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Report error Found 38 Enz. Inhib. hit(s) with all data for entry = 50020356
TargetHeat shock protein HSP 90-beta(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50610097(CHEMBL5273198)
Affinity DataKd: >5.00E+4nMAssay Description:Binding affinity HSP90beta (unknown origin) assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50610097(CHEMBL5273198)
Affinity DataKd:  840nMAssay Description:Binding affinity HSP90alpha (unknown origin) assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetHeat shock protein HSP 90-alpha(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629230(CHEMBL5399553)
Affinity DataIC50: 340nMAssay Description:Binding affinity HSP90alpha (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629232(CHEMBL5437480)
Affinity DataIC50: 360nMAssay Description:Binding affinity HSP90alpha (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629227(CHEMBL5414316)
Affinity DataIC50: 510nMAssay Description:Binding affinity HSP90alpha (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629229(CHEMBL5404406)
Affinity DataIC50: 650nMAssay Description:Binding affinity HSP90alpha (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629228(CHEMBL5432073)
Affinity DataIC50: 790nMAssay Description:Binding affinity HSP90alpha (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629226(CHEMBL5400343)
Affinity DataIC50: 850nMAssay Description:Binding affinity HSP90alpha (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629239(CHEMBL5439550)
Affinity DataIC50: 960nMAssay Description:Binding affinity HSP90alpha (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629238(CHEMBL5400074)
Affinity DataIC50: 960nMAssay Description:Binding affinity HSP90alpha (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629231(CHEMBL5425276)
Affinity DataIC50: 7.36E+3nMAssay Description:Binding affinity HSP90alpha (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629234(CHEMBL5434857)
Affinity DataIC50: 7.94E+3nMAssay Description:Binding affinity HSP90alpha (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHeat shock protein HSP 90-beta(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629232(CHEMBL5437480)
Affinity DataIC50: 8.39E+3nMAssay Description:Binding affinity HSP90beta (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629236(CHEMBL5397907)
Affinity DataIC50: 4.31E+4nMAssay Description:Binding affinity HSP90alpha (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629237(CHEMBL5419640)
Affinity DataIC50: 9.03E+4nMAssay Description:Binding affinity HSP90alpha (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHeat shock protein HSP 90-beta(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629226(CHEMBL5400343)
Affinity DataIC50: 9.61E+4nMAssay Description:Binding affinity HSP90beta (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629230(CHEMBL5399553)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity to Trap1 (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629227(CHEMBL5414316)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity to Trap1 (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629226(CHEMBL5400343)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity to Trap1 (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetEndoplasmin(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629230(CHEMBL5399553)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity to Grp94 (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetEndoplasmin(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629229(CHEMBL5404406)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity to Grp94 (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetEndoplasmin(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629227(CHEMBL5414316)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity to Grp94 (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHeat shock protein 75 kDa, mitochondrial(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629229(CHEMBL5404406)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity to Trap1 (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetEndoplasmin(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629226(CHEMBL5400343)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity to Grp94 (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHeat shock protein HSP 90-beta(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629239(CHEMBL5439550)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity HSP90beta (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHeat shock protein HSP 90-beta(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629238(CHEMBL5400074)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity HSP90beta (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHeat shock protein HSP 90-beta(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629237(CHEMBL5419640)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity HSP90beta (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHeat shock protein HSP 90-beta(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629236(CHEMBL5397907)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity HSP90beta (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHeat shock protein HSP 90-beta(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629235(CHEMBL5398408)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity HSP90beta (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHeat shock protein HSP 90-beta(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629234(CHEMBL5434857)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity HSP90beta (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHeat shock protein HSP 90-beta(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629233(CHEMBL5398860)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity HSP90beta (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHeat shock protein HSP 90-beta(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629231(CHEMBL5425276)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity HSP90beta (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHeat shock protein HSP 90-beta(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629230(CHEMBL5399553)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity HSP90beta (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHeat shock protein HSP 90-beta(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629229(CHEMBL5404406)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity HSP90beta (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHeat shock protein HSP 90-beta(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629228(CHEMBL5432073)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity HSP90beta (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHeat shock protein HSP 90-beta(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629227(CHEMBL5414316)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity HSP90beta (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629235(CHEMBL5398408)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity HSP90alpha (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
The University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50629233(CHEMBL5398860)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity HSP90alpha (unknown origin) incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed