Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50023269
Affinity DataIC50: 22nMAssay Description:Inhibition of full length USP7 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 41nMAssay Description:Inhibition of full length USP7 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 65nMAssay Description:Binding affinity to USP7 catalytic domain human USP7 (208 to 560 residues) (unknown origin) extracted from Escherichia coli assessed as dissociation ...More data for this Ligand-Target Pair
Affinity DataKd: 78nMAssay Description:Binding affinity to USP7 catalytic domain human USP7 (208 to 560 residues) (unknown origin) extracted from Escherichia coli assessed as dissociation ...More data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Inhibition of full length USP7 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of 6xHis-tagged full length USP7 (unknown origin) incubated for 15 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 420nMAssay Description:Inhibition of N-terminal 6xHis-tagged human recombinant USP7 catalytic domain (208 to 560 residues) extracted from Escherichia coli BL21 (DE3) measur...More data for this Ligand-Target Pair
Affinity DataIC50: 430nMAssay Description:Inhibition of N-terminal His-tagged USP7 catalytic domain (208 to 554 residues) (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 610nMAssay Description:Inhibition of N-terminal His-tagged USP7 catalytic domain (208 to 554 residues) (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 750nMAssay Description:Inhibition of N-terminal GST-tagged full length recombinant USP7 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of full length USP7 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.34E+3nMAssay Description:Inhibition of N-terminal GST-tagged full length recombinant USP7 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.20E+3nMAssay Description:Binding affinity to N-terminal His-tagged USP7 catalytic domain (208 to 560 residues) extracted from Escherichia coli Rosetta2 cells assessed as inhi...More data for this Ligand-Target Pair
Affinity DataKd: 7.80E+3nMAssay Description:Binding affinity to N-terminal His-tagged USP7 catalytic domain (208 to 560 residues) (unknonw origin) extracted from Escherichia coli Rosetta2 cells...More data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of N-terminal 6xHis-tagged human recombinant USP7 catalytic domain (208 to 560 residues) extracted from Escherichia coli BL21 (DE3) measur...More data for this Ligand-Target Pair
Affinity DataIC50: 8.20E+3nMAssay Description:Inhibition of full length USP7 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of full length USP7 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.23E+4nMAssay Description:Inhibition of USP7 catalytic domain human USP7 (208 to 560 residues) (unknown origin) extracted from Escherichia coliMore data for this Ligand-Target Pair
Affinity DataIC50: 5.20E+4nMAssay Description:Inhibition of USP7 catalytic domain human USP7 (208 to 560 residues) (unknown origin) extracted from Escherichia coliMore data for this Ligand-Target Pair
Affinity DataIC50: 7.92E+4nMAssay Description:Inhibition of N-terminal GST-tagged full length recombinant USP7 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibition of USP1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibition of USP47 (unknown origin)More data for this Ligand-Target Pair




3D Structure (crystal)








