Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50020919
TargetProtein cereblon/CUL4A/AR(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50634837(CHEMBL5437141)
Affinity DataIC50: 1.5nMAssay Description:Binding affinity to human androgen receptor transfected in HEK293 cell membrane co-transfected with ARC1 assessed as inhibition of [3H]-methyltrienol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50634846(CHEMBL5555049)
Affinity DataIC50: 3.70nMAssay Description:Binding affinity to human androgen receptor transfected in HEK293 cell membrane co-transfected with ARC1 assessed as inhibition of [3H]-methyltrienol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50634843(CHEMBL5517689)
Affinity DataIC50: 4.60nMAssay Description:Binding affinity to human androgen receptor transfected in HEK293 cell membrane co-transfected with ARC1 assessed as inhibition of [3H]-methyltrienol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50634845(CHEMBL5532063)
Affinity DataIC50: 5.40nMAssay Description:Binding affinity to human androgen receptor transfected in HEK293 cell membrane co-transfected with ARC1 assessed as inhibition of [3H]-methyltrienol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50634839(CHEMBL5531958)
Affinity DataIC50: 5.70nMAssay Description:Binding affinity to human androgen receptor transfected in HEK293 cell membrane co-transfected with ARC1 assessed as inhibition of [3H]-methyltrienol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50634840(CHEMBL5557418)
Affinity DataIC50: 6.80nMAssay Description:Binding affinity to human androgen receptor transfected in HEK293 cell membrane co-transfected with ARC1 assessed as inhibition of [3H]-methyltrienol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50634842(CHEMBL5559204)
Affinity DataIC50: 9.20nMAssay Description:Binding affinity to human androgen receptor transfected in HEK293 cell membrane co-transfected with ARC1 assessed as inhibition of [3H]-methyltrienol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50634841(CHEMBL5557813)
Affinity DataIC50: 9.5nMAssay Description:Binding affinity to human androgen receptor transfected in HEK293 cell membrane co-transfected with ARC1 assessed as inhibition of [3H]-methyltrienol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50634838(CHEMBL5555724)
Affinity DataIC50: 12nMAssay Description:Binding affinity to human androgen receptor transfected in HEK293 cell membrane co-transfected with ARC1 assessed as inhibition of [3H]-methyltrienol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50634835(CHEMBL5559421)
Affinity DataIC50: 26nMAssay Description:Antagonist activity at androgen receptor (unknown origin) transfected in HEK293T cells co-transfected with luciferase reporter gene assessed as inhib...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50634843(CHEMBL5517689)
Affinity DataIC50: 37nMAssay Description:Antagonist activity at androgen receptor (unknown origin) transfected in HEK293T cells co-transfected with luciferase reporter gene assessed as inhib...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50634836(CHEMBL5558125)
Affinity DataIC50: 38nMAssay Description:Antagonist activity at androgen receptor (unknown origin) transfected in HEK293T cells co-transfected with luciferase reporter gene assessed as inhib...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50634834(CHEMBL5518016)
Affinity DataIC50: 59nMAssay Description:Antagonist activity at androgen receptor (unknown origin) transfected in HEK293T cells co-transfected with luciferase reporter gene assessed as inhib...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50634837(CHEMBL5437141)
Affinity DataIC50: 61nMAssay Description:Antagonist activity at androgen receptor (unknown origin) transfected in HEK293T cells co-transfected with luciferase reporter gene assessed as inhib...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50634831(CHEMBL5505831)
Affinity DataIC50: 100nMAssay Description:Antagonist activity at androgen receptor (unknown origin) transfected in HEK293T cells co-transfected with luciferase reporter gene assessed as inhib...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50634832(CHEMBL5542890)
Affinity DataIC50: 101nMAssay Description:Antagonist activity at androgen receptor (unknown origin) transfected in HEK293T cells co-transfected with luciferase reporter gene assessed as inhib...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50634844(CHEMBL5542581)
Affinity DataIC50: 116nMAssay Description:Antagonist activity at androgen receptor (unknown origin) transfected in HEK293T cells co-transfected with luciferase reporter gene assessed as inhib...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50634833(CHEMBL5517813)
Affinity DataIC50: 146nMAssay Description:Antagonist activity at androgen receptor (unknown origin) transfected in HEK293T cells co-transfected with luciferase reporter gene assessed as inhib...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50634842(CHEMBL5559204)
Affinity DataIC50: 173nMAssay Description:Antagonist activity at androgen receptor (unknown origin) transfected in HEK293T cells co-transfected with luciferase reporter gene assessed as inhib...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50634841(CHEMBL5557813)
Affinity DataIC50: 311nMAssay Description:Antagonist activity at androgen receptor (unknown origin) transfected in HEK293T cells co-transfected with luciferase reporter gene assessed as inhib...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50634839(CHEMBL5531958)
Affinity DataIC50: 319nMAssay Description:Antagonist activity at androgen receptor (unknown origin) transfected in HEK293T cells co-transfected with luciferase reporter gene assessed as inhib...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50634840(CHEMBL5557418)
Affinity DataIC50: 394nMAssay Description:Antagonist activity at androgen receptor (unknown origin) transfected in HEK293T cells co-transfected with luciferase reporter gene assessed as inhib...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50634830(CHEMBL5531949)
Affinity DataIC50: 569nMAssay Description:Antagonist activity at androgen receptor (unknown origin) transfected in HEK293T cells co-transfected with luciferase reporter gene assessed as inhib...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetAndrogen receptor(Rat)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50634842(CHEMBL5559204)
Affinity DataKd:  590nMAssay Description:Binding affinity to GST/His-tagged recombinant rat androgen receptor (606 to 902 residues) ligand binding domain expressed in baculovirus expression ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50634842(CHEMBL5559204)
Affinity DataKd:  1.34E+3nMAssay Description:Binding affinity to androgen receptor N-terminal domain (unknown origin) assessed as dissociation constant by Biolayer interferometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50634838(CHEMBL5555724)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at androgen receptor (unknown origin) transfected in HEK293T cells co-transfected with luciferase reporter gene assessed as inhib...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50634845(CHEMBL5532063)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at androgen receptor (unknown origin) transfected in HEK293T cells co-transfected with luciferase reporter gene assessed as inhib...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50094975(US10053433, ARN-509 | ARN-509 | JNJ-56021927 | apa...)
Affinity DataKd:  4.52E+4nMAssay Description:Binding affinity to androgen receptor N-terminal domain (unknown origin) assessed as dissociation constant by Biolayer interferometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed