Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50021596
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
Chongqing Medical and Pharmaceutical College

Curated by ChEMBL
LigandPNGBDBM50236535(CHEMBL1231132)
Affinity DataKd:  148nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
Chongqing Medical and Pharmaceutical College

Curated by ChEMBL
LigandPNGBDBM50236535(CHEMBL1231132)
Affinity DataKd:  8.90E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
Chongqing Medical and Pharmaceutical College

Curated by ChEMBL
LigandPNGBDBM50414944(NSC-402538 | CHEMBL121556)
Affinity DataEC50:  49nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
Chongqing Medical and Pharmaceutical College

Curated by ChEMBL
LigandPNGBDBM50236535(CHEMBL1231132)
Affinity DataIC50: 32nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
Chongqing Medical and Pharmaceutical College

Curated by ChEMBL
LigandPNGBDBM50642384(CHEMBL5574690)
Affinity DataIC50: 40nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
Chongqing Medical and Pharmaceutical College

Curated by ChEMBL
LigandPNGBDBM50642383(CHEMBL5575203)
Affinity DataIC50: 60nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial(Human)
Chongqing Medical and Pharmaceutical College

Curated by ChEMBL
LigandPNGBDBM50236535(CHEMBL1231132)
Affinity DataIC50: 75nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
Chongqing Medical and Pharmaceutical College

Curated by ChEMBL
LigandPNGBDBM50642382(CHEMBL5563199)
Affinity DataIC50: 109nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 3, mitochondrial(Human)
Chongqing Medical and Pharmaceutical College

Curated by ChEMBL
LigandPNGBDBM50236535(CHEMBL1231132)
Affinity DataIC50: 121nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial(Human)
Chongqing Medical and Pharmaceutical College

Curated by ChEMBL
LigandPNGBDBM50642382(CHEMBL5563199)
Affinity DataIC50: 136nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 3, mitochondrial(Human)
Chongqing Medical and Pharmaceutical College

Curated by ChEMBL
LigandPNGBDBM50642382(CHEMBL5563199)
Affinity DataIC50: 459nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Human)
Chongqing Medical and Pharmaceutical College

Curated by ChEMBL
LigandPNGBDBM50236535(CHEMBL1231132)
Affinity DataIC50: 540nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Human)
Chongqing Medical and Pharmaceutical College

Curated by ChEMBL
LigandPNGBDBM50642382(CHEMBL5563199)
Affinity DataIC50: 8.67E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed