinant human CDK9 expressed in Insect cell in presence of ATPMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 321nMAssay Description:Inhibition of full length recombinant human CDK2 expressed in Insect cell in presence of ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 468nMAssay Description:Inhibition of CDK12 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 491nMAssay Description:Inhibition of GST-tagged recombinant human CDK12 (696 to 1082 residues) expressed in Insect cell in presence of ATP by high ATP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 628nMAssay Description:Inhibition of CDK13 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 893nMAssay Description:Inhibition of CDK12 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 1.09E+3nMAssay Description:Inhibition of full length recombinant human CDK9 expressed in Insect cell in presence of ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 2.68E+3nMAssay Description:Inhibition of full length recombinant human CDK2 expressed in Insect cell in presence of ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 3.41E+3nMAssay Description:Inhibition of full length recombinant human CDK1 expressed in Insect cell in presence of ATPMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKd: 5.10E+3nMAssay Description:Binding affinity to CDK6 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibition of recombinant human CDK7 expressed in baculovirus infected Insect cell measured after 30 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 9.09E+3nMAssay Description:Inhibition of full length recombinant human CDK9 expressed in Insect cell in presence of ATPMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to CDK9 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibition of recombinant human CDK9 expressed in baculovirus infected Insect cell measured after 30 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.12E+4nMAssay Description:Inhibition of full length recombinant human CDK7 expressed in Insect cell in presence of ATPMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 2.86E+4nMAssay Description:Inhibition of full length recombinant human CDK1 expressed in Insect cell in presence of ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of full length recombinant human CDK7 expressed in Insect cell in presence of ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of full length recombinant human CDK1 expressed in Insect cell in presence of ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of full length recombinant human CDK7 expressed in Insect cell in presence of ATPMore data for this Ligand-Target Pair
