Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50021763
TargetMixed lineage kinase domain-like protein(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50306682((R)-3-(1-(2,6-dichloro-3-fluorophenyl)ethoxy)-5-(1...)
Affinity DataKd:  217nMAssay Description:Binding affinity to NF-kappaB DNA binding domain fused full length human MLKL expressed in HEK293 cells assessed as dissociation constant by competit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetMixed lineage kinase domain-like protein(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50519647(CHEMBL4440337)
Affinity DataKd:  230nMAssay Description:Binding affinity to NF-kappaB DNA binding domain fused full length human MLKL expressed in HEK293 cells assessed as dissociation constant by competit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50306682((R)-3-(1-(2,6-dichloro-3-fluorophenyl)ethoxy)-5-(1...)
Affinity DataKd:  1.00E+3nMAssay Description:Binding affinity to RIPK1 (unknown origin) assessed as dissociation constant by displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 3(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50306682((R)-3-(1-(2,6-dichloro-3-fluorophenyl)ethoxy)-5-(1...)
Affinity DataKd:  7.00E+3nMAssay Description:Binding affinity to RIPK3 (unknown origin) assessed as dissociation constant by displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50519647(CHEMBL4440337)
Affinity DataKd: >3.00E+4nMAssay Description:Binding affinity to RIPK1 (unknown origin) assessed as dissociation constant by displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 3(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50519647(CHEMBL4440337)
Affinity DataKd: >3.00E+4nMAssay Description:Binding affinity to RIPK3 (unknown origin) assessed as dissociation constant by displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed