Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50028920
TargetKappa-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50045179(4-[2-(3,4-Dichloro-phenyl)-acetyl]-3-pyrrolidin-1-...)
Affinity DataIC50: 0.0200nMAssay Description:Agonistic activity at kappa opioid receptor of rabbit vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetKappa-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50280147(1-[4-Acetyl-2-((S)-3-hydroxy-pyrrolidin-1-ylmethyl...)
Affinity DataIC50: 0.220nMAssay Description:Agonistic activity at kappa opioid receptor of rabbit vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetKappa-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50280145(1-[4-Acetyl-2-((S)-3-hydroxy-pyrrolidin-1-ylmethyl...)
Affinity DataIC50: 0.900nMAssay Description:Agonistic activity at kappa opioid receptor of rabbit vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetKappa-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50280149(1-[4-Acetyl-2-((S)-3-hydroxy-pyrrolidin-1-ylmethyl...)
Affinity DataIC50: 1.5nMAssay Description:Agonistic activity at kappa opioid receptor of rabbit vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetKappa-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50280148(1-[4-Acetyl-2-((S)-3-hydroxy-pyrrolidin-1-ylmethyl...)
Affinity DataIC50: 4.60nMAssay Description:Agonistic activity at kappa opioid receptor of rabbit vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetKappa-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50280150(1-[4-Acetyl-2-((S)-3-hydroxy-pyrrolidin-1-ylmethyl...)
Affinity DataIC50: 6.30nMAssay Description:Agonistic activity at kappa opioid receptor of rabbit vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetKappa-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM83435(2-[3-[1-[2-(3,4-dichlorophenyl)ethanoyl-methyl-ami...)
Affinity DataIC50: 7.40nMAssay Description:Agonistic activity at kappa opioid receptor of rabbit vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetKappa-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50280142(1-[4-Acetyl-2-((S)-3-hydroxy-pyrrolidin-1-ylmethyl...)
Affinity DataIC50: 14nMAssay Description:Agonistic activity at kappa opioid receptor of rabbit vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetKappa-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50280143(1-[4-Acetyl-2-((S)-3-hydroxy-pyrrolidin-1-ylmethyl...)
Affinity DataIC50: 37nMAssay Description:Agonistic activity at kappa opioid receptor of rabbit vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetKappa-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50280144(1-[4-Acetyl-2-((S)-3-hydroxy-pyrrolidin-1-ylmethyl...)
Affinity DataIC50: 49nMAssay Description:Agonistic activity at kappa opioid receptor of rabbit vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetKappa-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50280151(1-[4-Acetyl-2-((S)-3-hydroxy-pyrrolidin-1-ylmethyl...)
Affinity DataIC50: 140nMAssay Description:Agonistic activity at kappa opioid receptor of rabbit vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetKappa-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50280146(1-[4-Acetyl-2-((S)-3-hydroxy-pyrrolidin-1-ylmethyl...)
Affinity DataIC50: 230nMAssay Description:Agonistic activity at kappa opioid receptor of rabbit vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetKappa-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50280141(1-[4-Acetyl-2-((S)-3-hydroxy-pyrrolidin-1-ylmethyl...)
Affinity DataIC50: 400nMAssay Description:Agonistic activity at kappa opioid receptor of rabbit vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article