Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50023643
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
The Affiliated Taizhou People's Hospital of Nanjing Medical University
Curated by ChEMBL
The Affiliated Taizhou People's Hospital of Nanjing Medical University
Curated by ChEMBL
Affinity DataIC50: 4.20nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) pre-incubated for 20 min followed by 32P-ATP addition and measured after 2 hrsMore data for this Ligand-Target Pair
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
The Affiliated Taizhou People's Hospital of Nanjing Medical University
Curated by ChEMBL
The Affiliated Taizhou People's Hospital of Nanjing Medical University
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) pre-incubated for 20 min followed by 32P-ATP addition and measured after 2 hrsMore data for this Ligand-Target Pair
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
The Affiliated Taizhou People's Hospital of Nanjing Medical University
Curated by ChEMBL
The Affiliated Taizhou People's Hospital of Nanjing Medical University
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) pre-incubated for 20 min followed by 32P-ATP addition and measured after 2 hrsMore data for this Ligand-Target Pair
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
The Affiliated Taizhou People's Hospital of Nanjing Medical University
Curated by ChEMBL
The Affiliated Taizhou People's Hospital of Nanjing Medical University
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) pre-incubated for 20 min followed by 32P-ATP addition and measured after 2 hrsMore data for this Ligand-Target Pair
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
The Affiliated Taizhou People's Hospital of Nanjing Medical University
Curated by ChEMBL
The Affiliated Taizhou People's Hospital of Nanjing Medical University
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) pre-incubated for 20 min followed by 32P-ATP addition and measured after 2 hrsMore data for this Ligand-Target Pair
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
The Affiliated Taizhou People's Hospital of Nanjing Medical University
Curated by ChEMBL
The Affiliated Taizhou People's Hospital of Nanjing Medical University
Curated by ChEMBL
Affinity DataIC50: 37nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) pre-incubated for 20 min followed by 32P-ATP addition and measured after 2 hrsMore data for this Ligand-Target Pair
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
The Affiliated Taizhou People's Hospital of Nanjing Medical University
Curated by ChEMBL
The Affiliated Taizhou People's Hospital of Nanjing Medical University
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) pre-incubated for 20 min followed by 32P-ATP addition and measured after 2 hrsMore data for this Ligand-Target Pair
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
The Affiliated Taizhou People's Hospital of Nanjing Medical University
Curated by ChEMBL
The Affiliated Taizhou People's Hospital of Nanjing Medical University
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) pre-incubated for 20 min followed by 32P-ATP addition and measured after 2 hrsMore data for this Ligand-Target Pair
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
The Affiliated Taizhou People's Hospital of Nanjing Medical University
Curated by ChEMBL
The Affiliated Taizhou People's Hospital of Nanjing Medical University
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) pre-incubated for 20 min followed by 32P-ATP addition and measured after 2 hrsMore data for this Ligand-Target Pair
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
The Affiliated Taizhou People's Hospital of Nanjing Medical University
Curated by ChEMBL
The Affiliated Taizhou People's Hospital of Nanjing Medical University
Curated by ChEMBL
Affinity DataIC50: 87nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) pre-incubated for 20 min followed by 32P-ATP addition and measured after 2 hrsMore data for this Ligand-Target Pair
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
The Affiliated Taizhou People's Hospital of Nanjing Medical University
Curated by ChEMBL
The Affiliated Taizhou People's Hospital of Nanjing Medical University
Curated by ChEMBL
Affinity DataIC50: 350nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) pre-incubated for 20 min followed by 32P-ATP addition and measured after 2 hrsMore data for this Ligand-Target Pair


3D Structure (crystal)







