Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50021853
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Valencia

Curated by ChEMBL
LigandPNGBDBM50030474(US9562012, rosiglitazone | CHEBI:50122 | Avandamet...)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at GAL4-tagged human PPARgamma transfected in African green monkey COS7 cells assessed as transcriptional activation by measuring ef...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Valencia

Curated by ChEMBL
LigandPNGBDBM28661(GW501516 | CHEMBL38943 | 2-{2-methyl-4-[({4-methyl...)
Affinity DataEC50:  0.900nMAssay Description:Agonist activity at GAL4-tagged human PPARbeta/delta transfected in African green monkey COS7 cells assessed as transcriptional activation by measuri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Valencia

Curated by ChEMBL
LigandPNGBDBM24566(JMC515449 Compound 1 | Wyeth 14,643 | 2-({4-chloro...)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at GAL4-tagged human PPARalpha transfected in African green monkey COS7 cells assessed as transcriptional activation by measuring ef...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Valencia

Curated by ChEMBL
LigandPNGBDBM50645467(CHEMBL5592559)
Affinity DataEC50:  1.5nMAssay Description:Agonist activity at GAL4-tagged human PPARbeta/delta transfected in African green monkey COS7 cells assessed as transcriptional activation by measuri...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Valencia

Curated by ChEMBL
LigandPNGBDBM50645466(CHEMBL5202264)
Affinity DataEC50:  1.60nMAssay Description:Agonist activity at GAL4-tagged human PPARgamma transfected in African green monkey COS7 cells assessed as transcriptional activation by measuring ef...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Valencia

Curated by ChEMBL
LigandPNGBDBM50645467(CHEMBL5592559)
Affinity DataEC50:  1.90nMAssay Description:Agonist activity at GAL4-tagged human PPARgamma transfected in African green monkey COS7 cells assessed as transcriptional activation by measuring ef...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Valencia

Curated by ChEMBL
LigandPNGBDBM50645466(CHEMBL5202264)
Affinity DataEC50:  2.20nMAssay Description:Agonist activity at GAL4-tagged human PPARbeta/delta transfected in African green monkey COS7 cells assessed as transcriptional activation by measuri...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Valencia

Curated by ChEMBL
LigandPNGBDBM50645466(CHEMBL5202264)
Affinity DataEC50:  3nMAssay Description:Agonist activity at GAL4-tagged human PPARalpha transfected in African green monkey COS7 cells assessed as transcriptional activation by measuring ef...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Valencia

Curated by ChEMBL
LigandPNGBDBM50645467(CHEMBL5592559)
Affinity DataEC50:  3.20nMAssay Description:Agonist activity at GAL4-tagged human PPARalpha transfected in African green monkey COS7 cells assessed as transcriptional activation by measuring ef...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed