Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50020371
TargetKetohexokinase(Human)
Tuojie Biotech (Shanghai) Co.

Curated by ChEMBL
LigandPNGBDBM50629381(CHEMBL5427050)
Affinity DataIC50: 22nMAssay Description:Inhibition of N-terminal his tagged human recombinant KHK-C expressed in Escherichia coli incubated for 60 mins in presence of ATP by ADP Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetKetohexokinase(Human)
Tuojie Biotech (Shanghai) Co.

Curated by ChEMBL
LigandPNGBDBM50629389(CHEMBL5402452)
Affinity DataIC50: 26nMAssay Description:Inhibition of N-terminal his tagged human recombinant KHK-C expressed in Escherichia coli incubated for 60 mins in presence of ATP by ADP Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetKetohexokinase(Human)
Tuojie Biotech (Shanghai) Co.

Curated by ChEMBL
LigandPNGBDBM319585(US10174007, Example 4 | US10787438, Example 4 | US...)
Affinity DataIC50: 32nMAssay Description:Inhibition of N-terminal his tagged human recombinant KHK-C expressed in Escherichia coli incubated for 60 mins in presence of ATP by ADP Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetKetohexokinase(Human)
Tuojie Biotech (Shanghai) Co.

Curated by ChEMBL
LigandPNGBDBM50629382(CHEMBL5401360)
Affinity DataIC50: 35nMAssay Description:Inhibition of N-terminal his tagged human recombinant KHK-C expressed in Escherichia coli incubated for 60 mins in presence of ATP by ADP Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetKetohexokinase(Human)
Tuojie Biotech (Shanghai) Co.

Curated by ChEMBL
LigandPNGBDBM50629384(CHEMBL5408214)
Affinity DataIC50: 35nMAssay Description:Inhibition of N-terminal his tagged human recombinant KHK-C expressed in Escherichia coli incubated for 60 mins in presence of ATP by ADP Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetKetohexokinase(Human)
Tuojie Biotech (Shanghai) Co.

Curated by ChEMBL
LigandPNGBDBM50629383(CHEMBL5434549 | US20250145619, Example 36)
Affinity DataIC50: 49nMAssay Description:Inhibition of N-terminal his tagged human recombinant KHK-C expressed in Escherichia coli incubated for 60 mins in presence of ATP by ADP Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetKetohexokinase(Human)
Tuojie Biotech (Shanghai) Co.

Curated by ChEMBL
LigandPNGBDBM50629385(CHEMBL5411144)
Affinity DataIC50: 54nMAssay Description:Inhibition of N-terminal his tagged human recombinant KHK-C expressed in Escherichia coli incubated for 60 mins in presence of ATP by ADP Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetKetohexokinase(Human)
Tuojie Biotech (Shanghai) Co.

Curated by ChEMBL
LigandPNGBDBM50629384(CHEMBL5408214)
Affinity DataIC50: 57nMAssay Description:Inhibition of N-terminal his tagged human recombinant KHK-A expressed in Escherichia coli incubated for 60 mins in presence of ATP by ADP Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetKetohexokinase(Human)
Tuojie Biotech (Shanghai) Co.

Curated by ChEMBL
LigandPNGBDBM50629386(CHEMBL5407523)
Affinity DataIC50: 90nMAssay Description:Inhibition of N-terminal his tagged human recombinant KHK-C expressed in Escherichia coli incubated for 60 mins in presence of ATP by ADP Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetKetohexokinase(Human)
Tuojie Biotech (Shanghai) Co.

Curated by ChEMBL
LigandPNGBDBM50629376(CHEMBL5419385)
Affinity DataIC50: 108nMAssay Description:Inhibition of N-terminal his tagged human recombinant KHK-C expressed in Escherichia coli incubated for 60 mins in presence of ATP by ADP Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetKetohexokinase(Human)
Tuojie Biotech (Shanghai) Co.

Curated by ChEMBL
LigandPNGBDBM50629378(CHEMBL5408159)
Affinity DataIC50: 108nMAssay Description:Inhibition of N-terminal his tagged human recombinant KHK-C expressed in Escherichia coli incubated for 60 mins in presence of ATP by ADP Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetKetohexokinase(Human)
Tuojie Biotech (Shanghai) Co.

Curated by ChEMBL
LigandPNGBDBM319585(US10174007, Example 4 | US10787438, Example 4 | US...)
Affinity DataIC50: 111nMAssay Description:Inhibition of N-terminal his tagged human recombinant KHK-A expressed in Escherichia coli incubated for 60 mins in presence of ATP by ADP Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetKetohexokinase(Human)
Tuojie Biotech (Shanghai) Co.

Curated by ChEMBL
LigandPNGBDBM50629375(CHEMBL5431020)
Affinity DataIC50: 138nMAssay Description:Inhibition of N-terminal his tagged human recombinant KHK-C expressed in Escherichia coli incubated for 60 mins in presence of ATP by ADP Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetKetohexokinase(Human)
Tuojie Biotech (Shanghai) Co.

Curated by ChEMBL
LigandPNGBDBM50629380(CHEMBL5430902 | US20250145619, Example 6)
Affinity DataIC50: 280nMAssay Description:Inhibition of N-terminal his tagged human recombinant KHK-C expressed in Escherichia coli incubated for 60 mins in presence of ATP by ADP Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetKetohexokinase(Human)
Tuojie Biotech (Shanghai) Co.

Curated by ChEMBL
LigandPNGBDBM50629387(CHEMBL5440941)
Affinity DataIC50: 849nMAssay Description:Inhibition of N-terminal his tagged human recombinant KHK-C expressed in Escherichia coli incubated for 60 mins in presence of ATP by ADP Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetKetohexokinase(Human)
Tuojie Biotech (Shanghai) Co.

Curated by ChEMBL
LigandPNGBDBM50629388(CHEMBL5433776)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of N-terminal his tagged human recombinant KHK-C expressed in Escherichia coli incubated for 60 mins in presence of ATP by ADP Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetKetohexokinase(Human)
Tuojie Biotech (Shanghai) Co.

Curated by ChEMBL
LigandPNGBDBM50629379(CHEMBL5415431)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of N-terminal his tagged human recombinant KHK-C expressed in Escherichia coli incubated for 60 mins in presence of ATP by ADP Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetKetohexokinase(Human)
Tuojie Biotech (Shanghai) Co.

Curated by ChEMBL
LigandPNGBDBM50629377(CHEMBL5424828)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of N-terminal his tagged human recombinant KHK-C expressed in Escherichia coli incubated for 60 mins in presence of ATP by ADP Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
Tuojie Biotech (Shanghai) Co.

Curated by ChEMBL
LigandPNGBDBM319585(US10174007, Example 4 | US10787438, Example 4 | US...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human Nav1.5 by manual-patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
Tuojie Biotech (Shanghai) Co.

Curated by ChEMBL
LigandPNGBDBM50629384(CHEMBL5408214)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human Nav1.5 by manual-patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed