Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50022446
TargetSerine/threonine-protein kinase DCLK1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50539944(CHEMBL4639395)
Affinity DataIC50: 38nMAssay Description:Inhibition of DCLK1 (unknown origin) preincubated for 10 mins followed by substrate/ATP addition measured after 60 mins by mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase DCLK1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50539944(CHEMBL4639395)
Affinity DataIC50: 57nMAssay Description:Inhibition of DCLK1 (unknown origin) in presence of 33P-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase DCLK1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50652324(CHEMBL5639361)
Affinity DataIC50: 171nMAssay Description:Inhibition of DCLK1 (unknown origin) preincubated for 10 mins followed by substrate/ATP addition measured after 60 mins by mobility shift assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase DCLK1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM482158(TAE684 | BDBM50242742)
Affinity DataIC50: 1.08E+3nMAssay Description:Inhibition of DCLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMedPDB3D3D Structure (crystal)