Report error Found 60 Enz. Inhib. hit(s) with all data for entry = 50023761
Affinity DataKd: 3.20nMAssay Description:Binding affinity to N-terminal 6xHis-tagged human STING R232H mutant CTD extracted from Escherichia coli BL21(DE3) assessed as dissociation constant ...More data for this Ligand-Target Pair
Affinity DataEC50: 60nMAssay Description:Agonist activity at STING in human THP1-Blue ISG cells harbouring SEAP reporter gene assessed as activation of cGAS-STING signaling pathway incubated...More data for this Ligand-Target Pair
Affinity DataKd: 216nMAssay Description:Binding affinity to N-terminal 6xHis-tagged human STING R232H mutant CTD extracted from Escherichia coli BL21(DE3) assessed as dissociation constant ...More data for this Ligand-Target Pair
Affinity DataKd: 279nMAssay Description:Binding affinity to N-terminal 6xHis-tagged human STING R232H mutant CTD extracted from Escherichia coli BL21(DE3) assessed as dissociation constant ...More data for this Ligand-Target Pair
Affinity DataEC50: 300nMAssay Description:Agonist activity at STING in human THP1-Blue ISG cells harbouring SEAP reporter gene assessed as activation of cGAS-STING signaling pathway incubated...More data for this Ligand-Target Pair
Affinity DataEC50: 330nMAssay Description:Agonist activity at STING in human THP1-Blue ISG cells harbouring SEAP reporter gene assessed as activation of cGAS-STING signaling pathway incubated...More data for this Ligand-Target Pair
Affinity DataEC50: 340nMAssay Description:Agonist activity at STING in human THP1-Blue ISG cells harbouring SEAP reporter gene assessed as activation of cGAS-STING signaling pathway incubated...More data for this Ligand-Target Pair
Affinity DataEC50: 350nMAssay Description:Agonist activity at STING in human THP1-Blue ISG cells harbouring SEAP reporter gene assessed as activation of cGAS-STING signaling pathway incubated...More data for this Ligand-Target Pair
Affinity DataEC50: 360nMAssay Description:Agonist activity at STING in human THP1-Blue ISG cells harbouring SEAP reporter gene assessed as activation of cGAS-STING signaling pathway incubated...More data for this Ligand-Target Pair
Affinity DataEC50: 380nMAssay Description:Agonist activity at STING in human THP1-Blue ISG cells harbouring SEAP reporter gene assessed as activation of cGAS-STING signaling pathway incubated...More data for this Ligand-Target Pair
Affinity DataKd: 526nMAssay Description:Binding affinity to N-terminal 6xHis-tagged human STING R232H mutant CTD extracted from Escherichia coli BL21(DE3) assessed as dissociation constant ...More data for this Ligand-Target Pair
Affinity DataEC50: 700nMAssay Description:Agonist activity at STING in human THP1-Blue ISG cells harbouring SEAP reporter gene assessed as activation of cGAS-STING signaling pathway incubated...More data for this Ligand-Target Pair
Affinity DataEC50: 710nMAssay Description:Agonist activity at STING in human THP1-Blue ISG cells harbouring SEAP reporter gene assessed as activation of cGAS-STING signaling pathway incubated...More data for this Ligand-Target Pair
Affinity DataIC50: 770nMAssay Description:Displacement of 5-FAM-labeled diABZI tracer from N-terminal 6xHis-tagged human STING R232H mutant CTD extracted from Escherichia coli BL21(DE3) incub...More data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Displacement of 5-FAM-labeled diABZI tracer from N-terminal 6xHis-tagged human STING G230A/R293Q mutant CTD extracted from Escherichia coli BL21(DE3)...More data for this Ligand-Target Pair
Affinity DataEC50: 820nMAssay Description:Agonist activity at STING in human THP1-Blue ISG cells harbouring SEAP reporter gene assessed as activation of cGAS-STING signaling pathway incubated...More data for this Ligand-Target Pair
Affinity DataIC50: 900nMAssay Description:Displacement of 5-FAM-labeled diABZI tracer from N-terminal 6xHis-tagged wild-type human STING CTD extracted from Escherichia coli BL21(DE3) incubate...More data for this Ligand-Target Pair
Affinity DataIC50: 940nMAssay Description:Displacement of 5-FAM-labeled diABZI tracer from N-terminal 6xHis-tagged human STING G230A/R293Q mutant CTD extracted from Escherichia coli BL21(DE3)...More data for this Ligand-Target Pair
Affinity DataIC50: 980nMAssay Description:Displacement of 5-FAM-labeled diABZI tracer from N-terminal 6xHis-tagged human STING G230A/R293Q mutant CTD extracted from Escherichia coli BL21(DE3)...More data for this Ligand-Target Pair
Affinity DataIC50: 1.15E+3nMAssay Description:Displacement of 5-FAM-labeled diABZI tracer from N-terminal 6xHis-tagged human STING R293Q mutant CTD extracted from Escherichia coli BL21(DE3) incub...More data for this Ligand-Target Pair
Affinity DataIC50: 1.36E+3nMAssay Description:Displacement of 5-FAM-labeled diABZI tracer from N-terminal 6xHis-tagged human STING R232H mutant CTD extracted from Escherichia coli BL21(DE3) incub...More data for this Ligand-Target Pair
Affinity DataIC50: 1.45E+3nMAssay Description:Displacement of 5-FAM-labeled diABZI tracer from N-terminal 6xHis-tagged human STING R293Q mutant CTD extracted from Escherichia coli BL21(DE3) incub...More data for this Ligand-Target Pair
Affinity DataIC50: 1.48E+3nMAssay Description:Displacement of 5-FAM-labeled diABZI tracer from N-terminal 6xHis-tagged wild-type human STING CTD extracted from Escherichia coli BL21(DE3) incubate...More data for this Ligand-Target Pair
Affinity DataIC50: 1.49E+3nMAssay Description:Displacement of 5-FAM-labeled diABZI tracer from N-terminal 6xHis-tagged human STING G230A/R293Q mutant CTD extracted from Escherichia coli BL21(DE3)...More data for this Ligand-Target Pair
Affinity DataIC50: 1.53E+3nMAssay Description:Displacement of 5-FAM-labeled diABZI tracer from N-terminal 6xHis-tagged wild-type mouse STING CTD extracted from Escherichia coli BL21(DE3) incubate...More data for this Ligand-Target Pair
Affinity DataEC50: 1.71E+3nMAssay Description:Agonist activity at STING in human THP1-Blue ISG cells harbouring SEAP reporter gene assessed as activation of cGAS-STING signaling pathway incubated...More data for this Ligand-Target Pair
Affinity DataIC50: 1.73E+3nMAssay Description:Displacement of 5-FAM-labeled diABZI tracer from N-terminal 6xHis-tagged human STING R232H mutant CTD extracted from Escherichia coli BL21(DE3) incub...More data for this Ligand-Target Pair
Affinity DataIC50: 1.84E+3nMAssay Description:Displacement of 5-FAM-labeled diABZI tracer from N-terminal 6xHis-tagged wild-type human STING CTD extracted from Escherichia coli BL21(DE3) incubate...More data for this Ligand-Target Pair
Affinity DataIC50: 1.87E+3nMAssay Description:Displacement of 5-FAM-labeled diABZI tracer from N-terminal 6xHis-tagged wild-type mouse STING CTD extracted from Escherichia coli BL21(DE3) incubate...More data for this Ligand-Target Pair
Affinity DataIC50: 1.91E+3nMAssay Description:Displacement of 5-FAM-labeled diABZI tracer from N-terminal 6xHis-tagged human STING R293Q mutant CTD extracted from Escherichia coli BL21(DE3) incub...More data for this Ligand-Target Pair
Affinity DataEC50: 2.23E+3nMAssay Description:Agonist activity at STING in human THP1-Blue ISG cells harbouring SEAP reporter gene assessed as activation of cGAS-STING signaling pathway incubated...More data for this Ligand-Target Pair
Affinity DataIC50: 2.51E+3nMAssay Description:Displacement of 5-FAM-labeled diABZI tracer from N-terminal 6xHis-tagged wild-type mouse STING CTD extracted from Escherichia coli BL21(DE3) incubate...More data for this Ligand-Target Pair
Affinity DataIC50: 2.64E+3nMAssay Description:Displacement of 5-FAM-labeled diABZI tracer from N-terminal 6xHis-tagged wild-type mouse STING CTD extracted from Escherichia coli BL21(DE3) incubate...More data for this Ligand-Target Pair
Affinity DataEC50: 2.85E+3nMAssay Description:Agonist activity at STING in human THP1-Blue ISG cells harbouring SEAP reporter gene assessed as activation of cGAS-STING signaling pathway incubated...More data for this Ligand-Target Pair
Affinity DataEC50: 3.29E+3nMAssay Description:Agonist activity at STING in human THP1-Blue ISG cells harbouring SEAP reporter gene assessed as activation of cGAS-STING signaling pathway incubated...More data for this Ligand-Target Pair
Affinity DataEC50: 3.91E+3nMAssay Description:Agonist activity at STING in human THP1-Blue ISG cells harbouring SEAP reporter gene assessed as activation of cGAS-STING signaling pathway incubated...More data for this Ligand-Target Pair
Affinity DataEC50: 5.16E+3nMAssay Description:Agonist activity at STING in human THP1-Blue ISG cells harbouring SEAP reporter gene assessed as activation of cGAS-STING signaling pathway incubated...More data for this Ligand-Target Pair
Affinity DataIC50: 6.07E+3nMAssay Description:Displacement of 5-FAM-labeled diABZI tracer from N-terminal 6xHis-tagged human STING R232H mutant CTD extracted from Escherichia coli BL21(DE3) incub...More data for this Ligand-Target Pair
Affinity DataEC50: 6.15E+3nMAssay Description:Agonist activity at STING in human THP1-Blue ISG cells harbouring SEAP reporter gene assessed as activation of cGAS-STING signaling pathway incubated...More data for this Ligand-Target Pair
Affinity DataEC50: 7.59E+3nMAssay Description:Agonist activity at STING in human THP1-Blue ISG cells harbouring SEAP reporter gene assessed as activation of cGAS-STING signaling pathway incubated...More data for this Ligand-Target Pair
Affinity DataEC50: 9.03E+3nMAssay Description:Agonist activity at STING in human THP1-Blue ISG cells harbouring SEAP reporter gene assessed as activation of cGAS-STING signaling pathway incubated...More data for this Ligand-Target Pair
Affinity DataIC50: 1.01E+4nMAssay Description:Displacement of 5-FAM-labeled diABZI tracer from N-terminal 6xHis-tagged wild-type human STING CTD extracted from Escherichia coli BL21(DE3) incubate...More data for this Ligand-Target Pair
Affinity DataIC50: 1.04E+4nMAssay Description:Displacement of 5-FAM-labeled diABZI tracer from N-terminal 6xHis-tagged human STING R293Q mutant CTD extracted from Escherichia coli BL21(DE3) incub...More data for this Ligand-Target Pair
Affinity DataEC50: 1.15E+4nMAssay Description:Agonist activity at STING in human THP1-Blue ISG cells harbouring SEAP reporter gene assessed as activation of cGAS-STING signaling pathway incubated...More data for this Ligand-Target Pair
Affinity DataEC50: 1.17E+4nMAssay Description:Agonist activity at STING in human THP1-Blue ISG cells harbouring SEAP reporter gene assessed as activation of cGAS-STING signaling pathway incubated...More data for this Ligand-Target Pair
Affinity DataEC50: 1.28E+4nMAssay Description:Agonist activity at STING in human THP1-Blue ISG cells harbouring SEAP reporter gene assessed as activation of cGAS-STING signaling pathway incubated...More data for this Ligand-Target Pair
Affinity DataEC50: 1.33E+4nMAssay Description:Agonist activity at STING in human THP1-Blue ISG cells harbouring SEAP reporter gene assessed as activation of cGAS-STING signaling pathway incubated...More data for this Ligand-Target Pair
Affinity DataEC50: 1.38E+4nMAssay Description:Agonist activity at STING in human THP1-Blue ISG cells harbouring SEAP reporter gene assessed as activation of cGAS-STING signaling pathway incubated...More data for this Ligand-Target Pair
Affinity DataEC50: 1.42E+4nMAssay Description:Agonist activity at STING in mouse RAW-Lucia ISG cells harbouring SEAP reporter gene assessed as activation of cGAS-STING signaling pathway incubated...More data for this Ligand-Target Pair
Affinity DataEC50: 2.46E+4nMAssay Description:Agonist activity at STING in mouse RAW-Lucia ISG cells harbouring SEAP reporter gene assessed as activation of cGAS-STING signaling pathway incubated...More data for this Ligand-Target Pair
