Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50019788
TargetMitogen-activated protein kinase kinase kinase 5(Human)
South China University

Curated by ChEMBL
LigandPNGBDBM50212258(GS-4997 | Selonsertib)
Affinity DataIC50: 17nMAssay Description:Inhibition of human full length recombinant ASK1 (654 to 971 residues) expressed in Sf21 cells using STK-substrate 3-biotin as substrate incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
South China University

Curated by ChEMBL
LigandPNGBDBM50623044(CHEMBL5417817)
Affinity DataIC50: 19nMAssay Description:Inhibition of human full length recombinant ASK1 (654 to 971 residues) expressed in Sf21 cells using STK-substrate 3-biotin as substrate incubated fo...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
South China University

Curated by ChEMBL
LigandPNGBDBM50623041(CHEMBL5437227)
Affinity DataIC50: 26nMAssay Description:Inhibition of human full length recombinant ASK1 (654 to 971 residues) expressed in Sf21 cells using STK-substrate 3-biotin as substrate incubated fo...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
South China University

Curated by ChEMBL
LigandPNGBDBM50623045(CHEMBL5411752)
Affinity DataIC50: 29nMAssay Description:Inhibition of human full length recombinant ASK1 (654 to 971 residues) expressed in Sf21 cells using STK-substrate 3-biotin as substrate incubated fo...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
South China University

Curated by ChEMBL
LigandPNGBDBM50623039(CHEMBL5431768)
Affinity DataIC50: 31nMAssay Description:Inhibition of human full length recombinant ASK1 (654 to 971 residues) expressed in Sf21 cells using STK-substrate 3-biotin as substrate incubated fo...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
South China University

Curated by ChEMBL
LigandPNGBDBM50623043(CHEMBL5406106)
Affinity DataIC50: 49nMAssay Description:Inhibition of human full length recombinant ASK1 (654 to 971 residues) expressed in Sf21 cells using STK-substrate 3-biotin as substrate incubated fo...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
South China University

Curated by ChEMBL
LigandPNGBDBM50623047(CHEMBL5401473)
Affinity DataIC50: 63nMAssay Description:Inhibition of human full length recombinant ASK1 (654 to 971 residues) expressed in Sf21 cells using STK-substrate 3-biotin as substrate incubated fo...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
South China University

Curated by ChEMBL
LigandPNGBDBM50623048(CHEMBL5430975)
Affinity DataIC50: 86nMAssay Description:Inhibition of human full length recombinant ASK1 (654 to 971 residues) expressed in Sf21 cells using STK-substrate 3-biotin as substrate incubated fo...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
South China University

Curated by ChEMBL
LigandPNGBDBM50623046(CHEMBL5411561)
Affinity DataIC50: 102nMAssay Description:Inhibition of human full length recombinant ASK1 (654 to 971 residues) expressed in Sf21 cells using STK-substrate 3-biotin as substrate incubated fo...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
South China University

Curated by ChEMBL
LigandPNGBDBM50623040(CHEMBL5411317)
Affinity DataIC50: 114nMAssay Description:Inhibition of human full length recombinant ASK1 (654 to 971 residues) expressed in Sf21 cells using STK-substrate 3-biotin as substrate incubated fo...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
South China University

Curated by ChEMBL
LigandPNGBDBM50623042(CHEMBL5399807)
Affinity DataIC50: 147nMAssay Description:Inhibition of human full length recombinant ASK1 (654 to 971 residues) expressed in Sf21 cells using STK-substrate 3-biotin as substrate incubated fo...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
South China University

Curated by ChEMBL
LigandPNGBDBM50623050(CHEMBL5421028)
Affinity DataIC50: 161nMAssay Description:Inhibition of human full length recombinant ASK1 (654 to 971 residues) expressed in Sf21 cells using STK-substrate 3-biotin as substrate incubated fo...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
South China University

Curated by ChEMBL
LigandPNGBDBM50623049(CHEMBL5406935)
Affinity DataIC50: 200nMAssay Description:Inhibition of human full length recombinant ASK1 (654 to 971 residues) expressed in Sf21 cells using STK-substrate 3-biotin as substrate incubated fo...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
South China University

Curated by ChEMBL
LigandPNGBDBM50623051(CHEMBL5433012)
Affinity DataIC50: 200nMAssay Description:Inhibition of human full length recombinant ASK1 (654 to 971 residues) expressed in Sf21 cells using STK-substrate 3-biotin as substrate incubated fo...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed