Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with all data for entry = 50019770
TargetTyrosine-protein kinase BTK(Human)
Nurix Therapeutics

Curated by ChEMBL
LigandPNGBDBM50622926(CHEMBL5435454)
Affinity DataKd:  45nMAssay Description:Binding affinity to BTK (unknown origin) assessed as dissociation constant by surface plasmon resonance assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Nurix Therapeutics

Curated by ChEMBL
LigandPNGBDBM50622926(CHEMBL5435454)
Affinity DataKd:  18nMAssay Description:Binding affinity to BTK C481S mutant (unknown origin) assessed as dissociation constant by surface plasmon resonance assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed