Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50020061
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50318486(CHEMBL422704 | 2-Methyl-2-(4-methyl-pent-3-enyl)-7...)
Affinity DataEC50:  90nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetCannabinoid receptor 2(Human)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50318486(CHEMBL422704 | 2-Methyl-2-(4-methyl-pent-3-enyl)-7...)
Affinity DataKi:  260nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in Sf9 cell membranes assessed as inhibition constant incubated for 90 mins by by scint...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetCannabinoid receptor 1(Human)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50318486(CHEMBL422704 | 2-Methyl-2-(4-methyl-pent-3-enyl)-7...)
Affinity DataKi:  710nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in Sf9 cell membranes assessed as inhibition constant incubated for 90 mins by by scint...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed