Report error Found 72 Enz. Inhib. hit(s) with all data for entry = 50021372
Affinity DataIC50: 0.0280nMAssay Description:Displacement of 125I-rat amylin from rat AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA meth...More data for this Ligand-Target Pair
Affinity DataIC50: 0.0300nMAssay Description:Displacement of 125I-Calcitonin from rat CTR expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA methodMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0660nMAssay Description:Displacement of 125I-Calcitonin from human CTR expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA methodMore data for this Ligand-Target Pair
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S
Curated by ChEMBL
Novo Nordisk A/S
Curated by ChEMBL
Affinity DataIC50: 0.0890nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S
Curated by ChEMBL
Novo Nordisk A/S
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S
Curated by ChEMBL
Novo Nordisk A/S
Curated by ChEMBL
Affinity DataIC50: 0.114nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S
Curated by ChEMBL
Novo Nordisk A/S
Curated by ChEMBL
Affinity DataIC50: 0.122nMAssay Description:Displacement of 125I-rat amylin from rat AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA meth...More data for this Ligand-Target Pair
Affinity DataIC50: 0.176nMAssay Description:Displacement of 125I-rat amylin from rat AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA meth...More data for this Ligand-Target Pair
Affinity DataIC50: 0.203nMAssay Description:Displacement of 125I-rat amylin from rat AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA meth...More data for this Ligand-Target Pair
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S
Curated by ChEMBL
Novo Nordisk A/S
Curated by ChEMBL
Affinity DataIC50: 0.213nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
Affinity DataIC50: 0.217nMAssay Description:Displacement of 125I-rat amylin from rat AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA meth...More data for this Ligand-Target Pair
Affinity DataIC50: 0.290nMAssay Description:Displacement of 125I-rat amylin from rat AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA meth...More data for this Ligand-Target Pair
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S
Curated by ChEMBL
Novo Nordisk A/S
Curated by ChEMBL
Affinity DataIC50: 0.344nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S
Curated by ChEMBL
Novo Nordisk A/S
Curated by ChEMBL
Affinity DataIC50: 0.355nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
Affinity DataIC50: 0.372nMAssay Description:Displacement of 125I-rat amylin from rat AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA meth...More data for this Ligand-Target Pair
Affinity DataIC50: 0.449nMAssay Description:Displacement of 125I-rat amylin from rat AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA meth...More data for this Ligand-Target Pair
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S
Curated by ChEMBL
Novo Nordisk A/S
Curated by ChEMBL
Affinity DataIC50: 0.484nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S
Curated by ChEMBL
Novo Nordisk A/S
Curated by ChEMBL
Affinity DataIC50: 0.561nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S
Curated by ChEMBL
Novo Nordisk A/S
Curated by ChEMBL
Affinity DataIC50: 0.589nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S
Curated by ChEMBL
Novo Nordisk A/S
Curated by ChEMBL
Affinity DataIC50: 0.662nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S
Curated by ChEMBL
Novo Nordisk A/S
Curated by ChEMBL
Affinity DataIC50: 0.745nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S
Curated by ChEMBL
Novo Nordisk A/S
Curated by ChEMBL
Affinity DataIC50: 0.885nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
Affinity DataIC50: 0.920nMAssay Description:Displacement of 125I-rat amylin from rat AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA meth...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Displacement of 125I-rat amylin from rat AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA meth...More data for this Ligand-Target Pair
Affinity DataIC50: 1.09nMAssay Description:Displacement of 125I-Calcitonin from human CTR expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA methodMore data for this Ligand-Target Pair
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S
Curated by ChEMBL
Novo Nordisk A/S
Curated by ChEMBL
Affinity DataIC50: 1.12nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S
Curated by ChEMBL
Novo Nordisk A/S
Curated by ChEMBL
Affinity DataIC50: 1.13nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S
Curated by ChEMBL
Novo Nordisk A/S
Curated by ChEMBL
Affinity DataIC50: 1.14nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S
Curated by ChEMBL
Novo Nordisk A/S
Curated by ChEMBL
Affinity DataIC50: 1.14nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
Affinity DataIC50: 1.17nMAssay Description:Displacement of 125I-rat amylin from rat AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA meth...More data for this Ligand-Target Pair
Affinity DataIC50: 1.24nMAssay Description:Displacement of 125I-rat amylin from rat AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA meth...More data for this Ligand-Target Pair
Affinity DataIC50: 1.29nMAssay Description:Displacement of 125I-rat amylin from rat AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA meth...More data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Displacement of 125I-rat amylin from rat AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA meth...More data for this Ligand-Target Pair
Affinity DataIC50: 1.49nMAssay Description:Displacement of 125I-Calcitonin from human CTR expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.72nMAssay Description:Displacement of 125I-rat amylin from rat AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA meth...More data for this Ligand-Target Pair
Affinity DataIC50: 1.77nMAssay Description:Displacement of 125I-rat amylin from rat AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA meth...More data for this Ligand-Target Pair
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S
Curated by ChEMBL
Novo Nordisk A/S
Curated by ChEMBL
Affinity DataIC50: 2.75nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
Affinity DataIC50: 3.01nMAssay Description:Displacement of 125I-rat amylin from rat AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA meth...More data for this Ligand-Target Pair
Affinity DataIC50: 4.69nMAssay Description:Displacement of 125I-rat amylin from rat AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA meth...More data for this Ligand-Target Pair
TargetCalcitonin receptor/Receptor activity-modifying protein 3(Homo sapiens)
Novo Nordisk A/S
Curated by ChEMBL
Novo Nordisk A/S
Curated by ChEMBL
Affinity DataIC50: 5.09nMAssay Description:Displacement of 125I-rat amylin from human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA me...More data for this Ligand-Target Pair
Affinity DataIC50: 5.83nMAssay Description:Displacement of 125I-Calcitonin from rat CTR expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA methodMore data for this Ligand-Target Pair
Affinity DataIC50: 5.98nMAssay Description:Displacement of 125I-Calcitonin from rat CTR expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA methodMore data for this Ligand-Target Pair
Affinity DataIC50: 7.55nMAssay Description:Displacement of 125I-Calcitonin from rat CTR expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA methodMore data for this Ligand-Target Pair
Affinity DataIC50: 11.7nMAssay Description:Displacement of 125I-Calcitonin from human CTR expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA methodMore data for this Ligand-Target Pair
Affinity DataIC50: 11.9nMAssay Description:Displacement of 125I-Calcitonin from human CTR expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA methodMore data for this Ligand-Target Pair
Affinity DataIC50: 14.1nMAssay Description:Displacement of 125I-Calcitonin from human CTR expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA methodMore data for this Ligand-Target Pair
Affinity DataIC50: 15.5nMAssay Description:Displacement of 125I-Calcitonin from human CTR expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA methodMore data for this Ligand-Target Pair
Affinity DataIC50: 17.1nMAssay Description:Displacement of 125I-Calcitonin from rat CTR expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA methodMore data for this Ligand-Target Pair
Affinity DataIC50: 19.3nMAssay Description:Displacement of 125I-Calcitonin from human CTR expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA methodMore data for this Ligand-Target Pair
Affinity DataIC50: 19.5nMAssay Description:Displacement of 125I-Calcitonin from human CTR expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA methodMore data for this Ligand-Target Pair

















