Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50028986
TargetProstaglandin G/H synthase 1/2(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM22971(Meclofenamate | CHEMBL509 | 2-[(2,6-dichloro-3-met...)
Affinity DataIC50: 100nMAssay Description:Compound was evaluated for its inhibitory activity against CO(cyclooxygenase)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article
PDB3D3D Structure (crystal)
TargetProstaglandin G/H synthase 1/2(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM17638(indometacin | Indocin | 2-{1-[(4-chlorophenyl)carb...)
Affinity DataIC50: 500nMAssay Description:Compound was evaluated for its inhibitory activity against CO(cyclooxygenase) in intact RBL-1 cell line assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article
PDB3D3D Structure (crystal)
LigandPNGBDBM50280512(5-[1-[2-(2,6-Dichloro-3-methyl-phenylamino)-phenyl...)
Affinity DataIC50: 820nMAssay Description:Compound was evaluated for its inhibitory activity against 5-LO (5-lipoxygenase)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50280511(5-[1-[1-(4-Chloro-benzoyl)-5-methoxy-2-methyl-1H-i...)
Affinity DataIC50: 1.40E+3nMAssay Description:Compound was evaluated for its inhibitory activity against 5-LO (5-lipoxygenase) in intact RBL-1 cell line assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50280514(5-[1-[2-(2,6-Dichloro-3-methyl-phenylamino)-phenyl...)
Affinity DataIC50: 1.50E+3nMAssay Description:Compound was evaluated for its inhibitory activity against 5-LO (5-lipoxygenase) in intact RBL-1 cell line assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetProstaglandin G/H synthase 1/2(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50280511(5-[1-[1-(4-Chloro-benzoyl)-5-methoxy-2-methyl-1H-i...)
Affinity DataIC50: 2.00E+3nMAssay Description:Compound was evaluated for its inhibitory activity against CO(cyclooxygenase) in intact RBL-1 cell line assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50280513({5-[1-[2-(2,6-Dichloro-3-methyl-phenylamino)-pheny...)
Affinity DataIC50: 2.20E+3nMAssay Description:Compound was evaluated for its inhibitory activity against 5-LO (5-lipoxygenase) in intact RBL-1 cell line assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetProstaglandin G/H synthase 1/2(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50280512(5-[1-[2-(2,6-Dichloro-3-methyl-phenylamino)-phenyl...)
Affinity DataIC50: 6.00E+3nMAssay Description:Compound was evaluated for its inhibitory activity against CO(cyclooxygenase)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetProstaglandin G/H synthase 1/2(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50280514(5-[1-[2-(2,6-Dichloro-3-methyl-phenylamino)-phenyl...)
Affinity DataIC50: 1.02E+4nMAssay Description:Compound was evaluated for its inhibitory activity against CO(cyclooxygenase) in intact RBL-1 cell line assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM22971(Meclofenamate | CHEMBL509 | 2-[(2,6-dichloro-3-met...)
Affinity DataIC50: 2.40E+4nMAssay Description:Compound was evaluated for its inhibitory activity against 5-LO (5-lipoxygenase)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM17638(indometacin | Indocin | 2-{1-[(4-chlorophenyl)carb...)
Affinity DataIC50: 1.00E+5nMAssay Description:Compound was evaluated for its inhibitory activity against 5-LO (5-lipoxygenase) in intact RBL-1 cell line assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article