Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50029054
TargetNeutrophil elastase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50281005([(5R,6S)-7-Oxo-6-((R)-1-phenylacetoxy-ethyl)-2,4-d...)
Affinity DataKi:  400nMAssay Description:Inhibitory activity against human leukocyte elastase (HLE) was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeutrophil elastase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50281006([(5R,6S)-6-((R)-1-Hydroxy-ethyl)-7-oxo-2,4-dithia-...)
Affinity DataKi:  1.50E+3nM Koff:  1.00E+3s-1Assay Description:Rate constant for the compound was determined (k2/ki) against human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeutrophil elastase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50281004([(5R,6S)-6-((R)-1-Hydroxy-ethyl)-7-oxo-2-thia-1-az...)
Affinity DataKi:  3.20E+3nM Koff:  130s-1Assay Description:Rate constant for the compound was determined (k2/ki) against human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeutrophil elastase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50281003([(5R,6S)-6-((R)-1-Hydroxy-ethyl)-7-oxo-4-thia-1-az...)
Affinity DataKi:  4.00E+3nM Koff:  170s-1Assay Description:Rate constant for the compound was determined (k2/ki) against human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeutrophil elastase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50281009([(5R,6S)-6-((R)-1-Hydroxy-ethyl)-7-oxo-2,4-dithia-...)
Affinity DataKi:  1.20E+4nMAssay Description:Inhibitory activity against human leukocyte elastase (HLE) was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeutrophil elastase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50281008([(5S,6R)-6-((R)-1-Hydroxy-ethyl)-7-oxo-2,4-dithia-...)
Affinity DataKi: >1.00E+5nMAssay Description:Rate constant for the compound was determined (k2/ki) against human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeutrophil elastase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50281007([(5R,6S)-6-((R)-1-Hydroxy-ethyl)-7-oxo-1-aza-bicyc...)
Affinity DataKi: >1.00E+5nMAssay Description:Rate constant for the compound was determined (k2/ki) against human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeutrophil elastase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50281009([(5R,6S)-6-((R)-1-Hydroxy-ethyl)-7-oxo-2,4-dithia-...)
Affinity DataKon:  0.00200M-1s-1Assay Description:Rate constant for the compound was determined (k2/ki) against human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeutrophil elastase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50281003([(5R,6S)-6-((R)-1-Hydroxy-ethyl)-7-oxo-4-thia-1-az...)
Affinity DataKon:  0.000670M-1s-1Assay Description:Rate constant for the compound was determined against human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeutrophil elastase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50281005([(5R,6S)-7-Oxo-6-((R)-1-phenylacetoxy-ethyl)-2,4-d...)
Affinity DataKon:  0.000400M-1s-1Assay Description:Rate constant for the compound was determined (k2/ki) against human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeutrophil elastase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50281003([(5R,6S)-6-((R)-1-Hydroxy-ethyl)-7-oxo-4-thia-1-az...)
Affinity DataKoff:  170s-1Assay Description:Rate constant for the compound was determined (k2/ki) against human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeutrophil elastase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50281009([(5R,6S)-6-((R)-1-Hydroxy-ethyl)-7-oxo-2,4-dithia-...)
Affinity DataKoff:  150s-1Assay Description:Rate constant for the compound was determined (k2/ki) against human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeutrophil elastase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50281006([(5R,6S)-6-((R)-1-Hydroxy-ethyl)-7-oxo-2,4-dithia-...)
Affinity DataKon:  0.00140M-1s-1Assay Description:Rate constant for the compound was determined against human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeutrophil elastase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50281004([(5R,6S)-6-((R)-1-Hydroxy-ethyl)-7-oxo-2-thia-1-az...)
Affinity DataKoff:  130s-1Assay Description:Rate constant for the compound was determined (k2/ki) against human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeutrophil elastase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50281006([(5R,6S)-6-((R)-1-Hydroxy-ethyl)-7-oxo-2,4-dithia-...)
Affinity DataKoff:  1.00E+3s-1Assay Description:Rate constant for the compound was determined (k2/ki) against human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeutrophil elastase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50281005([(5R,6S)-7-Oxo-6-((R)-1-phenylacetoxy-ethyl)-2,4-d...)
Affinity DataKoff:  970s-1Assay Description:Rate constant for the compound was determined (k2/ki) against human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeutrophil elastase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50281004([(5R,6S)-6-((R)-1-Hydroxy-ethyl)-7-oxo-2-thia-1-az...)
Affinity DataKon:  0.000400M-1s-1Assay Description:Rate constant for the compound was determined against human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article