Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50022439
TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Guizhou University

Curated by ChEMBL
LigandPNGBDBM431795(US10550105, Example 661)
Affinity DataKd:  0.220nMAssay Description:Binding affinity to PARP7 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Ligand InfoPDBSimilars
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Guizhou University

Curated by ChEMBL
LigandPNGBDBM700586(US20240336629, Compound 89A)
Affinity DataIC50: 0.560nMAssay Description:Inhibition of PARP7 (unknown origin) using histone as substrate incubated for 1 hr by chemiluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Guizhou University

Curated by ChEMBL
LigandPNGBDBM50652258(CHEMBL5647433)
Affinity DataIC50: 0.660nMAssay Description:Inhibition of PARP7 (unknown origin) using histone as substrate incubated for 1 hr by chemiluminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Guizhou University

Curated by ChEMBL
LigandPNGBDBM50652255(CHEMBL5646537)
Affinity DataIC50: 0.710nMAssay Description:Inhibition of PARP7 (unknown origin) using histone as substrate incubated for 1 hr by chemiluminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Guizhou University

Curated by ChEMBL
LigandPNGBDBM50652254(CHEMBL5647333)
Affinity DataIC50: 0.970nMAssay Description:Inhibition of PARP7 (unknown origin) using histone as substrate incubated for 1 hr by chemiluminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Guizhou University

Curated by ChEMBL
LigandPNGBDBM50595885(CHEMBL5183278 | US20240336629, Compound 51)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of PARP7 (unknown origin) using histone as substrate incubated for 1 hr by chemiluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Guizhou University

Curated by ChEMBL
LigandPNGBDBM700510(US20240336629, Compound 53B)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of PARP7 (unknown origin) using histone as substrate incubated for 1 hr by chemiluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Guizhou University

Curated by ChEMBL
LigandPNGBDBM700508(US20240336629, Compound 53)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of PARP7 (unknown origin) using histone as substrate incubated for 1 hr by chemiluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Guizhou University

Curated by ChEMBL
LigandPNGBDBM431795(US10550105, Example 661)
Affinity DataIC50: 3nMAssay Description:Inhibition of PARP7 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPDBSimilars
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Guizhou University

Curated by ChEMBL
LigandPNGBDBM431795(US10550105, Example 661)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of PARP7 (unknown origin) using histone as substrate incubated for 1 hr by chemiluminescence assayMore data for this Ligand-Target Pair
Ligand InfoPDBSimilars
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Guizhou University

Curated by ChEMBL
LigandPNGBDBM700509(US20240336629, Compound 53A)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of PARP7 (unknown origin) using histone as substrate incubated for 1 hr by chemiluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Guizhou University

Curated by ChEMBL
LigandPNGBDBM50652253(CHEMBL5639739)
Affinity DataIC50: 9.40nMAssay Description:Inhibition of PARP7 (unknown origin) using histone as substrate incubated for 1 hr by chemiluminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Guizhou University

Curated by ChEMBL
LigandPNGBDBM50652251(CHEMBL5646699)
Affinity DataIC50: 10nMAssay Description:Inhibition of PARP7 (unknown origin) using histone as substrate incubated for 1 hr by chemiluminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Guizhou University

Curated by ChEMBL
LigandPNGBDBM50652252(CHEMBL5639651)
Affinity DataIC50: 13nMAssay Description:Inhibition of PARP7 (unknown origin) using histone as substrate incubated for 1 hr by chemiluminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Guizhou University

Curated by ChEMBL
LigandPNGBDBM50652256(CHEMBL5646565)
Affinity DataIC50: 14nMAssay Description:Inhibition of PARP7 (unknown origin) using histone as substrate incubated for 1 hr by chemiluminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Guizhou University

Curated by ChEMBL
LigandPNGBDBM50652257(CHEMBL5647306)
Affinity DataIC50: 63nMAssay Description:Inhibition of PARP7 (unknown origin) using histone as substrate incubated for 1 hr by chemiluminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPoly [ADP-ribose] polymerase 2(Human)
Guizhou University

Curated by ChEMBL
LigandPNGBDBM700586(US20240336629, Compound 89A)
Affinity DataIC50: 221nMAssay Description:Inhibition of PARP2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein mono-ADP-ribosyltransferase PARP12(Human)
Guizhou University

Curated by ChEMBL
LigandPNGBDBM700586(US20240336629, Compound 89A)
Affinity DataIC50: 360nMAssay Description:Inhibition of PARP12 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Guizhou University

Curated by ChEMBL
LigandPNGBDBM700586(US20240336629, Compound 89A)
Affinity DataIC50: 492nMAssay Description:Inhibition of PARP1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
Guizhou University

Curated by ChEMBL
LigandPNGBDBM700586(US20240336629, Compound 89A)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PARP14 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein mono-ADP-ribosyltransferase PARP11(Human)
Guizhou University

Curated by ChEMBL
LigandPNGBDBM700586(US20240336629, Compound 89A)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PARP11 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed