Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50019624
Affinity DataKd: 243nMAssay Description:Binding affinity to LSD1 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataKd: 385nMAssay Description:Binding affinity to LSD1 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of EGFR L858R mutant (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of HDAC6 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Inhibition of LSD1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of HDAC6 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 210nMAssay Description:Inhibition of HDAC1 (unknown origin) by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 288nMAssay Description:Inhibition of human recombinant LSD1More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 290nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 540nMAssay Description:Inhibition of N-terminal human recombinant LSD1More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 570nMAssay Description:Inhibition of human recombinant HDAC3 incubated for 60 mins by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Inhibition of human N-terminal His-tagged LSD1 using histone H3 peptide (1 to 21 residues) K4me2 as substrate preincubated for 30 mins followed by su...More data for this Ligand-Target Pair
Affinity DataIC50: 778nMAssay Description:Inhibition of human G9a expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.12E+3nMAssay Description:Inhibition of human recombinant HDAC2 incubated for 60 mins by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human recombinant HDAC1 using fluorogenic HDAC substrate incubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.98E+3nMAssay Description:Inhibition of human recombinant LSD1 expressed in Escherichia coli BL21 (DE3) using H3K4me2 peptide as substrate incubated for 30 mins by fluorescenc...More data for this Ligand-Target Pair
Affinity DataIC50: 2.57E+4nMAssay Description:Inhibition of SMOX (unknown origin) using spermine as substrate preincubated for 1 hr followed by substrate addition and measured after 20 mins by lu...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 4.13E+4nMAssay Description:Inhibition of human G9a expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 440nMAssay Description:Binding affinity to LSD1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 1.06E+3nMAssay Description:Binding affinity to LSD1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
