Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50019604
TargetEpidermal growth factor receptor(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50620941(CHEMBL5423287)
Affinity DataIC50: 33nMAssay Description:Inhibition of EGFR L858R/T790M/C797S mutant (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50620938(CHEMBL5440989)
Affinity DataIC50: 45nMAssay Description:Inhibition of EGFR L858R/T790M/C797S mutant (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50620937(CHEMBL5439991)
Affinity DataIC50: 52nMAssay Description:Inhibition of EGFR L858R/T790M/C797S mutant (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50185140(AP-26113 | Brigatinib | US11248003, Example Brigat...)
Affinity DataIC50: 53nMAssay Description:Inhibition of EGFR L858R/T790M/C797S mutant (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetEpidermal growth factor receptor(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50620939(CHEMBL5435881)
Affinity DataIC50: 70nMAssay Description:Inhibition of EGFR L858R/T790M/C797S mutant (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50620940(CHEMBL5435735)
Affinity DataIC50: 72nMAssay Description:Inhibition of EGFR L858R/T790M/C797S mutant (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed