Compile Data Set for Download or QSAR
Report error Found 31 Enz. Inhib. hit(s) with all data for entry = 50021166
TargetTyrosine-protein kinase ABL1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50637644(CHEMBL5560252)
Affinity DataIC50: 0.179nMAssay Description:Inhibition of ABL (unknown origin) using Try-2 as substrate by FRET analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50511486(CHEMBL4559959)
Affinity DataKd:  2.20nMAssay Description:Binding affinity to DDR1 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetDiscoidin domain-containing receptor 2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50637642(CHEMBL5542762)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of flag-tagged DDR2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50637644(CHEMBL5560252)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of DDR1 (unknown origin) using Fluorescein-Poly GAT as substrate by TR-FRET analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50368455(CHEMBL4175086)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of DDR1 (unknown origin) by DiscoverX KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetDiscoidin domain-containing receptor 2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50637645(CHEMBL5537027)
Affinity DataIC50: 4.80nMAssay Description:Inhibition of DDR2 (unknown origin) by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetDiscoidin domain-containing receptor 2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM603901(US11655239, Compound S15)
Affinity DataIC50: 6.10nMAssay Description:Inhibition of flag-tagged DDR2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50511486(CHEMBL4559959)
Affinity DataIC50: 6.60nMAssay Description:Inhibition of DDR1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50430839(CHEMBL2336015)
Affinity DataIC50: 6.80nMAssay Description:Inhibition of DDR1 (unknown origin) by DiscoverX KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetDiscoidin domain-containing receptor 2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50637644(CHEMBL5560252)
Affinity DataIC50: 7nMAssay Description:Inhibition of DDR2 (unknown origin) using Fluorescein-Poly GAT as substrate by TR-FRET analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetDiscoidin domain-containing receptor 2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50368455(CHEMBL4175086)
Affinity DataIC50: 7nMAssay Description:Inhibition of DDR2 (unknown origin) by by DiscoverX KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50368455(CHEMBL4175086)
Affinity DataIC50: 9.40nMAssay Description:Inhibition of ABL (unknown origin) incubated for 1 hr by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50637638(CHEMBL5568512)
Affinity DataIC50: 10nMAssay Description:Inhibition of DDR1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50637641(CHEMBL5559968)
Affinity DataIC50: 10nMAssay Description:Inhibition of GST-tagged recombinant DDR1 (unknown origin) expressed in Escherichia coli BL21 by DiscoverX KINOMEscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50637639(CHEMBL5563319)
Affinity DataIC50: 11nMAssay Description:Inhibition of DDR1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50297825(5-[(2-methyl-5-{[3-(trifluoromethyl)phenyl]carbamo...)
Affinity DataIC50: 12nMAssay Description:Inhibition of DDR1 (unknown origin) by TR-FRET based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM371830(2-(8-(1H-Indazole-5-carbonyl)-4-oxo-1-phenyl-1,3,8...)
Affinity DataIC50: 15nMAssay Description:Inhibition of GST-tagged recombinant DDR1 (unknown origin) expressed in Escherichia coli BL21 by DiscoverX KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM603901(US11655239, Compound S15)
Affinity DataIC50: 17nMAssay Description:Inhibition of flag-tagged DDR1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM372068(2-(4-Oxo-1-phenyl-8-(1H-pyrazolo[4,3-b]pyridine-5-...)
Affinity DataIC50: 18nMAssay Description:Inhibition of GST-tagged recombinant DDR1 (unknown origin) expressed in Escherichia coli BL21 by DiscoverX KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetDiscoidin domain-containing receptor 2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50297825(5-[(2-methyl-5-{[3-(trifluoromethyl)phenyl]carbamo...)
Affinity DataIC50: 19nMAssay Description:Inhibition of DDR2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM438155(US10618897, Example 23)
Affinity DataIC50: 29nMAssay Description:Inhibition of GST-tagged recombinant DDR1 (unknown origin) expressed in Escherichia coli BL21 by DiscoverX KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetDiscoidin domain-containing receptor 2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50637643(CHEMBL5555076)
Affinity DataIC50: 31nMAssay Description:Inhibition of human DDR2 by discoverX kinome scan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50637640(CHEMBL5558279)
Affinity DataIC50: 93nMAssay Description:Inhibition of DDR1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetDiscoidin domain-containing receptor 2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50430839(CHEMBL2336015)
Affinity DataIC50: 101nMAssay Description:Inhibition of DDR2 (unknown origin) by by DiscoverX KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM104009(DDR1-IN-1)
Affinity DataIC50: 105nMAssay Description:Inhibition of DDR1 (unknown origin) (601 to 913 residues) expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetTyrosine-protein kinase ABL1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50430839(CHEMBL2336015)
Affinity DataIC50: 355nMAssay Description:Inhibition of ABL (unknown origin) incubated for 1 hr by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetDiscoidin domain-containing receptor 2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM371830(2-(8-(1H-Indazole-5-carbonyl)-4-oxo-1-phenyl-1,3,8...)
Affinity DataIC50: 820nMAssay Description:Inhibition of GST-tagged recombinant DDR2 (unknown origin) expressed in Escherichia coli BL21 by DiscoverX KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetDiscoidin domain-containing receptor 2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM372068(2-(4-Oxo-1-phenyl-8-(1H-pyrazolo[4,3-b]pyridine-5-...)
Affinity DataIC50: 858nMAssay Description:Inhibition of GST-tagged recombinant DDR2 (unknown origin) expressed in Escherichia coli BL21 by DiscoverX KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM371924(2-[8-(1H-Indazole-5-carbonyl)-4-oxo-1-phenyl-1,3,8...)
Affinity DataIC50: 1.41E+3nMAssay Description:Inhibition of GST-tagged recombinant DDR1 (unknown origin) expressed in Escherichia coli BL21 by DiscoverX KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetDiscoidin domain-containing receptor 2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM438155(US10618897, Example 23)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of GST-tagged recombinant DDR2 (unknown origin) expressed in Escherichia coli BL21 by DiscoverX KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetDiscoidin domain-containing receptor 2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM371924(2-[8-(1H-Indazole-5-carbonyl)-4-oxo-1-phenyl-1,3,8...)
Affinity DataIC50: 1.67E+5nMAssay Description:Inhibition of GST-tagged recombinant DDR2 (unknown origin) expressed in Escherichia coli BL21 by DiscoverX KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed