Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50028918
TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50280133((3S,4S)-4-[(Naphthalene-2-carbonyl)-amino]-5-oxo-1...)
Affinity DataIC50: 16nMAssay Description:Displacement of [125I]CCK-OP radioligand from Cholecystokinin type A receptor in rat pancreatic acinar membrane binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50280135((3S,4S)-4-[(1H-Indole-2-carbonyl)-amino]-5-oxo-1-p...)
Affinity DataIC50: 19nMAssay Description:Displacement of [125I]CCK-OP radioligand from Cholecystokinin type A receptor in rat pancreatic acinar membrane binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50008170(CHEMBL24938 | 4-(3,4-Dichloro-benzoylamino)-4-dipe...)
Affinity DataIC50: 22nMAssay Description:Displacement of [125I]CCK-OP radioligand from Cholecystokinin type A receptor in rat pancreatic acinar membrane binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50280136((3S,4S)-1-(2-Fluoro-phenyl)-4-[(naphthalene-2-carb...)
Affinity DataIC50: 62nMAssay Description:Displacement of [125I]CCK-OP radioligand from Cholecystokinin type A receptor in rat pancreatic acinar membrane binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50280139((3S,4S)-1-(2-Fluoro-phenyl)-5-oxo-4-[(quinoline-3-...)
Affinity DataIC50: 170nMAssay Description:Displacement of [125I]CCK-OP radioligand from Cholecystokinin type A receptor in rat pancreatic acinar membrane binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50280134((3S,4R)-4-[(Naphthalene-2-carbonyl)-amino]-5-oxo-1...)
Affinity DataIC50: 290nMAssay Description:Displacement of [125I]CCK-OP radioligand from Cholecystokinin type A receptor in rat pancreatic acinar membrane binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50280138((3S,4R)-4-[(1H-Indole-2-carbonyl)-amino]-5-oxo-1-p...)
Affinity DataIC50: 360nMAssay Description:Displacement of [125I]CCK-OP radioligand from Cholecystokinin type A receptor in rat pancreatic acinar membrane binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50280137((3S,4S)-1-Benzyl-4-[(1H-indole-2-carbonyl)-amino]-...)
Affinity DataIC50: 550nMAssay Description:Displacement of [125I]CCK-OP radioligand from Cholecystokinin type A receptor in rat pancreatic acinar membrane binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50280132((3S,4S)-1-Benzyl-4-[(naphthalene-2-carbonyl)-amino...)
Affinity DataIC50: 1.29E+3nMAssay Description:Displacement of [125I]CCK-OP radioligand from Cholecystokinin type A receptor in rat pancreatic acinar membrane binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50280137((3S,4S)-1-Benzyl-4-[(1H-indole-2-carbonyl)-amino]-...)
Affinity DataIC50: 2.00E+3nMAssay Description:Displacement of [125I]CCK-OP radioligand from Cholecystokinin type B receptor of guinea pig cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50280135((3S,4S)-4-[(1H-Indole-2-carbonyl)-amino]-5-oxo-1-p...)
Affinity DataIC50: 4.80E+3nMAssay Description:Displacement of [125I]CCK-OP radioligand from Cholecystokinin type B receptor of guinea pig cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50280132((3S,4S)-1-Benzyl-4-[(naphthalene-2-carbonyl)-amino...)
Affinity DataIC50: 7.35E+3nMAssay Description:Displacement of [125I]CCK-OP radioligand from Cholecystokinin type B receptor of guinea pig cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50280133((3S,4S)-4-[(Naphthalene-2-carbonyl)-amino]-5-oxo-1...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]CCK-OP radioligand from Cholecystokinin type B receptor of guinea pig cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50280138((3S,4R)-4-[(1H-Indole-2-carbonyl)-amino]-5-oxo-1-p...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]CCK-OP radioligand from Cholecystokinin type B receptor of guinea pig cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50280136((3S,4S)-1-(2-Fluoro-phenyl)-4-[(naphthalene-2-carb...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]CCK-OP radioligand from Cholecystokinin type B receptor of guinea pig cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50280139((3S,4S)-1-(2-Fluoro-phenyl)-5-oxo-4-[(quinoline-3-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]CCK-OP radioligand from Cholecystokinin type B receptor of guinea pig cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50280134((3S,4R)-4-[(Naphthalene-2-carbonyl)-amino]-5-oxo-1...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]CCK-OP radioligand from Cholecystokinin type B receptor of guinea pig cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article