Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50021688
TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Hubei Polytechnic University

Curated by ChEMBL
LigandPNGBDBM700589(US20240336629, Compound 90B)
Affinity DataIC50: 0.110nMAssay Description:Inhibition of PARP7 (unknown origin) incubated for 1 hr by chemiluminescence based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Hubei Polytechnic University

Curated by ChEMBL
LigandPNGBDBM700540(US20240336629, Compound 67A)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of PARP7 (unknown origin) incubated for 1 hr by chemiluminescence based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Hubei Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50643508(CHEMBL5568973)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of PARP7 (unknown origin) incubated for 1 hr by chemiluminescence based microplate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Hubei Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50643507(CHEMBL5569182)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of PARP7 (unknown origin) incubated for 1 hr by chemiluminescence based microplate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Hubei Polytechnic University

Curated by ChEMBL
LigandPNGBDBM700588(US20240336629, Compound 90A)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of PARP7 (unknown origin) incubated for 1 hr by chemiluminescence based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Hubei Polytechnic University

Curated by ChEMBL
LigandPNGBDBM700515(US20240336629, Compound 55B)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of PARP7 (unknown origin) incubated for 1 hr by chemiluminescence based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Hubei Polytechnic University

Curated by ChEMBL
LigandPNGBDBM700543(US20240336629, Compound 68B)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of PARP7 (unknown origin) incubated for 1 hr by chemiluminescence based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Hubei Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50643505(CHEMBL5572070)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of PARP7 (unknown origin) incubated for 1 hr by chemiluminescence based microplate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Hubei Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50643506(CHEMBL5592550)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of PARP7 (unknown origin) incubated for 1 hr by chemiluminescence based microplate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Hubei Polytechnic University

Curated by ChEMBL
LigandPNGBDBM431795(US10550105, Example 661)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of PARP7 (unknown origin) incubated for 1 hr by chemiluminescence based microplate reader assayMore data for this Ligand-Target Pair
Ligand InfoPDBSimilars
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Hubei Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50643509(CHEMBL5572774)
Affinity DataIC50: 5.70nMAssay Description:Inhibition of PARP7 (unknown origin) incubated for 1 hr by chemiluminescence based microplate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Hubei Polytechnic University

Curated by ChEMBL
LigandPNGBDBM700514(US20240336629, Compound 55A)
Affinity DataIC50: 7.30nMAssay Description:Inhibition of PARP7 (unknown origin) incubated for 1 hr by chemiluminescence based microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Hubei Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50643510(CHEMBL5575060)
Affinity DataIC50: 7.90nMAssay Description:Inhibition of PARP7 (unknown origin) incubated for 1 hr by chemiluminescence based microplate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPoly [ADP-ribose] polymerase 2(Human)
Hubei Polytechnic University

Curated by ChEMBL
LigandPNGBDBM431795(US10550105, Example 661)
Affinity DataIC50: 17nMAssay Description:Inhibition of PARP2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPDBSimilars
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein mono-ADP-ribosyltransferase TIPARP(Human)
Hubei Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50643511(CHEMBL5565931)
Affinity DataIC50: 37nMAssay Description:Inhibition of PARP7 (unknown origin) incubated for 1 hr by chemiluminescence based microplate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein mono-ADP-ribosyltransferase PARP14(Human)
Hubei Polytechnic University

Curated by ChEMBL
LigandPNGBDBM700589(US20240336629, Compound 90B)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PARP14 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein mono-ADP-ribosyltransferase PARP12(Human)
Hubei Polytechnic University

Curated by ChEMBL
LigandPNGBDBM700589(US20240336629, Compound 90B)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PARP12 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein mono-ADP-ribosyltransferase PARP11(Human)
Hubei Polytechnic University

Curated by ChEMBL
LigandPNGBDBM700589(US20240336629, Compound 90B)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PARP11 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Hubei Polytechnic University

Curated by ChEMBL
LigandPNGBDBM700589(US20240336629, Compound 90B)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PARP1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPoly [ADP-ribose] polymerase 2(Human)
Hubei Polytechnic University

Curated by ChEMBL
LigandPNGBDBM700589(US20240336629, Compound 90B)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PARP2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPoly [ADP-ribose] polymerase 2(Human)
Hubei Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50643505(CHEMBL5572070)
Affinity DataIC50: 2.09E+3nMAssay Description:Inhibition of PARP2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPoly [ADP-ribose] polymerase 2(Human)
Hubei Polytechnic University

Curated by ChEMBL
LigandPNGBDBM700543(US20240336629, Compound 68B)
Affinity DataIC50: 2.32E+3nMAssay Description:Inhibition of PARP2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPoly [ADP-ribose] polymerase 2(Human)
Hubei Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50643506(CHEMBL5592550)
Affinity DataIC50: 2.57E+3nMAssay Description:Inhibition of PARP2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed