Compile Data Set for Download or QSAR
Report error Found 56 Enz. Inhib. hit(s) with all data for entry = 50020528
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630861(CHEMBL5421312)
Affinity DataIC50: 90nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630877(CHEMBL5409469)
Affinity DataIC50: 120nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630902(CHEMBL5424031)
Affinity DataIC50: 120nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630860(CHEMBL5397445)
Affinity DataIC50: 120nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630903(CHEMBL5401872)
Affinity DataIC50: 130nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630882(CHEMBL5405109)
Affinity DataIC50: 240nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630904(CHEMBL5394108)
Affinity DataIC50: 260nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630868(CHEMBL5423748)
Affinity DataIC50: 270nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50425732(Xtandi | ENZALUTAMIDE | US10053433, FC 4.129 | US1...)
Affinity DataIC50: 340nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630853(CHEMBL5423482)
Affinity DataIC50: 600nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630869(CHEMBL5430613)
Affinity DataIC50: 600nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630856(CHEMBL5395364)
Affinity DataIC50: 700nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630873(CHEMBL5431700)
Affinity DataIC50: 760nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630864(CHEMBL5394445)
Affinity DataIC50: 800nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630865(CHEMBL5395976)
Affinity DataIC50: 800nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630900(CHEMBL5416300)
Affinity DataIC50: 800nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630859(CHEMBL5416819)
Affinity DataIC50: 920nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630896(CHEMBL5433104)
Affinity DataIC50: 940nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630858(CHEMBL5440496)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630884(CHEMBL5395092)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630854(CHEMBL5439835)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630905(CHEMBL5429958)
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630889(CHEMBL5405995)
Affinity DataIC50: 8.60E+3nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630857(CHEMBL5416202)
Affinity DataIC50: 1.03E+4nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630890(CHEMBL5437444)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630880(CHEMBL5420557)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630891(CHEMBL5425494)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630888(CHEMBL5421175)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630892(CHEMBL5404749)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630893(CHEMBL5405113)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630894(CHEMBL5410172)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630895(CHEMBL5416732)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630897(CHEMBL5408281)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630898(CHEMBL5413307)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630899(CHEMBL5437053)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630901(CHEMBL5405492)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630886(CHEMBL5431055)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630855(CHEMBL5441048)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630862(CHEMBL5426257)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630863(CHEMBL5427342)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630866(CHEMBL5430251)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630867(CHEMBL5428152)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630870(CHEMBL5418252)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630871(CHEMBL5435133)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630872(CHEMBL5439280)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630874(CHEMBL5417385)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630875(CHEMBL5423296)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630876(CHEMBL5415715)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630878(CHEMBL5440505)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAndrogen receptor(Human)
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50630879(CHEMBL5427904)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of androgen receptor in human VCaP cells expressing GRE-2-TATA-Luc co-expressing firefly luciferase incubated for 24 hrs in presence of DH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
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