Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50021258
TargetShort transient receptor potential channel 6(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50638826(CHEMBL5567030)
Affinity DataIC50: 0.220nMAssay Description:Antagonist activity at TRPC6 (unknown origin) assessed as inhibition of channel activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetShort transient receptor potential channel 3(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50439217(CHEMBL2418811)
Affinity DataIC50: 3nMAssay Description:Antagonist activity at TRPC3 (unknown origin) assessed as inhibition of channel activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetShort transient receptor potential channel 6(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50439218(CHEMBL2418809)
Affinity DataIC50: 4nMAssay Description:Antagonist activity at TRPC6 (unknown origin) assessed as inhibition of channel activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetShort transient receptor potential channel 3(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50439218(CHEMBL2418809)
Affinity DataIC50: 5nMAssay Description:Antagonist activity at TRPC3 (unknown origin) assessed as inhibition of channel activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetShort transient receptor potential channel 6(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50638825(CHEMBL5532633)
Affinity DataIC50: 5.80nMAssay Description:Antagonist activity at TRPC6 (unknown origin) assessed as inhibition of channel activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetShort transient receptor potential channel 6(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50273009(CHEMBL4129809)
Affinity DataIC50: 7.90nMAssay Description:Antagonist activity at TRPC6 (unknown origin) assessed as inhibition of channel activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetShort transient receptor potential channel 3(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50638824(CHEMBL5558723)
Affinity DataIC50: 10nMAssay Description:Antagonist activity at TRPC3 (unknown origin) assessed as inhibition of channel activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetShort transient receptor potential channel 6(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50638824(CHEMBL5558723)
Affinity DataIC50: 10nMAssay Description:Antagonist activity at TRPC6 (unknown origin) assessed as inhibition of channel activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetShort transient receptor potential channel 6(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50638822(CHEMBL5567783)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at TRPC6 (unknown origin) assessed as inhibition of channel activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetShort transient receptor potential channel 6(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50439217(CHEMBL2418811)
Affinity DataIC50: 21nMAssay Description:Antagonist activity at TRPC6 (unknown origin) assessed as inhibition of channel activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetShort transient receptor potential channel 3(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50450629(CHEMBL4177187)
Affinity DataIC50: 700nMAssay Description:Antagonist activity at TRPC3 (unknown origin) assessed as inhibition of channel activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetShort transient receptor potential channel 3(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50638825(CHEMBL5532633)
Affinity DataIC50: 840nMAssay Description:Antagonist activity at TRPC3 (unknown origin) assessed as inhibition of channel activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetShort transient receptor potential channel 6(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50638823(CHEMBL5561836)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at TRPC6 (unknown origin) assessed as inhibition of channel activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetShort transient receptor potential channel 3(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50638821(CHEMBL5561986)
Affinity DataIC50: 2.40E+3nMAssay Description:Antagonist activity at human TRPC3 stably expressed in HEK293 cells inhibition of calcium influx by calcium fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetShort transient receptor potential channel 6(Mouse)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50638821(CHEMBL5561986)
Affinity DataIC50: 2.90E+3nMAssay Description:Antagonist activity at mouse TRPC6 stably expressed in HEK293 cells inhibition of calcium influx by calcium fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetShort transient receptor potential channel 7(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50638821(CHEMBL5561986)
Affinity DataIC50: 3.40E+3nMAssay Description:Antagonist activity at human TRPC7 stably expressed in HEK293 cells inhibition of calcium influx by calcium fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetShort transient receptor potential channel 6(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50638827(CHEMBL1740853)
Affinity DataIC50: 4.20E+3nMAssay Description:Antagonist activity at TRPC6 (unknown origin) assessed as inhibition of channel activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetShort transient receptor potential channel 6(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50046268(6-[1-Bromo-meth-(E)-ylidene]-3-naphthalen-1-yl-tet...)
Affinity DataIC50: 7.20E+3nMAssay Description:Antagonist activity at TRPC6 (unknown origin) assessed as inhibition of channel activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50638821(CHEMBL5561986)
Affinity DataIC50: 7.60E+3nMAssay Description:Antagonist activity at human TRPC5 stably expressed in HEK293 cells inhibition of calcium influx by calcium fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetShort transient receptor potential channel 5(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50046268(6-[1-Bromo-meth-(E)-ylidene]-3-naphthalen-1-yl-tet...)
Affinity DataIC50: 1.06E+4nMAssay Description:Antagonist activity at TRPC5 (unknown origin) assessed as inhibition of channel activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetShort transient receptor potential channel 4(Mouse)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50638821(CHEMBL5561986)
Affinity DataIC50: 1.22E+4nMAssay Description:Antagonist activity at mouse TRPC4 stably expressed in HEK293 cells inhibition of calcium influx by calcium fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed