Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50020919
Affinity DataIC50: 1.5nMAssay Description:Binding affinity to human androgen receptor transfected in HEK293 cell membrane co-transfected with ARC1 assessed as inhibition of [3H]-methyltrienol...More data for this Ligand-Target Pair
Affinity DataIC50: 3.70nMAssay Description:Binding affinity to human androgen receptor transfected in HEK293 cell membrane co-transfected with ARC1 assessed as inhibition of [3H]-methyltrienol...More data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:Binding affinity to human androgen receptor transfected in HEK293 cell membrane co-transfected with ARC1 assessed as inhibition of [3H]-methyltrienol...More data for this Ligand-Target Pair
Affinity DataIC50: 5.40nMAssay Description:Binding affinity to human androgen receptor transfected in HEK293 cell membrane co-transfected with ARC1 assessed as inhibition of [3H]-methyltrienol...More data for this Ligand-Target Pair
Affinity DataIC50: 5.70nMAssay Description:Binding affinity to human androgen receptor transfected in HEK293 cell membrane co-transfected with ARC1 assessed as inhibition of [3H]-methyltrienol...More data for this Ligand-Target Pair
Affinity DataIC50: 6.80nMAssay Description:Binding affinity to human androgen receptor transfected in HEK293 cell membrane co-transfected with ARC1 assessed as inhibition of [3H]-methyltrienol...More data for this Ligand-Target Pair
Affinity DataIC50: 9.20nMAssay Description:Binding affinity to human androgen receptor transfected in HEK293 cell membrane co-transfected with ARC1 assessed as inhibition of [3H]-methyltrienol...More data for this Ligand-Target Pair
Affinity DataIC50: 9.5nMAssay Description:Binding affinity to human androgen receptor transfected in HEK293 cell membrane co-transfected with ARC1 assessed as inhibition of [3H]-methyltrienol...More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Binding affinity to human androgen receptor transfected in HEK293 cell membrane co-transfected with ARC1 assessed as inhibition of [3H]-methyltrienol...More data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Antagonist activity at androgen receptor (unknown origin) transfected in HEK293T cells co-transfected with luciferase reporter gene assessed as inhib...More data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Antagonist activity at androgen receptor (unknown origin) transfected in HEK293T cells co-transfected with luciferase reporter gene assessed as inhib...More data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:Antagonist activity at androgen receptor (unknown origin) transfected in HEK293T cells co-transfected with luciferase reporter gene assessed as inhib...More data for this Ligand-Target Pair
Affinity DataIC50: 59nMAssay Description:Antagonist activity at androgen receptor (unknown origin) transfected in HEK293T cells co-transfected with luciferase reporter gene assessed as inhib...More data for this Ligand-Target Pair
Affinity DataIC50: 61nMAssay Description:Antagonist activity at androgen receptor (unknown origin) transfected in HEK293T cells co-transfected with luciferase reporter gene assessed as inhib...More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Antagonist activity at androgen receptor (unknown origin) transfected in HEK293T cells co-transfected with luciferase reporter gene assessed as inhib...More data for this Ligand-Target Pair
Affinity DataIC50: 101nMAssay Description:Antagonist activity at androgen receptor (unknown origin) transfected in HEK293T cells co-transfected with luciferase reporter gene assessed as inhib...More data for this Ligand-Target Pair
Affinity DataIC50: 116nMAssay Description:Antagonist activity at androgen receptor (unknown origin) transfected in HEK293T cells co-transfected with luciferase reporter gene assessed as inhib...More data for this Ligand-Target Pair
Affinity DataIC50: 146nMAssay Description:Antagonist activity at androgen receptor (unknown origin) transfected in HEK293T cells co-transfected with luciferase reporter gene assessed as inhib...More data for this Ligand-Target Pair
Affinity DataIC50: 173nMAssay Description:Antagonist activity at androgen receptor (unknown origin) transfected in HEK293T cells co-transfected with luciferase reporter gene assessed as inhib...More data for this Ligand-Target Pair
Affinity DataIC50: 311nMAssay Description:Antagonist activity at androgen receptor (unknown origin) transfected in HEK293T cells co-transfected with luciferase reporter gene assessed as inhib...More data for this Ligand-Target Pair
Affinity DataIC50: 319nMAssay Description:Antagonist activity at androgen receptor (unknown origin) transfected in HEK293T cells co-transfected with luciferase reporter gene assessed as inhib...More data for this Ligand-Target Pair
Affinity DataIC50: 394nMAssay Description:Antagonist activity at androgen receptor (unknown origin) transfected in HEK293T cells co-transfected with luciferase reporter gene assessed as inhib...More data for this Ligand-Target Pair
Affinity DataIC50: 569nMAssay Description:Antagonist activity at androgen receptor (unknown origin) transfected in HEK293T cells co-transfected with luciferase reporter gene assessed as inhib...More data for this Ligand-Target Pair
Affinity DataKd: 590nMAssay Description:Binding affinity to GST/His-tagged recombinant rat androgen receptor (606 to 902 residues) ligand binding domain expressed in baculovirus expression ...More data for this Ligand-Target Pair
Affinity DataKd: 1.34E+3nMAssay Description:Binding affinity to androgen receptor N-terminal domain (unknown origin) assessed as dissociation constant by Biolayer interferometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at androgen receptor (unknown origin) transfected in HEK293T cells co-transfected with luciferase reporter gene assessed as inhib...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at androgen receptor (unknown origin) transfected in HEK293T cells co-transfected with luciferase reporter gene assessed as inhib...More data for this Ligand-Target Pair
Affinity DataKd: 4.52E+4nMAssay Description:Binding affinity to androgen receptor N-terminal domain (unknown origin) assessed as dissociation constant by Biolayer interferometric analysisMore data for this Ligand-Target Pair

















